UCSF

Tyrosine-protein Kinase LCK, Human (1,382 Compounds)

Swissprot:
LCK_HUMAN
Stitch:
LCK_HUMAN
UniProt:
P06239
ChEMBL:
CHEMBL258
Reactome:
REACT_19183
REACT_19358
REACT_19238
REACT_147727
REACT_19405
REACT_147814
REACT_12555
REACT_12623
REACT_1695
REACT_27283
REACT_11068
REACT_11166
REACT_19324
REACT_12519
REACT_12582
REACT_75829
REACT_111225
REACT_111040
REACT_12596
PDB:
1BHF (DOCK)
1BHH (DOCK)
1CWD (DOCK)
1CWE (DOCK)
1FBZ (DOCK)
1H92 (DOCK)
1IJR (DOCK)
1KIK (DOCK)
1LCJ (DOCK)
1LCK (DOCK)
1LKK (DOCK)
1LKL (DOCK)
1Q68 (DOCK)
1Q69 (DOCK)
1QPC (DOCK)
1QPD (DOCK)
1QPE (DOCK)
1QPJ (DOCK)
1X27 (DOCK)
2IIM (DOCK)
2OF2 (DOCK)
2OF4 (DOCK)
2OFU (DOCK)
2OFV (DOCK)
2OG8 (DOCK)
2PL0 (DOCK)
2ZM1 (DOCK)
2ZM4 (DOCK)
2ZYB (DOCK)
3AC1 (DOCK)
3AC2 (DOCK)
3AC3 (DOCK)
3AC4 (DOCK)
3AC5 (DOCK)
3AC8 (DOCK)
3ACJ (DOCK)
3ACK (DOCK)
3AD4 (DOCK)
3AD5 (DOCK)
3AD6 (DOCK)
3B2W (DOCK)
3BRH (DOCK)
3BYM (DOCK)
3BYO (DOCK)
3BYS (DOCK)
3BYU (DOCK)
3KMM (DOCK)
3KXZ (DOCK)
3LCK (DOCK)
3MPM (DOCK)
4D8K (DOCK)
LCK

Compound Summary

Annotation Type Substances Purchasable Natural In Man
Binding ≤ 10μM 1,382 96 26 48
Binding ≤ 1μM 1,107 62 20 35
Functional ≤ 10μM 21 7 0 0
Uniprot Swissprot Chembl Description Number Shared
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 60
LYN_HUMAN P07948 CHEMBL3905 Tyrosine-protein Kinase Lyn, Human 185
YES_HUMAN P07947 CHEMBL2073 Tyrosine-protein Kinase YES, Human 44

CD28 dependent PI3K/Akt signaling

Uniprot Swissprot Chembl Description Number Shared
AKT1_HUMAN P31749 CHEMBL4282 Serine/threonine-protein Kinase AKT, Human 3
AKT2_HUMAN P31751 CHEMBL2431 Serine/threonine-protein Kinase AKT2, Human 3
AKT3_HUMAN Q9Y243 CHEMBL4816 Serine/threonine-protein Kinase AKT3, Human 4
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 60
M3K14_HUMAN Q99558 CHEMBL5888 Mitogen-activated Protein Kinase Kinase Kinase 14, Human 1
M3K8_HUMAN P41279 CHEMBL4899 Mitogen-activated Protein Kinase Kinase Kinase 8, Human 1
P85A_HUMAN P27986 CHEMBL2506 PI3-kinase P85-alpha Subunit, Human 6
P85B_HUMAN O00459 CHEMBL4437 PI3-kinase P85-beta Subunit, Human 5
PDPK1_HUMAN O15530 CHEMBL2534 3-phosphoinositide Dependent Protein Kinase-1, Human 6

CD28 dependent Vav1 pathway

Uniprot Swissprot Chembl Description Number Shared
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 60
PAK1_HUMAN Q13153 CHEMBL4600 Serine/threonine-protein Kinase PAK 1, Human 5
PAK2_HUMAN Q13177 CHEMBL4487 Serine/threonine-protein Kinase PAK 2, Human 2
PAK3_HUMAN O75914 CHEMBL2999 Serine/threonine-protein Kinase PAK 3, Human 6

Constitutive PI3K/AKT Signaling in Cancer

Uniprot Swissprot Chembl Description Number Shared
AKT1_HUMAN P31749 CHEMBL4282 Serine/threonine-protein Kinase AKT, Human 3
AKT2_HUMAN P31751 CHEMBL2431 Serine/threonine-protein Kinase AKT2, Human 3
AKT3_HUMAN Q9Y243 CHEMBL4816 Serine/threonine-protein Kinase AKT3, Human 4
EGFR_HUMAN P00533 CHEMBL203 Epidermal Growth Factor Receptor ErbB1, Human 95
ERBB2_HUMAN P04626 CHEMBL1824 Receptor Protein-tyrosine Kinase ErbB-2, Human 30
FGFR4_HUMAN P22455 CHEMBL3973 Fibroblast Growth Factor Receptor 4, Human 13
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 60
GSK3A_HUMAN P49840 CHEMBL2850 Glycogen Synthase Kinase-3 Alpha, Human 4
GSK3B_HUMAN P49841 CHEMBL262 Glycogen Synthase Kinase-3 Beta, Human 12
IKKA_HUMAN O15111 CHEMBL3476 Inhibitor Of Nuclear Factor Kappa B Kinase Alpha Subunit, Human 5
KIT_HUMAN P10721 CHEMBL1936 Stem Cell Growth Factor Receptor, Human 70
KS6B2_HUMAN Q9UBS0 CHEMBL3111 Ribosomal Protein S6 Kinase 2, Human 1
P85A_HUMAN P27986 CHEMBL2506 PI3-kinase P85-alpha Subunit, Human 6
P85B_HUMAN O00459 CHEMBL4437 PI3-kinase P85-beta Subunit, Human 5
PDPK1_HUMAN O15530 CHEMBL2534 3-phosphoinositide Dependent Protein Kinase-1, Human 6
PGFRA_HUMAN P16234 CHEMBL2007 Platelet-derived Growth Factor Receptor Alpha, Human 39
PGFRB_HUMAN P09619 CHEMBL1913 Platelet-derived Growth Factor Receptor Beta, Human 51

CTLA4 inhibitory signaling

Uniprot Swissprot Chembl Description Number Shared
AKT1_HUMAN P31749 CHEMBL4282 Serine/threonine-protein Kinase AKT, Human 3
AKT2_HUMAN P31751 CHEMBL2431 Serine/threonine-protein Kinase AKT2, Human 3
AKT3_HUMAN Q9Y243 CHEMBL4816 Serine/threonine-protein Kinase AKT3, Human 4
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 60
LYN_HUMAN P07948 CHEMBL3905 Tyrosine-protein Kinase Lyn, Human 185
PDPK1_HUMAN O15530 CHEMBL2534 3-phosphoinositide Dependent Protein Kinase-1, Human 6
YES_HUMAN P07947 CHEMBL2073 Tyrosine-protein Kinase YES, Human 44

DAP12 signaling

Uniprot Swissprot Chembl Description Number Shared
BTK_HUMAN Q06187 CHEMBL5251 Tyrosine-protein Kinase BTK, Human 22
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 60
KSYK_HUMAN P43405 CHEMBL2599 Tyrosine-protein Kinase SYK, Human 19
P85A_HUMAN P27986 CHEMBL2506 PI3-kinase P85-alpha Subunit, Human 6
P85B_HUMAN O00459 CHEMBL4437 PI3-kinase P85-beta Subunit, Human 5
PLCG1_HUMAN P19174 CHEMBL3964 Phospholipase C-gamma-1, Human 1
PLCG2_HUMAN P16885 CHEMBL4100 Phospholipase C-gamma-2, Human 1

Downstream TCR signaling

Uniprot Swissprot Chembl Description Number Shared
IKKA_HUMAN O15111 CHEMBL3476 Inhibitor Of Nuclear Factor Kappa B Kinase Alpha Subunit, Human 5
IKKB_HUMAN O14920 CHEMBL1991 Inhibitor Of Nuclear Factor Kappa B Kinase Beta Subunit, Human 4
KPCT_HUMAN Q04759 CHEMBL3920 Protein Kinase C Theta, Human 20
M3K7_HUMAN O43318 CHEMBL5776 Mitogen-activated Protein Kinase Kinase Kinase 7, Human 4
P85A_HUMAN P27986 CHEMBL2506 PI3-kinase P85-alpha Subunit, Human 6
P85B_HUMAN O00459 CHEMBL4437 PI3-kinase P85-beta Subunit, Human 5
PDPK1_HUMAN O15530 CHEMBL2534 3-phosphoinositide Dependent Protein Kinase-1, Human 6
RIPK2_HUMAN O43353 CHEMBL5014 Serine/threonine-protein Kinase RIPK2, Human 15

Generation of second messenger molecules

Uniprot Swissprot Chembl Description Number Shared
ITK_HUMAN Q08881 CHEMBL2959 Tyrosine-protein Kinase ITK/TSK, Human 14
PAK1_HUMAN Q13153 CHEMBL4600 Serine/threonine-protein Kinase PAK 1, Human 5
PAK2_HUMAN Q13177 CHEMBL4487 Serine/threonine-protein Kinase PAK 2, Human 2
PAK3_HUMAN O75914 CHEMBL2999 Serine/threonine-protein Kinase PAK 3, Human 6
PLCG1_HUMAN P19174 CHEMBL3964 Phospholipase C-gamma-1, Human 1
ZAP70_HUMAN P43403 CHEMBL2803 Tyrosine-protein Kinase ZAP-70, Human 13

GPVI-mediated activation cascade

Uniprot Swissprot Chembl Description Number Shared
AKT1_HUMAN P31749 CHEMBL4282 Serine/threonine-protein Kinase AKT, Human 3
AKT2_HUMAN P31751 CHEMBL2431 Serine/threonine-protein Kinase AKT2, Human 3
AKT3_HUMAN Q9Y243 CHEMBL4816 Serine/threonine-protein Kinase AKT3, Human 4
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 60
KPCZ_HUMAN Q05513 CHEMBL3438 Protein Kinase C Zeta, Human 5
KSYK_HUMAN P43405 CHEMBL2599 Tyrosine-protein Kinase SYK, Human 19
LYN_HUMAN P07948 CHEMBL3905 Tyrosine-protein Kinase Lyn, Human 185
P85A_HUMAN P27986 CHEMBL2506 PI3-kinase P85-alpha Subunit, Human 6
P85B_HUMAN O00459 CHEMBL4437 PI3-kinase P85-beta Subunit, Human 5
PDPK1_HUMAN O15530 CHEMBL2534 3-phosphoinositide Dependent Protein Kinase-1, Human 6
PLCG2_HUMAN P16885 CHEMBL4100 Phospholipase C-gamma-2, Human 1

Interleukin-2 signaling

Uniprot Swissprot Chembl Description Number Shared
FAK2_HUMAN Q14289 CHEMBL5469 Protein Tyrosine Kinase 2 Beta, Human 10
JAK1_HUMAN P23458 CHEMBL2835 Tyrosine-protein Kinase JAK1, Human 6
JAK3_HUMAN P52333 CHEMBL2148 Tyrosine-protein Kinase JAK3, Human 62
KSYK_HUMAN P43405 CHEMBL2599 Tyrosine-protein Kinase SYK, Human 19

Nef and signal transduction

Uniprot Swissprot Chembl Description Number Shared
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 60
HCK_HUMAN P08631 CHEMBL3234 Tyrosine-protein Kinase HCK, Human 103
PAK2_HUMAN Q13177 CHEMBL4487 Serine/threonine-protein Kinase PAK 2, Human 2

PD-1 signaling

Uniprot Swissprot Chembl Description Number Shared
CSK_HUMAN P41240 CHEMBL2634 Tyrosine-protein Kinase CSK, Human 21

PECAM1 interactions

Uniprot Swissprot Chembl Description Number Shared
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 60
LYN_HUMAN P07948 CHEMBL3905 Tyrosine-protein Kinase Lyn, Human 185
PLCG1_HUMAN P19174 CHEMBL3964 Phospholipase C-gamma-1, Human 1
YES_HUMAN P07947 CHEMBL2073 Tyrosine-protein Kinase YES, Human 44

Phosphorylation of CD3 and TCR zeta chains

Uniprot Swissprot Chembl Description Number Shared
CSK_HUMAN P41240 CHEMBL2634 Tyrosine-protein Kinase CSK, Human 21
PTPRC_HUMAN P08575 CHEMBL3243 Leukocyte Common Antigen, Human 1

PIP3 activates AKT signaling

Uniprot Swissprot Chembl Description Number Shared
AKT1_HUMAN P31749 CHEMBL4282 Serine/threonine-protein Kinase AKT, Human 3
AKT2_HUMAN P31751 CHEMBL2431 Serine/threonine-protein Kinase AKT2, Human 3
AKT3_HUMAN Q9Y243 CHEMBL4816 Serine/threonine-protein Kinase AKT3, Human 4
EGFR_HUMAN P00533 CHEMBL203 Epidermal Growth Factor Receptor ErbB1, Human 95
ERBB2_HUMAN P04626 CHEMBL1824 Receptor Protein-tyrosine Kinase ErbB-2, Human 30
FGFR4_HUMAN P22455 CHEMBL3973 Fibroblast Growth Factor Receptor 4, Human 13
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 60
KIT_HUMAN P10721 CHEMBL1936 Stem Cell Growth Factor Receptor, Human 70
P85A_HUMAN P27986 CHEMBL2506 PI3-kinase P85-alpha Subunit, Human 6
P85B_HUMAN O00459 CHEMBL4437 PI3-kinase P85-beta Subunit, Human 5
PDPK1_HUMAN O15530 CHEMBL2534 3-phosphoinositide Dependent Protein Kinase-1, Human 6
PGFRA_HUMAN P16234 CHEMBL2007 Platelet-derived Growth Factor Receptor Alpha, Human 39
PGFRB_HUMAN P09619 CHEMBL1913 Platelet-derived Growth Factor Receptor Beta, Human 51

Regulation of KIT signaling

Uniprot Swissprot Chembl Description Number Shared
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 60
KIT_HUMAN P10721 CHEMBL1936 Stem Cell Growth Factor Receptor, Human 70
KPCA_HUMAN P17252 CHEMBL299 Protein Kinase C Alpha, Human 8
LYN_HUMAN P07948 CHEMBL3905 Tyrosine-protein Kinase Lyn, Human 185
YES_HUMAN P07947 CHEMBL2073 Tyrosine-protein Kinase YES, Human 44

Signaling by SCF-KIT

Uniprot Swissprot Chembl Description Number Shared
CHK1_HUMAN O14757 CHEMBL4630 Serine/threonine-protein Kinase Chk1, Human 14
FER_HUMAN P16591 CHEMBL3982 Tyrosine-protein Kinase FER, Human 9
FES_HUMAN P07332 CHEMBL5455 Tyrosine-protein Kinase FES, Human 8
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 60
JAK2_HUMAN O60674 CHEMBL2971 Tyrosine-protein Kinase JAK2, Human 20
KIT_HUMAN P10721 CHEMBL1936 Stem Cell Growth Factor Receptor, Human 70
KPCA_HUMAN P17252 CHEMBL299 Protein Kinase C Alpha, Human 8
LYN_HUMAN P07948 CHEMBL3905 Tyrosine-protein Kinase Lyn, Human 185
P85A_HUMAN P27986 CHEMBL2506 PI3-kinase P85-alpha Subunit, Human 6
P85B_HUMAN O00459 CHEMBL4437 PI3-kinase P85-beta Subunit, Human 5
TEC_HUMAN P42680 CHEMBL4246 Tyrosine-protein Kinase TEC, Human 5
YES_HUMAN P07947 CHEMBL2073 Tyrosine-protein Kinase YES, Human 44

Translocation of ZAP-70 to Immunological synapse

Uniprot Swissprot Chembl Description Number Shared
ZAP70_HUMAN P43403 CHEMBL2803 Tyrosine-protein Kinase ZAP-70, Human 13
UniProt Swissprot ChEMBL Description Substances Purchasable Natural In Man
LCK_MOUSE P06240 CHEMBL2480 Tyrosine-protein Kinase LCK, Mouse 85 9 1 3

Clustered By Gene (0)

Clustered By Organism (3)

Code Description Substances Purchasable Natural In Man
LCK-1-E Tyrosine-protein Kinase LCK (cluster #1 Of 4), Eukaryotic 1,333 71 18 44
LCK-2-E Tyrosine-protein Kinase LCK (cluster #2 Of 4), Eukaryotic 0 0 0 0
LCK-3-E Tyrosine-protein Kinase LCK (cluster #3 Of 4), Eukaryotic 106 27 7 3
LCK-4-E Tyrosine-protein Kinase LCK (cluster #4 Of 4), Eukaryotic 1 1 1 1
Uniprot Swissprot Chembl Description Number Shared
VGFR2_HUMAN P35968 CHEMBL279 Vascular Endothelial Growth Factor Receptor 2, Human 408
SRC_HUMAN P12931 CHEMBL267 Tyrosine-protein Kinase SRC, Human 307
LYN_HUMAN P07948 CHEMBL3905 Tyrosine-protein Kinase Lyn, Human 185
TIE2_HUMAN Q02763 CHEMBL4128 Tyrosine-protein Kinase TIE-2, Human 165
MK14_HUMAN Q16539 CHEMBL260 MAP Kinase P38 Alpha, Human 142
HCK_HUMAN P08631 CHEMBL3234 Tyrosine-protein Kinase HCK, Human 103
EGFR_HUMAN P00533 CHEMBL203 Epidermal Growth Factor Receptor ErbB1, Human 93
AURKB_HUMAN Q96GD4 CHEMBL2185 Serine/threonine-protein Kinase Aurora-B, Human 70
KIT_HUMAN P10721 CHEMBL1936 Stem Cell Growth Factor Receptor, Human 70
ABL1_HUMAN P00519 CHEMBL1862 Tyrosine-protein Kinase ABL, Human 64
INSR_HUMAN P06213 CHEMBL1981 Insulin Receptor, Human 62
JAK3_HUMAN P52333 CHEMBL2148 Tyrosine-protein Kinase JAK3, Human 62
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein Kinase FYN, Human 60
FGFR1_HUMAN P11362 CHEMBL3650 Fibroblast Growth Factor Receptor 1, Human 56
AURKA_HUMAN O14965 CHEMBL4722 Serine/threonine-protein Kinase Aurora-A, Human 55
PGFRB_HUMAN P09619 CHEMBL1913 Platelet-derived Growth Factor Receptor Beta, Human 50
MET_HUMAN P08581 CHEMBL3717 Hepatocyte Growth Factor Receptor, Human 44
YES_HUMAN P07947 CHEMBL2073 Tyrosine-protein Kinase YES, Human 44
FLT3_HUMAN P36888 CHEMBL1974 Tyrosine-protein Kinase Receptor FLT3, Human 41
ACK1_HUMAN Q07912 CHEMBL4599 Tyrosine Kinase Non-receptor Protein 2, Human 40
VGFR1_HUMAN P17948 CHEMBL1868 Vascular Endothelial Growth Factor Receptor 1, Human 39
PGFRA_HUMAN P16234 CHEMBL2007 Platelet-derived Growth Factor Receptor Alpha, Human 38
LCK_MOUSE P06240 CHEMBL2480 Tyrosine-protein Kinase LCK, Mouse 37
CSF1R_HUMAN P07333 CHEMBL1844 Macrophage Colony Stimulating Factor Receptor, Human 36
PTK6_HUMAN Q13882 CHEMBL4601 Tyrosine-protein Kinase BRK, Human 35
RET_HUMAN P07949 CHEMBL2041 Tyrosine-protein Kinase Receptor RET, Human 35
ERBB2_HUMAN P04626 CHEMBL1824 Receptor Protein-tyrosine Kinase ErbB-2, Human 29
BLK_HUMAN P51451 CHEMBL2250 Tyrosine-protein Kinase BLK, Human 28
VGFR3_HUMAN P35916 CHEMBL1955 Vascular Endothelial Growth Factor Receptor 3, Human 27
EPHB4_HUMAN P54760 CHEMBL5147 Ephrin Type-B Receptor 4, Human 25
FGR_HUMAN P09769 CHEMBL4454 Tyrosine-protein Kinase FGR, Human 24
MK09_HUMAN P45984 CHEMBL4179 C-Jun N-terminal Kinase 2, Human 24
ABL2_HUMAN P42684 CHEMBL4014 Tyrosine-protein Kinase ABL2, Human 23
FGFR2_HUMAN P21802 CHEMBL4142 Fibroblast Growth Factor Receptor 2, Human 23
KHDR1_HUMAN Q07666 CHEMBL1795190 KH Domain-containing, RNA-binding, Signal Transduction-associated Protein 1, Human 23
BTK_HUMAN Q06187 CHEMBL5251 Tyrosine-protein Kinase BTK, Human 22
STK10_HUMAN O94804 CHEMBL3981 Serine/threonine-protein Kinase 10, Human 22
CSK_HUMAN P41240 CHEMBL2634 Tyrosine-protein Kinase CSK, Human 21
EPHA2_HUMAN P29317 CHEMBL2068 Ephrin Type-A Receptor 2, Human 21
FRK_HUMAN P42685 CHEMBL4223 Tyrosine-protein Kinase FRK, Human 21
SLK_HUMAN Q9H2G2 CHEMBL4202 Serine/threonine-protein Kinase 2, Human 21
DDR1_HUMAN Q08345 CHEMBL5319 Epithelial Discoidin Domain-containing Receptor 1, Human 20
JAK2_HUMAN O60674 CHEMBL2971 Tyrosine-protein Kinase JAK2, Human 20
KPCT_HUMAN Q04759 CHEMBL3920 Protein Kinase C Theta, Human 20
ALK_HUMAN Q9UM73 CHEMBL4247 ALK Tyrosine Kinase Receptor, Human 19
CTRO_HUMAN O14578 CHEMBL5579 Citron Rho-interacting Kinase, Human 19
GAK_HUMAN O14976 CHEMBL4355 Serine/threonine-protein Kinase GAK, Human 19
KSYK_HUMAN P43405 CHEMBL2599 Tyrosine-protein Kinase SYK, Human 19
RAF1_HUMAN P04049 CHEMBL1906 Serine/threonine-protein Kinase RAF, Human 19
AURKC_HUMAN Q9UQB9 CHEMBL3935 Serine/threonine-protein Kinase Aurora-C, Human 18
BRAF_HUMAN P15056 CHEMBL5145 Serine/threonine-protein Kinase B-raf, Human 18
EPHA6_HUMAN Q9UF33 CHEMBL4526 Ephrin Type-A Receptor 6, Human 18
KPCD_HUMAN Q05655 CHEMBL2996 Protein Kinase C Delta, Human 17
KS6A1_HUMAN Q15418 CHEMBL2553 Ribosomal Protein S6 Kinase Alpha 1, Human 17
M4K5_HUMAN Q9Y4K4 CHEMBL4852 Mitogen-activated Protein Kinase Kinase Kinase Kinase 5, Human 17
MK10_HUMAN P53779 CHEMBL2637 C-Jun N-terminal Kinase 3, Human 17
NTRK1_HUMAN P04629 CHEMBL2815 Nerve Growth Factor Receptor Trk-A, Human 17
FGFR3_HUMAN P22607 CHEMBL2742 Fibroblast Growth Factor Receptor 3, Human 16
KC1D_HUMAN P48730 CHEMBL2828 Casein Kinase I Delta, Human 16
MKNK1_HUMAN Q9BUB5 CHEMBL4718 MAP Kinase-interacting Serine/threonine-protein Kinase MNK1, Human 16
MP2K1_HUMAN Q02750 CHEMBL3587 Dual Specificity Mitogen-activated Protein Kinase Kinase 1, Human 16
TNIK_HUMAN Q9UKE5 CHEMBL4527 TRAF2- And NCK-interacting Kinase, Human 16
UFO_HUMAN P30530 CHEMBL4895 Tyrosine-protein Kinase Receptor UFO, Human 16
M4K4_HUMAN O95819 CHEMBL6166 Mitogen-activated Protein Kinase Kinase Kinase Kinase 4, Human 15
RIPK2_HUMAN O43353 CHEMBL5014 Serine/threonine-protein Kinase RIPK2, Human 15
CHK1_HUMAN O14757 CHEMBL4630 Serine/threonine-protein Kinase Chk1, Human 14
CSK_MOUSE P41241 CHEMBL2333 Tyrosine-protein Kinase CSK, Mouse 14
DDR2_HUMAN Q16832 CHEMBL5122 Discoidin Domain-containing Receptor 2, Human 14
EPHA3_HUMAN P29320 CHEMBL4954 Ephrin Type-A Receptor 3, Human 14
EPHA8_HUMAN P29322 CHEMBL4134 Ephrin Type-A Receptor 8, Human 14
EPHB1_HUMAN P54762 CHEMBL5072 Ephrin Type-B Receptor 1, Human 14
EPHB2_HUMAN P29323 CHEMBL3290 Ephrin Type-B Receptor 2, Human 14
ITK_HUMAN Q08881 CHEMBL2959 Tyrosine-protein Kinase ITK/TSK, Human 14
KPCB_HUMAN P05771 CHEMBL3045 Protein Kinase C Beta, Human 14
KPCE_HUMAN Q02156 CHEMBL3582 Protein Kinase C Epsilon, Human 14
KPCL_HUMAN P24723 CHEMBL3616 Protein Kinase C Eta, Human 14
MERTK_HUMAN Q12866 CHEMBL5331 Proto-oncogene Tyrosine-protein Kinase MER, Human 14
MLTK_HUMAN Q9NYL2 CHEMBL3886 Mixed Lineage Kinase 7, Human 14
MP2K2_HUMAN P36507 CHEMBL2964 Dual Specificity Mitogen-activated Protein Kinase Kinase 2, Human 14
TIE1_HUMAN P35590 CHEMBL5274 Tyrosine-protein Kinase Receptor Tie-1, Human 14
AAPK2_HUMAN P54646 CHEMBL2116 AMP-activated Protein Kinase, Alpha-2 Subunit, Human 13
CDK2_HUMAN P24941 CHEMBL301 Cyclin-dependent Kinase 2, Human 13
EPHA5_HUMAN P54756 CHEMBL3987 Ephrin Type-A Receptor 5, Human 13
MK11_HUMAN Q15759 CHEMBL3961 MAP Kinase P38 Beta, Human 13
MK12_HUMAN P53778 CHEMBL4674 MAP Kinase P38 Gamma, Human 13
NTRK2_HUMAN Q16620 CHEMBL4898 Neurotrophic Tyrosine Kinase Receptor Type 2, Human 13
PLK4_HUMAN O00444 CHEMBL3788 Serine/threonine-protein Kinase PLK4, Human 13
TNI3K_HUMAN Q59H18 CHEMBL5260 Serine/threonine-protein Kinase TNNI3K, Human 13
TYK2_HUMAN P29597 CHEMBL3553 Tyrosine-protein Kinase TYK2, Human 13
ZAP70_HUMAN P43403 CHEMBL2803 Tyrosine-protein Kinase ZAP-70, Human 13
BMX_HUMAN P51813 CHEMBL3834 Tyrosine-protein Kinase BMX, Human 12
EPHA4_HUMAN P54764 CHEMBL3988 Ephrin Type-A Receptor 4, Human 12
GSK3B_HUMAN P49841 CHEMBL262 Glycogen Synthase Kinase-3 Beta, Human 12
KC1E_HUMAN P49674 CHEMBL4937 Casein Kinase I Epsilon, Human 12
KS6A6_HUMAN Q9UK32 CHEMBL4924 Ribosomal Protein S6 Kinase Alpha 6, Human 12
M4K3_HUMAN Q8IVH8 CHEMBL5432 Mitogen-activated Protein Kinase Kinase Kinase Kinase 3, Human 12
MYLK2_HUMAN Q9H1R3 CHEMBL2777 Myosin Light Chain Kinase 2, Human 12
SIK2_HUMAN Q9H0K1 CHEMBL5699 Serine/threonine-protein Kinase SIK2, Human 12
STK3_HUMAN Q13188 CHEMBL4708 Serine/threonine-protein Kinase MST2, Human 12
TXK_HUMAN P42681 CHEMBL4367 Tyrosine-protein Kinase TXK, Human 12
TYRO3_HUMAN Q06418 CHEMBL5314 Tyrosine-protein Kinase Receptor TYRO3, Human 12
BMP2K_HUMAN Q9NSY1 CHEMBL4522 BMP-2-inducible Protein Kinase, Human 11
CDK16_HUMAN Q00536 CHEMBL4597 Serine/threonine-protein Kinase PCTAIRE-1, Human 11
DAPK3_HUMAN O43293 CHEMBL2468 Death-associated Protein Kinase 3, Human 11
E2AK4_HUMAN Q9P2K8 CHEMBL5358 Eukaryotic Translation Initiation Factor 2-alpha Kinase 4, Human 11
EPHA1_HUMAN P21709 CHEMBL5810 Ephrin Type-A Receptor 1, Human 11
FGFR4_HUMAN P22455 CHEMBL3973 Fibroblast Growth Factor Receptor 4, Human 11
KS6A3_HUMAN P51812 CHEMBL2345 Ribosomal Protein S6 Kinase Alpha 3, Human 11
M3K9_HUMAN P80192 CHEMBL2872 Mitogen-activated Protein Kinase Kinase Kinase 9, Human 11
M4K1_HUMAN Q92918 CHEMBL5749 Mitogen-activated Protein Kinase Kinase Kinase Kinase 1, Human 11
MK13_HUMAN O15264 CHEMBL2939 MAP Kinase P38 Delta, Human 11
MKNK2_HUMAN Q9HBH9 CHEMBL4204 MAP Kinase Signal-integrating Kinase 2, Human 11
MUSK_HUMAN O15146 CHEMBL5684 Muscle, Skeletal Receptor Tyrosine Protein Kinase, Human 11
PHKG1_HUMAN Q16816 CHEMBL4004 Phosphorylase Kinase Gamma Subunit 1, Human 11
TNK1_HUMAN Q13470 CHEMBL5334 Non-receptor Tyrosine-protein Kinase TNK1, Human 11
TTK_HUMAN P33981 CHEMBL3983 Dual Specificity Protein Kinase TTK, Human 11
AAK1_HUMAN Q2M2I8 CHEMBL3830 Adaptor-associated Kinase, Human 10
CLK1_HUMAN P49759 CHEMBL4224 Dual Specificty Protein Kinase CLK1, Human 10
E2AK2_HUMAN P19525 CHEMBL5785 Interferon-induced, Double-stranded RNA-activated Protein Kinase, Human 10
FAK2_HUMAN Q14289 CHEMBL5469 Protein Tyrosine Kinase 2 Beta, Human 10
IGF1R_HUMAN P08069 CHEMBL1957 Insulin-like Growth Factor I Receptor, Human 10
KS6A2_HUMAN Q15349 CHEMBL3906 Ribosomal Protein S6 Kinase Alpha 2, Human 10
LTK_HUMAN P29376 CHEMBL5627 Leukocyte Tyrosine Kinase Receptor, Human 10
M3K11_HUMAN Q16584 CHEMBL2708 Mitogen-activated Protein Kinase Kinase Kinase 11, Human 10
NTRK3_HUMAN Q16288 CHEMBL5608 NT-3 Growth Factor Receptor, Human 10
SIK1_HUMAN P57059 CHEMBL6082 Serine/threonine-protein Kinase SIK1, Human 10
SRMS_HUMAN Q9H3Y6 CHEMBL5703 Tyrosine-protein Kinase Srms, Human 10
ST17A_HUMAN Q9UEE5 CHEMBL4525 Serine/threonine-protein Kinase 17A, Human 10
STK36_HUMAN Q9NRP7 CHEMBL4312 Serine/threonine-protein Kinase 36, Human 10
AAPK1_HUMAN Q13131 CHEMBL4045 AMP-activated Protein Kinase, Alpha-1 Subunit, Human 9
ANKK1_HUMAN Q8NFD2 CHEMBL5547 Ankyrin Repeat And Protein Kinase Domain-containing Protein 1, Human 9
CLK2_HUMAN P49760 CHEMBL4225 Dual Specificity Protein Kinase CLK2, Human 9
CLK4_HUMAN Q9HAZ1 CHEMBL4203 Dual Specificity Protein Kinase CLK4, Human 9
EPHA7_HUMAN Q15375 CHEMBL4602 Ephrin Type-A Receptor 7, Human 9
FAK1_HUMAN Q05397 CHEMBL2695 Focal Adhesion Kinase 1, Human 9
FER_HUMAN P16591 CHEMBL3982 Tyrosine-protein Kinase FER, Human 9
IRAK3_HUMAN Q9Y616 CHEMBL5081 Interleukin-1 Receptor-associated Kinase 3, Human 9
KCC1A_HUMAN Q14012 CHEMBL2493 CaM Kinase I Alpha, Human 9
KPCD1_HUMAN Q15139 CHEMBL3863 Protein Kinase C Mu, Human 9
KPCD3_HUMAN O94806 CHEMBL2595 Protein Kinase C Nu, Human 9
NEK2_HUMAN P51955 CHEMBL3835 Serine/threonine-protein Kinase NEK2, Human 9
NUAK2_HUMAN Q9H093 CHEMBL5698 NUAK Family SNF1-like Kinase 2, Human 9
PHKG2_HUMAN P15735 CHEMBL2349 Phosphorylase Kinase Gamma Subunit 2, Human 9
STK33_HUMAN Q9BYT3 CHEMBL6005 Serine/threonine-protein Kinase 33, Human 9
STK4_HUMAN Q13043 CHEMBL4598 Serine/threonine-protein Kinase MST1, Human 9
CDK7_HUMAN P50613 CHEMBL3055 Cyclin-dependent Kinase 7, Human 8
DCLK3_HUMAN Q9C098 CHEMBL6123 Serine/threonine-protein Kinase DCLK3, Human 8
FES_HUMAN P07332 CHEMBL5455 Tyrosine-protein Kinase FES, Human 8
KCC1D_HUMAN Q8IU85 CHEMBL5073 CaM Kinase I Delta, Human 8
KKCC1_HUMAN Q8N5S9 CHEMBL5256 CaM-kinase Kinase Alpha, Human 8
KKCC2_HUMAN Q96RR4 CHEMBL5284 CaM-kinase Kinase Beta, Human 8
KPCA_HUMAN P17252 CHEMBL299 Protein Kinase C Alpha, Human 8
KS6A4_HUMAN O75676 CHEMBL3125 Ribosomal Protein S6 Kinase Alpha 4, Human 8
LATS1_HUMAN O95835 CHEMBL6167 Serine/threonine-protein Kinase LATS1, Human 8
M3K4_HUMAN Q9Y6R4 CHEMBL4853 Mitogen-activated Protein Kinase Kinase Kinase 4, Human 8
MARK3_HUMAN P27448 CHEMBL5600 Serine/threonine-protein Kinase C-TAK1, Human 8
MELK_HUMAN Q14680 CHEMBL4578 Maternal Embryonic Leucine Zipper Kinase, Human 8
MK08_HUMAN P45983 CHEMBL2276 C-Jun N-terminal Kinase 1, Human 8
NLK_HUMAN Q9UBE8 CHEMBL5364 Serine/threonine Protein Kinase NLK, Human 8
PI42B_HUMAN P78356 CHEMBL5667 Phosphatidylinositol-5-phosphate 4-kinase Type-2 Beta, Human 8
PKN1_HUMAN Q16512 CHEMBL3384 Protein Kinase N1, Human 8
ST17B_HUMAN O94768 CHEMBL3980 Serine/threonine-protein Kinase 17B, Human 8
STK24_HUMAN Q9Y6E0 CHEMBL5082 Serine/threonine-protein Kinase 24, Human 8
STK25_HUMAN O00506 CHEMBL5552 Serine/threonine-protein Kinase 25, Human 8
TBA1A_RAT P68370 CHEMBL4139 Tubulin Alpha-1 Chain, Rat 8
WEE1_HUMAN P30291 CHEMBL5491 Serine/threonine-protein Kinase WEE1, Human 8
AAKB1_HUMAN Q9Y478 CHEMBL3847 AMP-activated Protein Kinase, Beta-1 Subunit, Human 7
AAKG1_HUMAN P54619 CHEMBL2393 AMP-activated Protein Kinase, Gamma-1 Subunit, Human 7
ADCK4_HUMAN Q96D53 CHEMBL5753 Uncharacterized AarF Domain-containing Protein Kinase 4, Human 7
CSK21_HUMAN P68400 CHEMBL3629 Casein Kinase II Alpha, Human 7
CSK22_HUMAN P19784 CHEMBL4070 Casein Kinase II Alpha (prime), Human 7
ERBB4_HUMAN Q15303 CHEMBL3009 Receptor Protein-tyrosine Kinase ErbB-4, Human 7
KAPCA_HUMAN P17612 CHEMBL4101 CAMP-dependent Protein Kinase Alpha-catalytic Subunit, Human 7
KAPCB_HUMAN P22694 CHEMBL2918 CAMP-dependent Protein Kinase Beta-1 Catalytic Subunit, Human 7
KC1AL_HUMAN Q8N752 CHEMBL5520 Casein Kinase I Isoform Alpha-like, Human 7
KPCD2_HUMAN Q9BZL6 CHEMBL4900 Serine/threonine-protein Kinase D2, Human 7
KPCG_HUMAN P05129 CHEMBL2938 Protein Kinase C Gamma, Human 7
KS6A5_HUMAN O75582 CHEMBL4237 Ribosomal Protein S6 Kinase Alpha 5, Human 7
LATS2_HUMAN Q9NRM7 CHEMBL5907 Serine/threonine-protein Kinase LATS2, Human 7
MARK1_HUMAN Q9P0L2 CHEMBL5940 Serine/threonine-protein Kinase MARK1, Human 7
MARK2_HUMAN Q7KZI7 CHEMBL3831 MAP/microtubule Affinity-regulating Kinase 2, Human 7
MK01_HUMAN P28482 CHEMBL4040 MAP Kinase ERK2, Human 7
MRCKG_HUMAN Q6DT37 CHEMBL5615 Serine/threonine-protein Kinase MRCK Gamma, Human 7
MST4_HUMAN Q9P289 CHEMBL5941 Serine/threonine-protein Kinase MST4, Human 7
NUAK1_HUMAN O60285 CHEMBL5784 NUAK Family SNF1-like Kinase 1, Human 7
PI51A_HUMAN Q99755 CHEMBL5969 Phosphatidylinositol-4-phosphate 5-kinase Type-1 Alpha, Human 7
RIOK1_HUMAN Q9BRS2 CHEMBL5975 Serine/threonine-protein Kinase RIO1, Human 7
RIPK1_HUMAN Q13546 CHEMBL5464 Receptor-interacting Serine/threonine-protein Kinase 1, Human 7
CDK19_HUMAN Q9BWU1 CHEMBL6002 Cell Division Cycle 2-like Protein Kinase 6, Human 6
CDK1_HUMAN P06493 CHEMBL308 Cyclin-dependent Kinase 1, Human 6
DMPK_HUMAN Q09013 CHEMBL5320 Myotonin-protein Kinase, Human 6
DYR1B_HUMAN Q9Y463 CHEMBL5543 Dual Specificity Tyrosine-phosphorylation-regulated Kinase 1B, Human 6
IKKE_HUMAN Q14164 CHEMBL3529 Inhibitor Of Nuclear Factor Kappa B Kinase Epsilon Subunit, Human 6
INSRR_HUMAN P14616 CHEMBL5483 Insulin Receptor-related Protein, Human 6
IRAK4_HUMAN Q9NWZ3 CHEMBL3778 Interleukin-1 Receptor-associated Kinase 4, Human 6
JAK1_HUMAN P23458 CHEMBL2835 Tyrosine-protein Kinase JAK1, Human 6
KC1G2_HUMAN P78368 CHEMBL2543 Casein Kinase I Gamma 2, Human 6
KCC2G_HUMAN Q13555 CHEMBL3829 CaM Kinase II Gamma, Human 6
KCC4_HUMAN Q16566 CHEMBL2494 CaM Kinase IV, Human 6
KS6B1_HUMAN P23443 CHEMBL4501 Ribosomal Protein S6 Kinase 1, Human 6
LIMK1_HUMAN P53667 CHEMBL3836 LIM Domain Kinase 1, Human 6
MARK4_HUMAN Q96L34 CHEMBL5754 MAP/microtubule Affinity-regulating Kinase 4, Human 6
MRCKA_HUMAN Q5VT25 CHEMBL4516 Serine/threonine-protein Kinase MRCK-A, Human 6
MRCKB_HUMAN Q9Y5S2 CHEMBL5052 Serine/threonine-protein Kinase MRCK Beta, Human 6
MYLK4_HUMAN Q86YV6 CHEMBL5426 Myosin Light Chain Kinase Family Member 4, Human 6
MYLK_CHICK P11799 CHEMBL3062 Myosin Light Chain Kinase, Smooth Muscle, Chick 6
MYLK_HUMAN Q15746 CHEMBL2428 Myosin Light Chain Kinase, Smooth Muscle, Human 6
P85A_HUMAN P27986 CHEMBL2506 PI3-kinase P85-alpha Subunit, Human 6
PAK3_HUMAN O75914 CHEMBL2999 Serine/threonine-protein Kinase PAK 3, Human 6
PDPK1_HUMAN O15530 CHEMBL2534 3-phosphoinositide Dependent Protein Kinase-1, Human 6
PIM3_HUMAN Q86V86 CHEMBL5407 Serine/threonine-protein Kinase PIM3, Human 6
PKN2_HUMAN Q16513 CHEMBL3032 Protein Kinase N2, Human 6
RIOK3_HUMAN O14730 CHEMBL5659 Serine/threonine-protein Kinase RIO3, Human 6
RON_HUMAN Q04912 CHEMBL2689 Macrophage-stimulating Protein Receptor, Human 6
ROS1_HUMAN P08922 CHEMBL5568 Proto-oncogene Tyrosine-protein Kinase ROS, Human 6
SRPK1_HUMAN Q96SB4 CHEMBL4375 Serine/threonine-protein Kinase SRPK1, Human 6
SRPK2_HUMAN P78362 CHEMBL5668 Serine/threonine-protein Kinase SRPK2, Human 6
STK11_HUMAN Q15831 CHEMBL5606 Serine/threonine-protein Kinase 11, Human 6
STK16_HUMAN O75716 CHEMBL3938 Serine/threonine-protein Kinase 16, Human 6
TESK1_HUMAN Q15569 CHEMBL5604 Dual Specificity Testis-specific Protein Kinase 1, Human 6
ACVR1_HUMAN Q04771 CHEMBL5903 Activin Receptor Type-1, Human 5
BCR_HUMAN P11274 CHEMBL5146 Breakpoint Cluster Region Protein, Human 5
BLK_MOUSE P16277 CHEMBL3343 Tyrosine-protein Kinase BLK, Mouse 5
BMPR2_HUMAN Q13873 CHEMBL5467 Bone Morphogenetic Protein Receptor Type-2, Human 5
CDK17_HUMAN Q00537 CHEMBL5790 Serine/threonine-protein Kinase PCTAIRE-2, Human 5
DAPK1_HUMAN P53355 CHEMBL2558 Death-associated Protein Kinase 1, Human 5
DAPK2_HUMAN Q9UIK4 CHEMBL3123 Death-associated Protein Kinase 2, Human 5
IKKA_HUMAN O15111 CHEMBL3476 Inhibitor Of Nuclear Factor Kappa B Kinase Alpha Subunit, Human 5
KAPCG_HUMAN P22612 CHEMBL2743 CAMP-dependent Protein Kinase, Gamma Catalytic Subunit, Human 5
KC1A_HUMAN P48729 CHEMBL2793 Casein Kinase I Alpha, Human 5
KC1G1_HUMAN Q9HCP0 CHEMBL2426 Casein Kinase I Gamma 1, Human 5
KCC1G_HUMAN Q96NX5 CHEMBL5258 CaM Kinase I Gamma, Human 5
KCC2A_HUMAN Q9UQM7 CHEMBL4147 CaM Kinase II Alpha, Human 5
KCC2B_HUMAN Q13554 CHEMBL4121 CaM Kinase II Beta, Human 5
KCC2D_HUMAN Q13557 CHEMBL2801 CaM Kinase II Delta, Human 5
KPCI_HUMAN P41743 CHEMBL2598 Protein Kinase C Iota, Human 5
KPCZ_HUMAN Q05513 CHEMBL3438 Protein Kinase C Zeta, Human 5
MK15_HUMAN Q8TD08 CHEMBL5198 Mitogen-activated Protein Kinase 15, Human 5
MP2K4_HUMAN P45985 CHEMBL2897 Dual Specificity Mitogen-activated Protein Kinase Kinase 4, Human 5
MP2K6_HUMAN P52564 CHEMBL2171 Dual Specificity Mitogen-activated Protein Kinase Kinase 6, Human 5
NEK5_HUMAN Q6P3R8 CHEMBL5044 Serine/threonine-protein Kinase Nek5, Human 5
NEK7_HUMAN Q8TDX7 CHEMBL4849 Serine/threonine-protein Kinase NEK7, Human 5
P85B_HUMAN O00459 CHEMBL4437 PI3-kinase P85-beta Subunit, Human 5
PAK1_HUMAN Q13153 CHEMBL4600 Serine/threonine-protein Kinase PAK 1, Human 5
ROCK1_HUMAN Q13464 CHEMBL3231 Rho-associated Protein Kinase 1, Human 5
SRC_CHICK P00523 CHEMBL3655 Tyrosine-protein Kinase SRC, Chick 5
ST38L_HUMAN Q9Y2H1 CHEMBL4851 Serine/threonine-protein Kinase 38-like, Human 5
TEC_HUMAN P42680 CHEMBL4246 Tyrosine-protein Kinase TEC, Human 5
TGFR1_HUMAN P36897 CHEMBL4439 TGF-beta Receptor Type I, Human 5
TGFR2_HUMAN P37173 CHEMBL4267 TGF-beta Receptor Type II, Human 5
TLK2_HUMAN Q86UE8 CHEMBL5404 Serine/threonine-protein Kinase Tousled-like 2, Human 5
ULK3_MOUSE Q3U3Q1 CHEMBL3832 ULK3 Kinase, Mouse 5
ACV1B_HUMAN P36896 CHEMBL5310 Activin Receptor Type-1B, Human 4
ADCK3_HUMAN Q8NI60 CHEMBL5550 Chaperone Activity Of Bc1 Complex-like, Mitochondrial, Human 4
AKT3_HUMAN Q9Y243 CHEMBL4816 Serine/threonine-protein Kinase AKT3, Human 4
BRSK1_HUMAN Q8TDC3 CHEMBL5650 BR Serine/threonine-protein Kinase 1, Human 4
BRSK2_HUMAN Q8IWQ3 CHEMBL4574 BR Serine/threonine-protein Kinase 2, Human 4
CD11A_HUMAN Q9UQ88 CHEMBL5416 PITSLRE Serine/threonine-protein Kinase CDC2L2, Human 4
CD11B_HUMAN P21127 CHEMBL5808 PITSLRE Serine/threonine-protein Kinase CDC2L1, Human 4
CDK14_HUMAN O94921 CHEMBL6162 Serine/threonine-protein Kinase PFTAIRE-1, Human 4
CDK5_HUMAN Q00535 CHEMBL4036 Cyclin-dependent Kinase 5, Human 4
CDK8_HUMAN P49336 CHEMBL5719 Cell Division Protein Kinase 8, Human 4
CDK9_HUMAN P50750 CHEMBL3116 Cyclin-dependent Kinase 9, Human 4
DCLK1_HUMAN O15075 CHEMBL5683 Serine/threonine-protein Kinase DCLK1, Human 4
GRB2_HUMAN P62993 CHEMBL3663 Growth Factor Receptor-bound Protein 2, Human 4
GSK3A_HUMAN P49840 CHEMBL2850 Glycogen Synthase Kinase-3 Alpha, Human 4
IKKB_HUMAN O14920 CHEMBL1991 Inhibitor Of Nuclear Factor Kappa B Kinase Beta Subunit, Human 4
KC1G3_HUMAN Q9Y6M4 CHEMBL5084 Casein Kinase I Isoform Gamma-3, Human 4
LIMK2_HUMAN P53671 CHEMBL5932 LIM Domain Kinase 2, Human 4
M3K10_HUMAN Q02779 CHEMBL2873 Mitogen-activated Protein Kinase Kinase Kinase 10, Human 4
M3K7_HUMAN O43318 CHEMBL5776 Mitogen-activated Protein Kinase Kinase Kinase 7, Human 4
MAPK2_HUMAN P49137 CHEMBL2208 MAP Kinase-activated Protein Kinase 2, Human 4
MAPK5_HUMAN Q8IW41 CHEMBL3094 MAP Kinase-activated Protein Kinase 5, Human 4
MK14_MOUSE P47811 CHEMBL2336 MAP Kinase P38 Alpha, Mouse 4
PAK4_HUMAN O96013 CHEMBL4482 Serine/threonine-protein Kinase PAK 4, Human 4
PIM1_HUMAN P11309 CHEMBL2147 Serine/threonine-protein Kinase PIM1, Human 4
PIM2_HUMAN Q9P1W9 CHEMBL4523 Serine/threonine-protein Kinase PIM2, Human 4
PLK1_HUMAN P53350 CHEMBL3024 Serine/threonine-protein Kinase PLK1, Human 4
SGK1_HUMAN O00141 CHEMBL2343 Serine/threonine-protein Kinase Sgk1, Human 4
ST32B_HUMAN Q9NY57 CHEMBL5912 Serine/threonine-protein Kinase 32B, Human 4
STK3_MOUSE Q9JI10 CHEMBL4310 Serine/threonine-protein Kinase MST2, Mouse 4
SYK_HUMAN Q15046 CHEMBL5575 Lysyl-tRNA Synthetase, Human 4
TLK1_HUMAN Q9UKI8 CHEMBL5388 Serine/threonine-protein Kinase Tousled-like 1, Human 4
ABL1_MOUSE P00520 CHEMBL3099 Tyrosine-protein Kinase ABL, Mouse 3
AKT1_HUMAN P31749 CHEMBL4282 Serine/threonine-protein Kinase AKT, Human 3
AKT2_HUMAN P31751 CHEMBL2431 Serine/threonine-protein Kinase AKT2, Human 3
AVR2B_HUMAN Q13705 CHEMBL5466 Activin Receptor Type-2B, Human 3
CCNB1_HUMAN P14635 CHEMBL2412 G2/mitotic-specific Cyclin B1, Human 3
CCNB2_HUMAN O95067 CHEMBL3723 G2/mitotic-specific Cyclin B2, Human 3
CCNB3_HUMAN Q8WWL7 CHEMBL3606 G2/mitotic-specific Cyclin B3, Human 3
CDK18_HUMAN Q07002 CHEMBL5316 Serine/threonine-protein Kinase PCTAIRE-3, Human 3
CDK4_HUMAN P11802 CHEMBL331 Cyclin-dependent Kinase 4, Human 3
CHK2_HUMAN O96017 CHEMBL2527 Serine/threonine-protein Kinase Chk2, Human 3
CLK3_HUMAN P49761 CHEMBL4226 Dual Specificity Protein Kinase CLK3, Human 3
EPHB3_HUMAN P54753 CHEMBL4901 Ephrin Type-B Receptor 3, Human 3
MINK1_HUMAN Q8N4C8 CHEMBL5518 Misshapen-like Kinase 1, Human 3
MK06_HUMAN Q16659 CHEMBL5121 Mitogen-activated Protein Kinase 6, Human 3
MYO3B_HUMAN Q8WXR4 CHEMBL5654 Myosin-IIIB, Human 3
PAK7_HUMAN Q9P286 CHEMBL4524 Serine/threonine-protein Kinase PAK7, Human 3
PGFRB_MOUSE P05622 CHEMBL2749 Platelet-derived Growth Factor Receptor Beta, Mouse 3
ROCK2_HUMAN O75116 CHEMBL2973 Rho-associated Protein Kinase 2, Human 3
VGFR2_MOUSE P35918 CHEMBL3337 Vascular Endothelial Growth Factor Receptor 2, Mouse 3
Z80840 Z80840 CHEMBL614490 ER22 Cell Line 3
ABCG2_HUMAN Q9UNQ0 CHEMBL5393 ATP-binding Cassette Sub-family G Member 2, Human 2
ACVL1_HUMAN P37023 CHEMBL5311 Serine/threonine-protein Kinase Receptor R3, Human 2
ALDR_RAT P07943 CHEMBL2622 Aldose Reductase, Rat 2
BMP4_HUMAN P12644 CHEMBL5350 Bone Morphogenetic Protein 4, Human 2
CCNA2_HUMAN P20248 CHEMBL2582 Cyclin A2, Human 2
CCNT1_HUMAN O60563 CHEMBL2108 Cyclin T1, Human 2
CDK3_HUMAN Q00526 CHEMBL4442 Cyclin-dependent Kinase 3, Human 2
CDK6_HUMAN Q00534 CHEMBL2508 Cyclin-dependent Kinase 6, Human 2
CDKL2_HUMAN Q92772 CHEMBL5728 Cyclin-dependent Kinase-like 2, Human 2
DCLK2_HUMAN Q8N568 CHEMBL5519 Serine/threonine-protein Kinase DCLK2, Human 2
DYR1A_HUMAN Q13627 CHEMBL2292 Dual-specificity Tyrosine-phosphorylation Regulated Kinase 1A, Human 2
EPHB6_HUMAN O15197 CHEMBL5836 Ephrin Type-B Receptor 6, Human 2
F16P1_HUMAN P09467 CHEMBL3975 Fructose-1,6-bisphosphatase, Human 2
HGF_HUMAN P14210 CHEMBL5479 Hepatocyte Growth Factor, Human 2
HIPK1_HUMAN Q86Z02 CHEMBL5427 Homeodomain-interacting Protein Kinase 1, Human 2
HIPK2_HUMAN Q9H2X6 CHEMBL4576 Homeodomain-interacting Protein Kinase 2, Human 2
HIPK3_HUMAN Q9H422 CHEMBL4577 Homeodomain-interacting Protein Kinase 3, Human 2
HIPK4_HUMAN Q8NE63 CHEMBL1075167 Homeodomain-interacting Protein Kinase 4, Human 2
KGP2_HUMAN Q13237 CHEMBL2896 CGMP-dependent Protein Kinase 2, Human 2
KPCA_RAT P05696 CHEMBL2855 Protein Kinase C Alpha, Rat 2
KPCB_RAT P68403 CHEMBL3020 Protein Kinase C Beta, Rat 2
KPCD_RAT P09215 CHEMBL3633 Protein Kinase C Delta, Rat 2
KPCE_RAT P09216 CHEMBL3424 Protein Kinase C Epsilon, Rat 2
KPCG_RAT P63319 CHEMBL3604 Protein Kinase C Gamma, Rat 2
KPCL_RAT Q64617 CHEMBL3990 Protein Kinase C Eta, Rat 2
KPCT_MOUSE Q02111 CHEMBL1075295 Protein Kinase C Theta Type, Mouse 2
KPCT_RAT Q9WTQ0 CHEMBL4563 Protein Kinase C Theta, Rat 2
KPCZ_RAT P09217 CHEMBL5379 Protein Kinase C Zeta, Rat 2
M4K2_HUMAN Q12851 CHEMBL5330 Mitogen-activated Protein Kinase Kinase Kinase Kinase 2, Human 2
MK04_HUMAN P31152 CHEMBL5759 Mitogen-activated Protein Kinase 4, Human 2
MYO3A_HUMAN Q8NEV4 CHEMBL5546 Myosin IIIA, Human 2
NEK1_HUMAN Q96PY6 CHEMBL5855 Serine/threonine-protein Kinase Nek1, Human 2
NEK9_HUMAN Q8TD19 CHEMBL5257 Serine/threonine-protein Kinase NEK9, Human 2
NPM_HUMAN P06748 CHEMBL5178 Nucleophosmin, Human 2
PAK2_HUMAN Q13177 CHEMBL4487 Serine/threonine-protein Kinase PAK 2, Human 2
PAK6_HUMAN Q9NQU5 CHEMBL4311 Serine/threonine-protein Kinase PAK6, Human 2
PDK1_HUMAN Q15118 CHEMBL4766 Pyruvate Dehydrogenase Kinase Isoform 1, Human 2
PGH1_HUMAN P23219 CHEMBL221 Cyclooxygenase-1, Human 2
PLK2_HUMAN Q9NYY3 CHEMBL5938 Serine/threonine-protein Kinase PLK2, Human 2
PLK3_HUMAN Q9H4B4 CHEMBL4897 Serine/threonine-protein Kinase PLK3, Human 2
PMYT1_HUMAN Q99640 CHEMBL3984 Tyrosine- And Threonine-specific Cdc2-inhibitory Kinase, Human 2
Q5SC61_TOXGO Q5SC61 CHEMBL6051 Mitogen-activated Protein Kinase 1, Toxgo 2
TAOK1_HUMAN Q7L7X3 CHEMBL5261 Serine/threonine-protein Kinase TAO1, Human 2
TAOK3_HUMAN Q9H2K8 CHEMBL5701 Serine/threonine-protein Kinase TAO3, Human 2
TBK1_HUMAN Q9UHD2 CHEMBL5408 Serine/threonine-protein Kinase TBK1, Human 2
TSSK1_HUMAN Q9BXA7 CHEMBL6003 Testis-specific Serine/threonine-protein Kinase 1, Human 2
VGFR1_MOUSE P35969 CHEMBL3516 Vascular Endothelial Growth Factor Receptor 1, Mouse 2
YSK4_HUMAN Q56UN5 CHEMBL6191 SPS1/STE20-related Protein Kinase YSK4, Human 2
Z104294 Z104294 CHEMBL1907600 Cyclin-dependent Kinase 5/CDK5 Activator 1 2
Z104299 Z104299 CHEMBL1907605 Cyclin-dependent Kinase 2/cyclin E1 2
A1Z199_HUMAN A1Z199 CHEMBL6105 BCR/ABL P210 Fusion Protein, Human 1
ABL2_MOUSE Q4JIM5 CHEMBL5222 Tyrosine-protein Kinase ABL2, Mouse 1
ABL_MLVAB P00521 CHEMBL5166 Tyrosine-protein Kinase V-ABL, Mlvab 1
AKIP_HUMAN Q9NWT8 CHEMBL5910 Aurora Kinase A-interacting Protein, Human 1
AURKA_MOUSE P97477 CHEMBL2211 Serine/threonine-protein Kinase Aurora-A, Mouse 1
AURKB_MOUSE O70126 CHEMBL1075275 Serine/threonine-protein Kinase 12, Mouse 1
AVR2A_HUMAN P27037 CHEMBL5616 Activin Receptor Type-2A, Human 1
BMR1A_HUMAN P36894 CHEMBL5275 Bone Morphogenetic Protein Receptor Type-1A, Human 1
BRD4_HUMAN O60885 CHEMBL1163125 Bromodomain-containing Protein 4, Human 1
CAH12_HUMAN O43570 CHEMBL3242 Carbonic Anhydrase XII, Human 1
CAH13_MOUSE Q9D6N1 CHEMBL2186 Carbonic Anhydrase XIII, Mouse 1
CAH14_HUMAN Q9ULX7 CHEMBL3510 Carbonic Anhydrase XIV, Human 1
CAH15_MOUSE Q99N23 CHEMBL5973 Carbonic Anhydrase 15, Mouse 1
CAH1_HUMAN P00915 CHEMBL261 Carbonic Anhydrase I, Human 1
CAH2_HUMAN P00918 CHEMBL205 Carbonic Anhydrase II, Human 1
CAH3_HUMAN P07451 CHEMBL2885 Carbonic Anhydrase III, Human 1
CAH4_HUMAN P22748 CHEMBL3729 Carbonic Anhydrase IV, Human 1
CAH6_HUMAN P23280 CHEMBL3025 Carbonic Anhydrase VI, Human 1
CAH7_HUMAN P43166 CHEMBL2326 Carbonic Anhydrase VII, Human 1
CAH9_HUMAN Q16790 CHEMBL3594 Carbonic Anhydrase IX, Human 1
CATL1_HUMAN P07711 CHEMBL3837 Cathepsin L, Human 1
CATS_HUMAN P25774 CHEMBL2954 Cathepsin S, Human 1
CCNA1_HUMAN P78396 CHEMBL3609 Cyclin A1, Human 1
CCND1_HUMAN P24385 CHEMBL3610 G1/S-specific Cyclin D1, Human 1
CCND2_HUMAN P30279 CHEMBL3613 G1/S-specific Cyclin D2, Human 1
CCNE1_HUMAN P24864 CHEMBL3617 G1/S-specific Cyclin E1, Human 1
CCNE2_HUMAN O96020 CHEMBL2884 G1/S-specific Cyclin E2, Human 1
CDK15_HUMAN Q96Q40 CHEMBL5856 Serine/threonine-protein Kinase PFTAIRE-2, Human 1
CDK1_MOUSE P11440 CHEMBL4084 Cyclin-dependent Kinase 1, Mouse 1
CDKL3_HUMAN Q8IVW4 CHEMBL1163117 Cyclin-dependent Kinase-like 3, Human 1
CSK21_RAT P19139 CHEMBL2661 Casein Kinase II Alpha, Rat 1
CSK2B_HUMAN P67870 CHEMBL2358 Casein Kinase II Beta, Human 1
CSK2B_RAT P67874 CHEMBL2463 Casein Kinase II Beta, Rat 1
DLK1_HUMAN P80370 CHEMBL5671 Protein Delta Homolog 1, Human 1
DYRK2_HUMAN Q92630 CHEMBL4376 Dual-specificity Tyrosine-phosphorylation Regulated Kinase 2, Human 1
ERN1_HUMAN O75460 CHEMBL1163101 Serine/threonine-protein Kinase/endoribonuclease IRE1, Human 1
GRK4_HUMAN P32298 CHEMBL5861 G Protein-coupled Receptor Kinase 4, Human 1
GRK7_HUMAN Q8WTQ7 CHEMBL1075133 G Protein-coupled Receptor Kinase 7, Human 1
HDA10_HUMAN Q969S8 CHEMBL5103 Histone Deacetylase 10, Human 1
HDAC1_HUMAN Q13547 CHEMBL325 Histone Deacetylase 1, Human 1
HDAC2_HUMAN Q92769 CHEMBL1937 Histone Deacetylase 2, Human 1
HDAC3_HUMAN O15379 CHEMBL1829 Histone Deacetylase 3, Human 1
HDAC4_HUMAN P56524 CHEMBL3524 Histone Deacetylase 4, Human 1
HDAC5_HUMAN Q9UQL6 CHEMBL2563 Histone Deacetylase 5, Human 1
HDAC6_HUMAN Q9UBN7 CHEMBL1865 Histone Deacetylase 6, Human 1
HDAC7_HUMAN Q8WUI4 CHEMBL2716 Histone Deacetylase 7, Human 1
HDAC8_HUMAN Q9BY41 CHEMBL3192 Histone Deacetylase 8, Human 1
HDAC9_HUMAN Q9UKV0 CHEMBL4145 Histone Deacetylase 9, Human 1
HSPB1_HUMAN P04792 CHEMBL5976 Heat Shock Protein Beta-1, Human 1
ICK_HUMAN Q9UPZ9 CHEMBL1163126 Serine/threonine-protein Kinase ICK, Human 1
IGF1R_MOUSE Q60751 CHEMBL5381 Insulin-like Growth Factor 1 Receptor, Mouse 1
INSR_MOUSE P15208 CHEMBL3187 Insulin Receptor, Mouse 1
IRAK1_HUMAN P51617 CHEMBL3357 Interleukin-1 Receptor-associated Kinase 1, Human 1
JAK3_MOUSE Q62137 CHEMBL5250 Tyrosine-protein Kinase JAK3, Mouse 1
KAP2_BOVIN P00515 CHEMBL3654 CAMP-dependent Protein Kinase Type II-alpha Regulatory Subunit, Bovin 1
KAPCA_BOVIN P00517 CHEMBL2654 CAMP-dependent Protein Kinase Alpha-catalytic Subunit, Bovin 1
KAPCA_MOUSE P05132 CHEMBL4991 CAMP-dependent Protein Kinase Alpha-catalytic Subunit, Mouse 1
KAPCA_RAT P27791 CHEMBL3390 CAMP-dependent Protein Kinase Alpha-catalytic Subunit, Rat 1
KAPCB_BOVIN P05131 CHEMBL3279 CAMP-dependent Protein Kinase Beta-1 Catalytic Subunit, Bovin 1
KAPCB_MOUSE P68181 CHEMBL2481 CAMP-dependent Protein Kinase Beta-1 Catalytic Subunit, Mouse 1
KC1A_MOUSE Q8BK63 CHEMBL5148 Casein Kinase I Alpha, Mouse 1
KC1D_MOUSE Q9DC28 CHEMBL5175 Casein Kinase I Delta, Mouse 1
KC1E_MOUSE Q9JMK2 CHEMBL5140 Casein Kinase I Epsilon, Mouse 1
KC1G1_MOUSE Q8BTH8 CHEMBL4455 Casein Kinase I Gamma 1, Mouse 1
KCC2A_MOUSE P11798 CHEMBL3347 CaM Kinase II Alpha, Mouse 1
KCC2A_RAT P11275 CHEMBL2359 CaM Kinase II Alpha, Rat 1
KCC2B_MOUSE P28652 CHEMBL4735 CaM Kinase II Beta, Mouse 1
KCC2G_MOUSE Q923T9 CHEMBL4456 CaM Kinase II Gamma, Mouse 1
KGP1_BOVIN P00516 CHEMBL3183 CGMP-dependent Protein Kinase 1 Alpha, Bovin 1
KGP1_HUMAN Q13976 CHEMBL4273 CGMP-dependent Protein Kinase 1 Beta, Human 1
KPB1_HUMAN P46020 CHEMBL2905 Phosphorylase Kinase Alpha M Subunit, Human 1
KPB2_HUMAN P46019 CHEMBL2906 Phosphorylase Kinase Alpha L Subunit, Human 1
KPBB_HUMAN Q93100 CHEMBL3844 Phosphorylase Kinase Beta Subunit, Human 1
KS6B2_HUMAN Q9UBS0 CHEMBL3111 Ribosomal Protein S6 Kinase 2, Human 1
M3K13_HUMAN O43283 CHEMBL1163124 Mitogen-activated Protein Kinase Kinase Kinase 13, Human 1
M3K14_HUMAN Q99558 CHEMBL5888 Mitogen-activated Protein Kinase Kinase Kinase 14, Human 1
M3K15_HUMAN Q6ZN16 CHEMBL1163127 Mitogen-activated Protein Kinase Kinase Kinase 15, Human 1
M3K2_HUMAN Q9Y2U5 CHEMBL5914 Mitogen-activated Protein Kinase Kinase Kinase 2, Human 1
M3K3_HUMAN Q99759 CHEMBL5970 Mitogen-activated Protein Kinase Kinase Kinase 3, Human 1
M3K5_HUMAN Q99683 CHEMBL5285 Mitogen-activated Protein Kinase Kinase Kinase 5, Human 1
M3K8_HUMAN P41279 CHEMBL4899 Mitogen-activated Protein Kinase Kinase Kinase 8, Human 1
MAPK3_HUMAN Q16644 CHEMBL4670 MAP Kinase-activated Protein Kinase 3, Human 1
MAST1_HUMAN Q9Y2H9 CHEMBL1163128 Microtubule-associated Serine/threonine-protein Kinase 1, Human 1
MET_MOUSE P16056 CHEMBL5585 Hepatocyte Growth Factor Receptor, Mouse 1
MK03_HUMAN P27361 CHEMBL3385 MAP Kinase ERK1, Human 1
MK07_HUMAN Q13164 CHEMBL5332 Mitogen-activated Protein Kinase 7, Human 1
MP2K3_HUMAN P46734 CHEMBL2109 Dual Specificity Mitogen-activated Protein Kinase Kinase 3, Human 1
NEK6_HUMAN Q9HC98 CHEMBL4309 Serine/threonine-protein Kinase NEK6, Human 1
NIM1_HUMAN Q8IY84 CHEMBL3542 Serine/threonine-protein Kinase NIM1, Human 1
NOX4_HUMAN Q9NPH5 CHEMBL1250375 NADPH Oxidase 4, Human 1
OXSR1_HUMAN O95747 CHEMBL1163104 Serine/threonine-protein Kinase OSR1, Human 1
P90584_PLAFA P90584 CHEMBL4090 Protein Kinase Pfmrk, Plafa 1
PGFRA_MOUSE P26618 CHEMBL3466 Platelet-derived Growth Factor Receptor Alpha, Mouse 1
PGFRA_RAT P20786 CHEMBL2513 Platelet-derived Growth Factor Receptor Alpha, Rat 1
PLCG1_HUMAN P19174 CHEMBL3964 Phospholipase C-gamma-1, Human 1
PLCG2_HUMAN P16885 CHEMBL4100 Phospholipase C-gamma-2, Human 1
PRKX_HUMAN P51817 CHEMBL5818 Serine/threonine-protein Kinase PRKX, Human 1
PRP4_HUMAN O43172 CHEMBL1163119 U4/U6 Small Nuclear Ribonucleoprotein Prp4, Human 1
PTN13_HUMAN Q12923 CHEMBL2976 Protein-tyrosine Phosphatase 1E, Human 1
PTPRC_HUMAN P08575 CHEMBL3243 Leukocyte Common Antigen, Human 1
Q7ZJM1_9HIV1 Q7ZJM1 CHEMBL3471 Human Immunodeficiency Virus Type 1 Integrase, 9hiv1 1
Q95J97_RABIT Q95J97 CHEMBL4885 CAMP-dependent Protein Kinase Alpha-catalytic Subunit, Rabit 1
RIOK2_HUMAN Q9BVS4 CHEMBL6000 Serine/threonine-protein Kinase RIO2, Human 1
RIPK4_HUMAN P57078 CHEMBL6083 Receptor-interacting Serine/threonine-protein Kinase 4, Human 1
RK_HUMAN Q15835 CHEMBL5607 Rhodopsin Kinase, Human 1
RON_MOUSE Q62190 CHEMBL1795170 Macrophage-stimulating Protein Receptor, Mouse 1
SG110_HUMAN P0C264 CHEMBL5116 Putative Uncharacterized Serine/threonine-protein Kinase SgK110, Human 1
SRPK3_HUMAN Q9UPE1 CHEMBL5415 Serine/threonine-protein Kinase SRPK3, Human 1
ST32C_HUMAN Q86UX6 CHEMBL5405 Serine/threonine-protein Kinase 32C, Human 1
STK35_HUMAN Q8TDR2 CHEMBL5651 Serine/threonine-protein Kinase 35, Human 1
STK38_HUMAN Q15208 CHEMBL1075155 Serine/threonine-protein Kinase 38, Human 1
STK39_HUMAN Q9UEW8 CHEMBL1163108 STE20/SPS1-related Proline-alanine-rich Protein Kinase, Human 1
TAB1_HUMAN Q15750 CHEMBL5605 Mitogen-activated Protein Kinase Kinase Kinase 7-interacting Protein 1, Human 1
TIE2_MOUSE Q02858 CHEMBL5199 Tyrosine-protein Kinase TIE-2, Mouse 1
TNFA_HUMAN P01375 CHEMBL1825 TNF-alpha, Human 1
TNKS2_HUMAN Q9H2K2 CHEMBL6154 Tankyrase-2, Human 1
TNR1A_HUMAN P19438 CHEMBL3378 Tumor Necrosis Factor Receptor R1, Human 1
TPX2_HUMAN Q9ULW0 CHEMBL5389 Targeting Protein For Xklp2, Human 1
ULK1_HUMAN O75385 CHEMBL6006 Serine/threonine-protein Kinase ULK1, Human 1
ULK2_HUMAN Q8IYT8 CHEMBL5435 Serine/threonine-protein Kinase ULK2, Human 1
ULK3_HUMAN Q6PHR2 CHEMBL5047 Serine/threonine-protein Kinase ULK3, Human 1
VGFR3_MOUSE P35917 CHEMBL4758 Vascular Endothelial Growth Factor Receptor 3, Mouse 1
Z104295 Z104295 CHEMBL1907601 Cyclin-dependent Kinase 4/cyclin D1 1
Z104296 Z104296 CHEMBL1907602 Cyclin-dependent Kinase 1/cyclin B1 1
Z50594 Z50594 CHEMBL375 Mus Musculus 1
Z80384 Z80384 CHEMBL614233 PBL (Peripheral Blood Lymphocytes) 1
Z80416 Z80416 CHEMBL614630 Rat1 (Fibroblast Cells) 1
Z81072 Z81072 CHEMBL397 Jurkat (Acute Leukemic T-cells) 1
Z81338 Z81338 CHEMBL614309 T-cells 1