UCSF

Cyclin A1, Human (597 Compounds)

Swissprot:
CCNA1_HUMAN
Stitch:
CCNA1_HUMAN
UniProt:
P78396
ChEMBL:
CHEMBL3609
Reactome:
REACT_1857
REACT_9029
REACT_169185
REACT_471
REACT_111214
REACT_683
REACT_1915
REACT_1156
REACT_6362
REACT_6837
REACT_9003
REACT_169168
PDB:
CCNA1

Compound Summary

Annotation Type Substances Purchasable Natural In Man
Binding ≤ 10μM 597 21 4 15
Binding ≤ 1μM 438 15 2 11
Uniprot Swissprot Chembl Description Number Shared
CCNA2_HUMAN P20248 CHEMBL2582 Cyclin A2, Human 539
CCNB1_HUMAN P14635 CHEMBL2412 G2/mitotic-specific Cyclin B1, Human 72
CCNB2_HUMAN O95067 CHEMBL3723 G2/mitotic-specific Cyclin B2, Human 72
CCNH_HUMAN P51946 CHEMBL2165 Cyclin H, Human 3
CDK1_HUMAN P06493 CHEMBL308 Cyclin-dependent Kinase 1, Human 78
CDK2_HUMAN P24941 CHEMBL301 Cyclin-dependent Kinase 2, Human 566
CDK7_HUMAN P50613 CHEMBL3055 Cyclin-dependent Kinase 7, Human 4
MAT1_HUMAN P51948 CHEMBL5053 CDK-activating Kinase Assembly Factor MAT1, Human 1
PLK1_HUMAN P53350 CHEMBL3024 Serine/threonine-protein Kinase PLK1, Human 12
WEE1_HUMAN P30291 CHEMBL5491 Serine/threonine-protein Kinase WEE1, Human 1

Cyclin A:Cdk2-associated events at S phase entry

Uniprot Swissprot Chembl Description Number Shared
CCNA2_HUMAN P20248 CHEMBL2582 Cyclin A2, Human 539
CCNH_HUMAN P51946 CHEMBL2165 Cyclin H, Human 3
CDK2_HUMAN P24941 CHEMBL301 Cyclin-dependent Kinase 2, Human 566
CDK7_HUMAN P50613 CHEMBL3055 Cyclin-dependent Kinase 7, Human 4
MAT1_HUMAN P51948 CHEMBL5053 CDK-activating Kinase Assembly Factor MAT1, Human 1
WEE1_HUMAN P30291 CHEMBL5491 Serine/threonine-protein Kinase WEE1, Human 1

DNA Damage/Telomere Stress Induced Senescence

Uniprot Swissprot Chembl Description Number Shared
CCNA2_HUMAN P20248 CHEMBL2582 Cyclin A2, Human 539
CCNE1_HUMAN P24864 CHEMBL3617 G1/S-specific Cyclin E1, Human 114
CCNE2_HUMAN O96020 CHEMBL2884 G1/S-specific Cyclin E2, Human 114
CDK2_HUMAN P24941 CHEMBL301 Cyclin-dependent Kinase 2, Human 566

E2F mediated regulation of DNA replication

Uniprot Swissprot Chembl Description Number Shared
CCNE1_HUMAN P24864 CHEMBL3617 G1/S-specific Cyclin E1, Human 114
CDK1_HUMAN P06493 CHEMBL308 Cyclin-dependent Kinase 1, Human 78

G0 and Early G1

Uniprot Swissprot Chembl Description Number Shared
CCNA2_HUMAN P20248 CHEMBL2582 Cyclin A2, Human 539
CCNE1_HUMAN P24864 CHEMBL3617 G1/S-specific Cyclin E1, Human 114
CCNE2_HUMAN O96020 CHEMBL2884 G1/S-specific Cyclin E2, Human 114
CDK1_HUMAN P06493 CHEMBL308 Cyclin-dependent Kinase 1, Human 78
CDK2_HUMAN P24941 CHEMBL301 Cyclin-dependent Kinase 2, Human 566
DYR1A_HUMAN Q13627 CHEMBL2292 Dual-specificity Tyrosine-phosphorylation Regulated Kinase 1A, Human 2

G1/S-Specific Transcription

Uniprot Swissprot Chembl Description Number Shared
CCNE1_HUMAN P24864 CHEMBL3617 G1/S-specific Cyclin E1, Human 114
CDK1_HUMAN P06493 CHEMBL308 Cyclin-dependent Kinase 1, Human 78

G2 Phase

Uniprot Swissprot Chembl Description Number Shared
CCNA2_HUMAN P20248 CHEMBL2582 Cyclin A2, Human 539
CDK2_HUMAN P24941 CHEMBL301 Cyclin-dependent Kinase 2, Human 566

Orc1 removal from chromatin

Uniprot Swissprot Chembl Description Number Shared
CCNA2_HUMAN P20248 CHEMBL2582 Cyclin A2, Human 539
CDK2_HUMAN P24941 CHEMBL301 Cyclin-dependent Kinase 2, Human 566

Phosphorylation of proteins involved in the G2/M transition by Cyclin A:Cdc2 com

Uniprot Swissprot Chembl Description Number Shared
CCNA2_HUMAN P20248 CHEMBL2582 Cyclin A2, Human 539
CDK1_HUMAN P06493 CHEMBL308 Cyclin-dependent Kinase 1, Human 78

Regulation of APC/C activators between G1/S and early anaphase

Uniprot Swissprot Chembl Description Number Shared
CCNA2_HUMAN P20248 CHEMBL2582 Cyclin A2, Human 539
CCNB1_HUMAN P14635 CHEMBL2412 G2/mitotic-specific Cyclin B1, Human 72
CDK1_HUMAN P06493 CHEMBL308 Cyclin-dependent Kinase 1, Human 78
CDK2_HUMAN P24941 CHEMBL301 Cyclin-dependent Kinase 2, Human 566

SCF(Skp2)-mediated degradation of p27/p21

Uniprot Swissprot Chembl Description Number Shared
CCNA2_HUMAN P20248 CHEMBL2582 Cyclin A2, Human 539
CCNE1_HUMAN P24864 CHEMBL3617 G1/S-specific Cyclin E1, Human 114
CCNE2_HUMAN O96020 CHEMBL2884 G1/S-specific Cyclin E2, Human 114
CDK2_HUMAN P24941 CHEMBL301 Cyclin-dependent Kinase 2, Human 566

Senescence-Associated Secretory Phenotype (SASP)

Uniprot Swissprot Chembl Description Number Shared
CCNA2_HUMAN P20248 CHEMBL2582 Cyclin A2, Human 539
CDK2_HUMAN P24941 CHEMBL301 Cyclin-dependent Kinase 2, Human 566
CDK4_HUMAN P11802 CHEMBL331 Cyclin-dependent Kinase 4, Human 49
CDK6_HUMAN Q00534 CHEMBL2508 Cyclin-dependent Kinase 6, Human 5
KS6A1_HUMAN Q15418 CHEMBL2553 Ribosomal Protein S6 Kinase Alpha 1, Human 2
KS6A2_HUMAN Q15349 CHEMBL3906 Ribosomal Protein S6 Kinase Alpha 2, Human 3
KS6A3_HUMAN P51812 CHEMBL2345 Ribosomal Protein S6 Kinase Alpha 3, Human 3
MK01_HUMAN P28482 CHEMBL4040 MAP Kinase ERK2, Human 5
MK03_HUMAN P27361 CHEMBL3385 MAP Kinase ERK1, Human 2
MK07_HUMAN Q13164 CHEMBL5332 Mitogen-activated Protein Kinase 7, Human 2
UniProt Swissprot ChEMBL Description Substances Purchasable Natural In Man
CCNA2_HUMAN P20248 CHEMBL2582 Cyclin A2, Human 650 26 6 23

Clustered By Gene (0)

Clustered By Organism (2)

Code Description Substances Purchasable Natural In Man
CCNA1-1-E Cyclin A1 (cluster #1 Of 3), Eukaryotic 578 20 4 14
CCNA1-2-E Cyclin A1 (cluster #2 Of 3), Eukaryotic 22 0 0 0
CCNA1-3-E Cyclin A1 (cluster #3 Of 3), Eukaryotic 11 1 0 1
Uniprot Swissprot Chembl Description Number Shared
CDK2_HUMAN P24941 CHEMBL301 Cyclin-dependent Kinase 2, Human 566
CCNA2_HUMAN P20248 CHEMBL2582 Cyclin A2, Human 539
CCNE1_HUMAN P24864 CHEMBL3617 G1/S-specific Cyclin E1, Human 114
CCNE2_HUMAN O96020 CHEMBL2884 G1/S-specific Cyclin E2, Human 114
CHK1_HUMAN O14757 CHEMBL4630 Serine/threonine-protein Kinase Chk1, Human 79
CDK1_HUMAN P06493 CHEMBL308 Cyclin-dependent Kinase 1, Human 78
CCNB1_HUMAN P14635 CHEMBL2412 G2/mitotic-specific Cyclin B1, Human 72
CCNB2_HUMAN O95067 CHEMBL3723 G2/mitotic-specific Cyclin B2, Human 72
Z104295 Z104295 CHEMBL1907601 Cyclin-dependent Kinase 4/cyclin D1 57
CDK4_HUMAN P11802 CHEMBL331 Cyclin-dependent Kinase 4, Human 49
Z104296 Z104296 CHEMBL1907602 Cyclin-dependent Kinase 1/cyclin B1 40
CCNB3_HUMAN Q8WWL7 CHEMBL3606 G2/mitotic-specific Cyclin B3, Human 38
CCND2_HUMAN P30279 CHEMBL3613 G1/S-specific Cyclin D2, Human 38
CCND1_HUMAN P24385 CHEMBL3610 G1/S-specific Cyclin D1, Human 34
CCND3_HUMAN P30281 CHEMBL2422 G1/S-specific Cyclin D3, Human 32
GSK3B_HUMAN P49841 CHEMBL262 Glycogen Synthase Kinase-3 Beta, Human 27
Z104299 Z104299 CHEMBL1907605 Cyclin-dependent Kinase 2/cyclin E1 20
Z104294 Z104294 CHEMBL1907600 Cyclin-dependent Kinase 5/CDK5 Activator 1 17
AURKA_HUMAN O14965 CHEMBL4722 Serine/threonine-protein Kinase Aurora-A, Human 13
FGFR2_HUMAN P21802 CHEMBL4142 Fibroblast Growth Factor Receptor 2, Human 12
PLK1_HUMAN P53350 CHEMBL3024 Serine/threonine-protein Kinase PLK1, Human 12
VGFR2_HUMAN P35968 CHEMBL279 Vascular Endothelial Growth Factor Receptor 2, Human 12
FGFR1_HUMAN P11362 CHEMBL3650 Fibroblast Growth Factor Receptor 1, Human 11
GSK3A_HUMAN P49840 CHEMBL2850 Glycogen Synthase Kinase-3 Alpha, Human 11
FGFR3_HUMAN P22607 CHEMBL2742 Fibroblast Growth Factor Receptor 3, Human 10
PLK3_HUMAN Q9H4B4 CHEMBL4897 Serine/threonine-protein Kinase PLK3, Human 10
CDK5_HUMAN Q00535 CHEMBL4036 Cyclin-dependent Kinase 5, Human 9
FGFR4_HUMAN P22455 CHEMBL3973 Fibroblast Growth Factor Receptor 4, Human 9
PLK2_HUMAN Q9NYY3 CHEMBL5938 Serine/threonine-protein Kinase PLK2, Human 9
FAK1_HUMAN Q05397 CHEMBL2695 Focal Adhesion Kinase 1, Human 7
KPCD_HUMAN Q05655 CHEMBL2996 Protein Kinase C Delta, Human 7
PGFRB_HUMAN P09619 CHEMBL1913 Platelet-derived Growth Factor Receptor Beta, Human 7
SRC_HUMAN P12931 CHEMBL267 Tyrosine-protein Kinase SRC, Human 6
CDK6_HUMAN Q00534 CHEMBL2508 Cyclin-dependent Kinase 6, Human 5
GSK3B_RAT P18266 CHEMBL3669 Glycogen Synthase Kinase-3 Beta, Rat 5
KAPCA_HUMAN P17612 CHEMBL4101 CAMP-dependent Protein Kinase Alpha-catalytic Subunit, Human 5
KAPCB_HUMAN P22694 CHEMBL2918 CAMP-dependent Protein Kinase Beta-1 Catalytic Subunit, Human 5
KAPCG_HUMAN P22612 CHEMBL2743 CAMP-dependent Protein Kinase, Gamma Catalytic Subunit, Human 5
KC1E_HUMAN P49674 CHEMBL4937 Casein Kinase I Epsilon, Human 5
KC1G1_HUMAN Q9HCP0 CHEMBL2426 Casein Kinase I Gamma 1, Human 5
KC1G2_HUMAN P78368 CHEMBL2543 Casein Kinase I Gamma 2, Human 5
KPCB_HUMAN P05771 CHEMBL3045 Protein Kinase C Beta, Human 5
MK01_HUMAN P28482 CHEMBL4040 MAP Kinase ERK2, Human 5
MK10_HUMAN P53779 CHEMBL2637 C-Jun N-terminal Kinase 3, Human 5
NTRK1_HUMAN P04629 CHEMBL2815 Nerve Growth Factor Receptor Trk-A, Human 5
CDK7_HUMAN P50613 CHEMBL3055 Cyclin-dependent Kinase 7, Human 4
CDK9_HUMAN P50750 CHEMBL3116 Cyclin-dependent Kinase 9, Human 4
E2AK2_HUMAN P19525 CHEMBL5785 Interferon-induced, Double-stranded RNA-activated Protein Kinase, Human 4
EGFR_HUMAN P00533 CHEMBL203 Epidermal Growth Factor Receptor ErbB1, Human 4
FLT3_HUMAN P36888 CHEMBL1974 Tyrosine-protein Kinase Receptor FLT3, Human 4
INSR_HUMAN P06213 CHEMBL1981 Insulin Receptor, Human 4
KC1D_HUMAN P48730 CHEMBL2828 Casein Kinase I Delta, Human 4
MK08_HUMAN P45983 CHEMBL2276 C-Jun N-terminal Kinase 1, Human 4
PLK4_HUMAN O00444 CHEMBL3788 Serine/threonine-protein Kinase PLK4, Human 4
TTK_HUMAN P33981 CHEMBL3983 Dual Specificity Protein Kinase TTK, Human 4
VGFR2_MOUSE P35918 CHEMBL3337 Vascular Endothelial Growth Factor Receptor 2, Mouse 4
ABL1_HUMAN P00519 CHEMBL1862 Tyrosine-protein Kinase ABL, Human 3
ALK_HUMAN Q9UM73 CHEMBL4247 ALK Tyrosine Kinase Receptor, Human 3
CCNB_MARGL P15206 CHEMBL4260 G2/mitotic-specific Cyclin B, Margl 3
CCNH_HUMAN P51946 CHEMBL2165 Cyclin H, Human 3
CDK16_HUMAN Q00536 CHEMBL4597 Serine/threonine-protein Kinase PCTAIRE-1, Human 3
CDK1_YEAST P00546 CHEMBL5213 Cell Division Control Protein 28, Yeast 3
CLK1_HUMAN P49759 CHEMBL4224 Dual Specificty Protein Kinase CLK1, Human 3
CLK2_HUMAN P49760 CHEMBL4225 Dual Specificity Protein Kinase CLK2, Human 3
KC1A_HUMAN P48729 CHEMBL2793 Casein Kinase I Alpha, Human 3
KIT_HUMAN P10721 CHEMBL1936 Stem Cell Growth Factor Receptor, Human 3
KPCA_HUMAN P17252 CHEMBL299 Protein Kinase C Alpha, Human 3
KPCE_HUMAN Q02156 CHEMBL3582 Protein Kinase C Epsilon, Human 3
KPCL_HUMAN P24723 CHEMBL3616 Protein Kinase C Eta, Human 3
KPCT_HUMAN Q04759 CHEMBL3920 Protein Kinase C Theta, Human 3
KPCZ_HUMAN Q05513 CHEMBL3438 Protein Kinase C Zeta, Human 3
KS6A2_HUMAN Q15349 CHEMBL3906 Ribosomal Protein S6 Kinase Alpha 2, Human 3
KS6A3_HUMAN P51812 CHEMBL2345 Ribosomal Protein S6 Kinase Alpha 3, Human 3
MK09_HUMAN P45984 CHEMBL4179 C-Jun N-terminal Kinase 2, Human 3
PAK4_HUMAN O96013 CHEMBL4482 Serine/threonine-protein Kinase PAK 4, Human 3
PGFRA_HUMAN P16234 CHEMBL2007 Platelet-derived Growth Factor Receptor Alpha, Human 3
UFO_HUMAN P30530 CHEMBL4895 Tyrosine-protein Kinase Receptor UFO, Human 3
VGFR1_HUMAN P17948 CHEMBL1868 Vascular Endothelial Growth Factor Receptor 1, Human 3
VGFR3_HUMAN P35916 CHEMBL1955 Vascular Endothelial Growth Factor Receptor 3, Human 3
Z104300 Z104300 CHEMBL1907606 Mitogen-activated Protein Kinase; ERK1/ERK2 3
AAK1_HUMAN Q2M2I8 CHEMBL3830 Adaptor-associated Kinase, Human 2
AAPK1_HUMAN Q13131 CHEMBL4045 AMP-activated Protein Kinase, Alpha-1 Subunit, Human 2
ACVR1_HUMAN Q04771 CHEMBL5903 Activin Receptor Type-1, Human 2
AURKB_HUMAN Q96GD4 CHEMBL2185 Serine/threonine-protein Kinase Aurora-B, Human 2
AVR2B_HUMAN Q13705 CHEMBL5466 Activin Receptor Type-2B, Human 2
CCNT1_HUMAN O60563 CHEMBL2108 Cyclin T1, Human 2
CCNT2_HUMAN O60583 CHEMBL1293321 Cyclin-T2, Human 2
CDC7_HUMAN O00311 CHEMBL5443 Cell Division Cycle 7-related Protein Kinase, Human 2
CDK14_HUMAN O94921 CHEMBL6162 Serine/threonine-protein Kinase PFTAIRE-1, Human 2
CDK17_HUMAN Q00537 CHEMBL5790 Serine/threonine-protein Kinase PCTAIRE-2, Human 2
CDK18_HUMAN Q07002 CHEMBL5316 Serine/threonine-protein Kinase PCTAIRE-3, Human 2
CDK3_HUMAN Q00526 CHEMBL4442 Cyclin-dependent Kinase 3, Human 2
CLK3_HUMAN P49761 CHEMBL4226 Dual Specificity Protein Kinase CLK3, Human 2
CLK4_HUMAN Q9HAZ1 CHEMBL4203 Dual Specificity Protein Kinase CLK4, Human 2
CSF1R_HUMAN P07333 CHEMBL1844 Macrophage Colony Stimulating Factor Receptor, Human 2
CSK22_HUMAN P19784 CHEMBL4070 Casein Kinase II Alpha (prime), Human 2
DCLK1_HUMAN O15075 CHEMBL5683 Serine/threonine-protein Kinase DCLK1, Human 2
DCLK3_HUMAN Q9C098 CHEMBL6123 Serine/threonine-protein Kinase DCLK3, Human 2
DMPK_HUMAN Q09013 CHEMBL5320 Myotonin-protein Kinase, Human 2
DYR1A_HUMAN Q13627 CHEMBL2292 Dual-specificity Tyrosine-phosphorylation Regulated Kinase 1A, Human 2
DYR1B_HUMAN Q9Y463 CHEMBL5543 Dual Specificity Tyrosine-phosphorylation-regulated Kinase 1B, Human 2
FGFR1_MOUSE P16092 CHEMBL3960 Fibroblast Growth Factor Receptor 1, Mouse 2
GAK_HUMAN O14976 CHEMBL4355 Serine/threonine-protein Kinase GAK, Human 2
IKKB_HUMAN O14920 CHEMBL1991 Inhibitor Of Nuclear Factor Kappa B Kinase Beta Subunit, Human 2
IKKE_HUMAN Q14164 CHEMBL3529 Inhibitor Of Nuclear Factor Kappa B Kinase Epsilon Subunit, Human 2
JAK1_HUMAN P23458 CHEMBL2835 Tyrosine-protein Kinase JAK1, Human 2
JAK2_HUMAN O60674 CHEMBL2971 Tyrosine-protein Kinase JAK2, Human 2
JAK3_HUMAN P52333 CHEMBL2148 Tyrosine-protein Kinase JAK3, Human 2
KC1G3_HUMAN Q9Y6M4 CHEMBL5084 Casein Kinase I Isoform Gamma-3, Human 2
KCC2A_HUMAN Q9UQM7 CHEMBL4147 CaM Kinase II Alpha, Human 2
KCC2B_HUMAN Q13554 CHEMBL4121 CaM Kinase II Beta, Human 2
KKCC1_HUMAN Q8N5S9 CHEMBL5256 CaM-kinase Kinase Alpha, Human 2
KKCC2_HUMAN Q96RR4 CHEMBL5284 CaM-kinase Kinase Beta, Human 2
KPCD1_HUMAN Q15139 CHEMBL3863 Protein Kinase C Mu, Human 2
KPCD3_HUMAN O94806 CHEMBL2595 Protein Kinase C Nu, Human 2
KPCG_HUMAN P05129 CHEMBL2938 Protein Kinase C Gamma, Human 2
KS6A1_HUMAN Q15418 CHEMBL2553 Ribosomal Protein S6 Kinase Alpha 1, Human 2
KS6A4_HUMAN O75676 CHEMBL3125 Ribosomal Protein S6 Kinase Alpha 4, Human 2
KS6A5_HUMAN O75582 CHEMBL4237 Ribosomal Protein S6 Kinase Alpha 5, Human 2
M3K9_HUMAN P80192 CHEMBL2872 Mitogen-activated Protein Kinase Kinase Kinase 9, Human 2
M4K1_HUMAN Q92918 CHEMBL5749 Mitogen-activated Protein Kinase Kinase Kinase Kinase 1, Human 2
M4K3_HUMAN Q8IVH8 CHEMBL5432 Mitogen-activated Protein Kinase Kinase Kinase Kinase 3, Human 2
MERTK_HUMAN Q12866 CHEMBL5331 Proto-oncogene Tyrosine-protein Kinase MER, Human 2
MK03_HUMAN P27361 CHEMBL3385 MAP Kinase ERK1, Human 2
MK07_HUMAN Q13164 CHEMBL5332 Mitogen-activated Protein Kinase 7, Human 2
MK15_HUMAN Q8TD08 CHEMBL5198 Mitogen-activated Protein Kinase 15, Human 2
MP2K1_HUMAN Q02750 CHEMBL3587 Dual Specificity Mitogen-activated Protein Kinase Kinase 1, Human 2
MP2K6_HUMAN P52564 CHEMBL2171 Dual Specificity Mitogen-activated Protein Kinase Kinase 6, Human 2
NUAK2_HUMAN Q9H093 CHEMBL5698 NUAK Family SNF1-like Kinase 2, Human 2
PDPK1_HUMAN O15530 CHEMBL2534 3-phosphoinositide Dependent Protein Kinase-1, Human 2
PGFRA_RAT P20786 CHEMBL2513 Platelet-derived Growth Factor Receptor Alpha, Rat 2
PHKG1_HUMAN Q16816 CHEMBL4004 Phosphorylase Kinase Gamma Subunit 1, Human 2
PHKG2_HUMAN P15735 CHEMBL2349 Phosphorylase Kinase Gamma Subunit 2, Human 2
PIM1_HUMAN P11309 CHEMBL2147 Serine/threonine-protein Kinase PIM1, Human 2
PIM3_HUMAN Q86V86 CHEMBL5407 Serine/threonine-protein Kinase PIM3, Human 2
Q17066_ASTPE Q17066 CHEMBL5124 Cdc2, Astpe 2
Q95J97_RABIT Q95J97 CHEMBL4885 CAMP-dependent Protein Kinase Alpha-catalytic Subunit, Rabit 2
SGK1_HUMAN O00141 CHEMBL2343 Serine/threonine-protein Kinase Sgk1, Human 2
STK3_HUMAN Q13188 CHEMBL4708 Serine/threonine-protein Kinase MST2, Human 2
TIE2_HUMAN Q02763 CHEMBL4128 Tyrosine-protein Kinase TIE-2, Human 2
TNI3K_HUMAN Q59H18 CHEMBL5260 Serine/threonine-protein Kinase TNNI3K, Human 2
AAPK2_HUMAN P54646 CHEMBL2116 AMP-activated Protein Kinase, Alpha-2 Subunit, Human 1
ACVL1_HUMAN P37023 CHEMBL5311 Serine/threonine-protein Kinase Receptor R3, Human 1
ADCK3_HUMAN Q8NI60 CHEMBL5550 Chaperone Activity Of Bc1 Complex-like, Mitochondrial, Human 1
ANKK1_HUMAN Q8NFD2 CHEMBL5547 Ankyrin Repeat And Protein Kinase Domain-containing Protein 1, Human 1
AURKC_HUMAN Q9UQB9 CHEMBL3935 Serine/threonine-protein Kinase Aurora-C, Human 1
AVR2A_HUMAN P27037 CHEMBL5616 Activin Receptor Type-2A, Human 1
BLK_HUMAN P51451 CHEMBL2250 Tyrosine-protein Kinase BLK, Human 1
BMP2K_HUMAN Q9NSY1 CHEMBL4522 BMP-2-inducible Protein Kinase, Human 1
BMPR2_HUMAN Q13873 CHEMBL5467 Bone Morphogenetic Protein Receptor Type-2, Human 1
BMX_HUMAN P51813 CHEMBL3834 Tyrosine-protein Kinase BMX, Human 1
BRSK1_HUMAN Q8TDC3 CHEMBL5650 BR Serine/threonine-protein Kinase 1, Human 1
BRSK2_HUMAN Q8IWQ3 CHEMBL4574 BR Serine/threonine-protein Kinase 2, Human 1
CD11A_HUMAN Q9UQ88 CHEMBL5416 PITSLRE Serine/threonine-protein Kinase CDC2L2, Human 1
CD11B_HUMAN P21127 CHEMBL5808 PITSLRE Serine/threonine-protein Kinase CDC2L1, Human 1
CD5R1_HUMAN Q15078 CHEMBL2783 Cyclin-dependent Kinase 5 Regulatory Subunit 1, Human 1
CDK19_HUMAN Q9BWU1 CHEMBL6002 Cell Division Cycle 2-like Protein Kinase 6, Human 1
CDK8_HUMAN P49336 CHEMBL5719 Cell Division Protein Kinase 8, Human 1
CFTR_HUMAN P13569 CHEMBL4051 Cystic Fibrosis Transmembrane Conductance Regulator, Human 1
CSK21_HUMAN P68400 CHEMBL3629 Casein Kinase II Alpha, Human 1
CSK2B_HUMAN P67870 CHEMBL2358 Casein Kinase II Beta, Human 1
CTRO_HUMAN O14578 CHEMBL5579 Citron Rho-interacting Kinase, Human 1
DAPK3_HUMAN O43293 CHEMBL2468 Death-associated Protein Kinase 3, Human 1
DCLK2_HUMAN Q8N568 CHEMBL5519 Serine/threonine-protein Kinase DCLK2, Human 1
DYR1A_MOUSE Q61214 CHEMBL4750 Dual-specificity Tyrosine-phosphorylation Regulated Kinase 1A, Mouse 1
DYRK2_HUMAN Q92630 CHEMBL4376 Dual-specificity Tyrosine-phosphorylation Regulated Kinase 2, Human 1
E2AK4_HUMAN Q9P2K8 CHEMBL5358 Eukaryotic Translation Initiation Factor 2-alpha Kinase 4, Human 1
EPHA2_HUMAN P29317 CHEMBL2068 Ephrin Type-A Receptor 2, Human 1
EPHA3_HUMAN P29320 CHEMBL4954 Ephrin Type-A Receptor 3, Human 1
EPHA5_HUMAN P54756 CHEMBL3987 Ephrin Type-A Receptor 5, Human 1
EPHA7_HUMAN Q15375 CHEMBL4602 Ephrin Type-A Receptor 7, Human 1
EPHB1_HUMAN P54762 CHEMBL5072 Ephrin Type-B Receptor 1, Human 1
EPHB4_HUMAN P54760 CHEMBL5147 Ephrin Type-B Receptor 4, Human 1
FGR_HUMAN P09769 CHEMBL4454 Tyrosine-protein Kinase FGR, Human 1
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 1
IGF1R_HUMAN P08069 CHEMBL1957 Insulin-like Growth Factor I Receptor, Human 1
IRAK3_HUMAN Q9Y616 CHEMBL5081 Interleukin-1 Receptor-associated Kinase 3, Human 1
ITK_HUMAN Q08881 CHEMBL2959 Tyrosine-protein Kinase ITK/TSK, Human 1
KAP2_BOVIN P00515 CHEMBL3654 CAMP-dependent Protein Kinase Type II-alpha Regulatory Subunit, Bovin 1
KCC2D_HUMAN Q13557 CHEMBL2801 CaM Kinase II Delta, Human 1
KCC2G_HUMAN Q13555 CHEMBL3829 CaM Kinase II Gamma, Human 1
KCC4_HUMAN Q16566 CHEMBL2494 CaM Kinase IV, Human 1
KGP1_HUMAN Q13976 CHEMBL4273 CGMP-dependent Protein Kinase 1 Beta, Human 1
KGP2_HUMAN Q13237 CHEMBL2896 CGMP-dependent Protein Kinase 2, Human 1
KPBB_HUMAN Q93100 CHEMBL3844 Phosphorylase Kinase Beta Subunit, Human 1
KPCD2_HUMAN Q9BZL6 CHEMBL4900 Serine/threonine-protein Kinase D2, Human 1
KPCI_HUMAN P41743 CHEMBL2598 Protein Kinase C Iota, Human 1
KS6A6_HUMAN Q9UK32 CHEMBL4924 Ribosomal Protein S6 Kinase Alpha 6, Human 1
KSYK_HUMAN P43405 CHEMBL2599 Tyrosine-protein Kinase SYK, Human 1
LCK_HUMAN P06239 CHEMBL258 Tyrosine-protein Kinase LCK, Human 1
LIMK1_HUMAN P53667 CHEMBL3836 LIM Domain Kinase 1, Human 1
LIMK2_HUMAN P53671 CHEMBL5932 LIM Domain Kinase 2, Human 1
LTK_HUMAN P29376 CHEMBL5627 Leukocyte Tyrosine Kinase Receptor, Human 1
LYN_HUMAN P07948 CHEMBL3905 Tyrosine-protein Kinase Lyn, Human 1
M3K10_HUMAN Q02779 CHEMBL2873 Mitogen-activated Protein Kinase Kinase Kinase 10, Human 1
M4K5_HUMAN Q9Y4K4 CHEMBL4852 Mitogen-activated Protein Kinase Kinase Kinase Kinase 5, Human 1
MARK1_HUMAN Q9P0L2 CHEMBL5940 Serine/threonine-protein Kinase MARK1, Human 1
MARK2_HUMAN Q7KZI7 CHEMBL3831 MAP/microtubule Affinity-regulating Kinase 2, Human 1
MARK3_HUMAN P27448 CHEMBL5600 Serine/threonine-protein Kinase C-TAK1, Human 1
MARK4_HUMAN Q96L34 CHEMBL5754 MAP/microtubule Affinity-regulating Kinase 4, Human 1
MAT1_HUMAN P51948 CHEMBL5053 CDK-activating Kinase Assembly Factor MAT1, Human 1
MET_HUMAN P08581 CHEMBL3717 Hepatocyte Growth Factor Receptor, Human 1
MK04_HUMAN P31152 CHEMBL5759 Mitogen-activated Protein Kinase 4, Human 1
MK06_HUMAN Q16659 CHEMBL5121 Mitogen-activated Protein Kinase 6, Human 1
MK10_RAT P49187 CHEMBL4092 C-Jun N-terminal Kinase 3, Rat 1
MK14_HUMAN Q16539 CHEMBL260 MAP Kinase P38 Alpha, Human 1
MKNK2_HUMAN Q9HBH9 CHEMBL4204 MAP Kinase Signal-integrating Kinase 2, Human 1
MP2K2_HUMAN P36507 CHEMBL2964 Dual Specificity Mitogen-activated Protein Kinase Kinase 2, Human 1
MP2K3_HUMAN P46734 CHEMBL2109 Dual Specificity Mitogen-activated Protein Kinase Kinase 3, Human 1
MP2K4_HUMAN P45985 CHEMBL2897 Dual Specificity Mitogen-activated Protein Kinase Kinase 4, Human 1
MRCKA_HUMAN Q5VT25 CHEMBL4516 Serine/threonine-protein Kinase MRCK-A, Human 1
MRCKB_HUMAN Q9Y5S2 CHEMBL5052 Serine/threonine-protein Kinase MRCK Beta, Human 1
MST4_HUMAN Q9P289 CHEMBL5941 Serine/threonine-protein Kinase MST4, Human 1
MYLK_HUMAN Q15746 CHEMBL2428 Myosin Light Chain Kinase, Smooth Muscle, Human 1
NEK2_HUMAN P51955 CHEMBL3835 Serine/threonine-protein Kinase NEK2, Human 1
NUAK1_HUMAN O60285 CHEMBL5784 NUAK Family SNF1-like Kinase 1, Human 1
PAK3_HUMAN O75914 CHEMBL2999 Serine/threonine-protein Kinase PAK 3, Human 1
PAK6_HUMAN Q9NQU5 CHEMBL4311 Serine/threonine-protein Kinase PAK6, Human 1
PAK7_HUMAN Q9P286 CHEMBL4524 Serine/threonine-protein Kinase PAK7, Human 1
PDK1_HUMAN Q15118 CHEMBL4766 Pyruvate Dehydrogenase Kinase Isoform 1, Human 1
PI42B_HUMAN P78356 CHEMBL5667 Phosphatidylinositol-5-phosphate 4-kinase Type-2 Beta, Human 1
PI51A_HUMAN Q99755 CHEMBL5969 Phosphatidylinositol-4-phosphate 5-kinase Type-1 Alpha, Human 1
PIM2_HUMAN Q9P1W9 CHEMBL4523 Serine/threonine-protein Kinase PIM2, Human 1
PKN1_HUMAN Q16512 CHEMBL3384 Protein Kinase N1, Human 1
PKN2_HUMAN Q16513 CHEMBL3032 Protein Kinase N2, Human 1
PYGM_HUMAN P11217 CHEMBL3526 Muscle Glycogen Phosphorylase, Human 1
Q8MMZ8_EIMTE Q8MMZ8 CHEMBL5036 CGMP-dependent Protein Kinase, Eimte 1
RAF1_HUMAN P04049 CHEMBL1906 Serine/threonine-protein Kinase RAF, Human 1
RET_HUMAN P07949 CHEMBL2041 Tyrosine-protein Kinase Receptor RET, Human 1
RIOK1_HUMAN Q9BRS2 CHEMBL5975 Serine/threonine-protein Kinase RIO1, Human 1
RIOK3_HUMAN O14730 CHEMBL5659 Serine/threonine-protein Kinase RIO3, Human 1
RIPK1_HUMAN Q13546 CHEMBL5464 Receptor-interacting Serine/threonine-protein Kinase 1, Human 1
ROCK2_HUMAN O75116 CHEMBL2973 Rho-associated Protein Kinase 2, Human 1
SIK1_HUMAN P57059 CHEMBL6082 Serine/threonine-protein Kinase SIK1, Human 1
SIK2_HUMAN Q9H0K1 CHEMBL5699 Serine/threonine-protein Kinase SIK2, Human 1
SLK_HUMAN Q9H2G2 CHEMBL4202 Serine/threonine-protein Kinase 2, Human 1
SRMS_HUMAN Q9H3Y6 CHEMBL5703 Tyrosine-protein Kinase Srms, Human 1
SRPK1_HUMAN Q96SB4 CHEMBL4375 Serine/threonine-protein Kinase SRPK1, Human 1
ST17A_HUMAN Q9UEE5 CHEMBL4525 Serine/threonine-protein Kinase 17A, Human 1
ST17B_HUMAN O94768 CHEMBL3980 Serine/threonine-protein Kinase 17B, Human 1
STK10_HUMAN O94804 CHEMBL3981 Serine/threonine-protein Kinase 10, Human 1
STK16_HUMAN O75716 CHEMBL3938 Serine/threonine-protein Kinase 16, Human 1
STK24_HUMAN Q9Y6E0 CHEMBL5082 Serine/threonine-protein Kinase 24, Human 1
STK25_HUMAN O00506 CHEMBL5552 Serine/threonine-protein Kinase 25, Human 1
STK33_HUMAN Q9BYT3 CHEMBL6005 Serine/threonine-protein Kinase 33, Human 1
STK4_HUMAN Q13043 CHEMBL4598 Serine/threonine-protein Kinase MST1, Human 1
TAOK1_HUMAN Q7L7X3 CHEMBL5261 Serine/threonine-protein Kinase TAO1, Human 1
TEC_HUMAN P42680 CHEMBL4246 Tyrosine-protein Kinase TEC, Human 1
TESK1_HUMAN Q15569 CHEMBL5604 Dual Specificity Testis-specific Protein Kinase 1, Human 1
TGFR2_HUMAN P37173 CHEMBL4267 TGF-beta Receptor Type II, Human 1
TIE1_HUMAN P35590 CHEMBL5274 Tyrosine-protein Kinase Receptor Tie-1, Human 1
TLK1_HUMAN Q9UKI8 CHEMBL5388 Serine/threonine-protein Kinase Tousled-like 1, Human 1
TLK2_HUMAN Q86UE8 CHEMBL5404 Serine/threonine-protein Kinase Tousled-like 2, Human 1
TYK2_HUMAN P29597 CHEMBL3553 Tyrosine-protein Kinase TYK2, Human 1
WEE1_HUMAN P30291 CHEMBL5491 Serine/threonine-protein Kinase WEE1, Human 1