Names
Compounds (1,424)
Reactome (2)
Related By:
Pathway (2)
Organism (2)
Gene (1)
Org. Clust. (4)
ChEMBL (32)
Rings (49)

Cannabinoid CB1 Receptor, Rat (1,424 Compounds)

Swissprot:: CNR1_RAT
Stitch:: CNR1_RAT
UniProt:: P20272
ChEMBL:: CHEMBL3571
Reactome:: REACT_262979; REACT_233455
PDB:: Cnr1

Compound Summary

Annotation Type	Substances	Purchasable	Natural	In Man
Binding ≤ 10μM	1,424	89	26	10
Binding ≤ 1μM	1,252	73	19	8
Functional ≤ 10μM	45	8	3	2

Reactome ID	Description	Species
REACT_262979	Class A/1 (Rhodopsin-like receptors)	Rattus norvegicus
REACT_233455	G alpha (i) signalling events	Rattus norvegicus

Uniprot	Swissprot	Chembl	Description	Number Shared
CNR2_RAT	Q9QZN9	CHEMBL2470	Cannabinoid CB2 Receptor, Rat	113

G alpha (i) signalling events

Uniprot	Swissprot	Chembl	Description	Number Shared
CNR2_RAT	Q9QZN9	CHEMBL2470	Cannabinoid CB2 Receptor, Rat	113

UniProt	Swissprot	ChEMBL	Description	Substances	Purchasable	Natural	In Man
CNR1_HUMAN	P21554	CHEMBL218	Cannabinoid CB1 Receptor, Human	2,791	161	19	12
CNR1_MOUSE	P47746	CHEMBL3037	Cannabinoid CB1 Receptor, Mouse	103	19	5	3

UniProt	Swissprot	ChEMBL	Description	Substances	Purchasable	Natural	In Man
CNR2_RAT	Q9QZN9	CHEMBL2470	Cannabinoid CB2 Receptor, Rat	130	21	8	3

Clustered By Gene (0)

Clustered By Organism (4)

Code	Description	Substances	Purchasable	Natural	In Man
CNR1-1-E	Cannabinoid CB1 Receptor (cluster #1 Of 5), Eukaryotic	3,810	186	15	14
CNR1-2-E	Cannabinoid CB1 Receptor (cluster #2 Of 5), Eukaryotic	68	14	9	3
CNR1-3-E	Cannabinoid CB1 Receptor (cluster #3 Of 5), Eukaryotic	290	38	12	1
CNR1-4-E	Cannabinoid CB1 Receptor (cluster #4 Of 5), Eukaryotic	3	0	0	0
CNR1-5-E	Cannabinoid CB1 Receptor (cluster #5 Of 5), Eukaryotic	18	3	1	1

Uniprot	Swissprot	Chembl	Description	Number Shared
CNR2_HUMAN	P34972	CHEMBL253	Cannabinoid CB2 Receptor, Human	389
CNR2_MOUSE	P47936	CHEMBL5373	Cannabinoid CB2 Receptor, Mouse	216
CNR1_HUMAN	P21554	CHEMBL218	Cannabinoid CB1 Receptor, Human	176
CNR2_RAT	Q9QZN9	CHEMBL2470	Cannabinoid CB2 Receptor, Rat	113
CNR1_MOUSE	P47746	CHEMBL3037	Cannabinoid CB1 Receptor, Mouse	18
FAAH1_HUMAN	O00519	CHEMBL2243	Anandamide Amidohydrolase, Human	11
FAAH1_RAT	P97612	CHEMBL3229	Anandamide Amidohydrolase, Rat	6
FAAH1_MOUSE	O08914	CHEMBL3455	Anandamide Amidohydrolase, Mouse	5
KCNH2_HUMAN	Q12809	CHEMBL240	HERG, Human	5
Z50594	Z50594	CHEMBL375	Mus Musculus	5
ADCY5_RAT	Q04400	CHEMBL2880	Adenylate Cyclase Type V, Rat	4
PTGDS_MOUSE	O09114	CHEMBL4334	Prostaglandin-H2 D-isomerase, Mouse	4
MGLL_MOUSE	O35678	CHEMBL5774	Monoglyceride Lipase, Mouse	3
ACES_MOUSE	P21836	CHEMBL3198	Acetylcholinesterase, Mouse	2
MGLL_HUMAN	Q99685	CHEMBL4191	Monoglyceride Lipase, Human	2
PA24A_HUMAN	P47712	CHEMBL3816	Cytosolic Phospholipase A2, Human	2
Z104302	Z104302	CHEMBL1907608	Glutamate NMDA Receptor	2
Z50425	Z50425	CHEMBL364	Plasmodium Falciparum	2
Z50597	Z50597	CHEMBL376	Rattus Norvegicus	2
ABD12_HUMAN	Q8N2K0	CHEMBL5516	Monoacylglycerol Lipase ABHD12, Human	1
ABHGA_HUMAN	O95870	CHEMBL6168	Protein BAT5, Human	1
DGLA_HUMAN	Q9Y4D2	CHEMBL5545	Sn1-specific Diacylglycerol Lipase Alpha, Human	1
DGLB_HUMAN	Q8NCG7	CHEMBL5521	Sn1-specific Diacylglycerol Lipase Beta, Human	1
GPR55_HUMAN	Q9Y2T6	CHEMBL1075322	G-protein Coupled Receptor 55, Human	1
LIPP_PIG	P00591	CHEMBL1687677	Pancreatic Triacylglycerol Lipase, Pig	1
NR1I2_HUMAN	O75469	CHEMBL3401	Pregnane X Receptor, Human	1
PAFA_HUMAN	Q13093	CHEMBL3514	LDL-associated Phospholipase A2, Human	1
PPARA_HUMAN	Q07869	CHEMBL239	Peroxisome Proliferator-activated Receptor Alpha, Human	1
TRPA1_RAT	Q6RI86	CHEMBL5160	Transient Receptor Potential Cation Channel Subfamily A Member 1, Rat	1
TRPV1_HUMAN	Q8NER1	CHEMBL4794	Vanilloid Receptor, Human	1
TRPV1_RAT	O35433	CHEMBL5102	Vanilloid Receptor, Rat	1
Z50512	Z50512	CHEMBL369	Cavia Porcellus	1