ZINC 12

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Quick Search ZINC ID or SMILES

Names
Compounds (2,609)
Reactome (2)
Related By:
Pathway (37)
Organism (2)
Gene (0)
Org. Clust. (3)
ChEMBL (248)
Rings (50)

Serotonin 1a (5-HT1a) Receptor, Human (2,609 Compounds)

Swissprot:: 5HT1A_HUMAN
Stitch:: 5HT1A_HUMAN
UniProt:: P08908
ChEMBL:: CHEMBL214
Reactome:: REACT_19231; REACT_17064
PDB:: HTR1A

Compound Summary

Annotation Type	Substances	Purchasable	Natural	In Man
Binding ≤ 10μM	2,609	146	55	49
Binding ≤ 1μM	2,436	128	43	44
Functional ≤ 10μM	286	24	6	6

Reactome ID	Description	Species
REACT_19231	G alpha (i) signalling events	Homo sapiens
REACT_17064	Serotonin receptors	Homo sapiens

Uniprot	Swissprot	Chembl	Description	Number Shared
5HT1B_HUMAN	P28222	CHEMBL1898	Serotonin 1b (5-HT1b) Receptor, Human	422
5HT1D_HUMAN	P28221	CHEMBL1983	Serotonin 1d (5-HT1d) Receptor, Human	434
5HT1E_HUMAN	P28566	CHEMBL2182	Serotonin 1e (5-HT1e) Receptor, Human	42
5HT1F_HUMAN	P30939	CHEMBL1805	Serotonin 1f (5-HT1f) Receptor, Human	72
5HT5A_HUMAN	P47898	CHEMBL3426	Serotonin 5a (5-HT5a) Receptor, Human	74
AA1R_HUMAN	P30542	CHEMBL226	Adenosine A1 Receptor, Human	3
AA3R_HUMAN	P33765	CHEMBL256	Adenosine A3 Receptor, Human	13
ACM2_HUMAN	P08172	CHEMBL211	Muscarinic Acetylcholine Receptor M2, Human	11
ACM4_HUMAN	P08173	CHEMBL1821	Muscarinic Acetylcholine Receptor M4, Human	11
ADA2A_HUMAN	P08913	CHEMBL1867	Alpha-2a Adrenergic Receptor, Human	51
ADA2B_HUMAN	P18089	CHEMBL1942	Alpha-2b Adrenergic Receptor, Human	29
ADA2C_HUMAN	P18825	CHEMBL1916	Alpha-2c Adrenergic Receptor, Human	35
ADCY1_HUMAN	Q08828	CHEMBL2899	Brain Adenylate Cyclase 1, Human	1
ADCY2_HUMAN	Q08462	CHEMBL3760	Adenylate Cyclase Type II, Human	1
ADCY8_HUMAN	P40145	CHEMBL2960	Adenylate Cyclase Type VIII, Human	1
CNR1_HUMAN	P21554	CHEMBL218	Cannabinoid CB1 Receptor, Human	5
CNR2_HUMAN	P34972	CHEMBL253	Cannabinoid CB2 Receptor, Human	1
CXCR3_HUMAN	P49682	CHEMBL4441	C-X-C Chemokine Receptor Type 3, Human	1
DRD2_HUMAN	P14416	CHEMBL217	Dopamine D2 Receptor, Human	607
DRD3_HUMAN	P35462	CHEMBL234	Dopamine D3 Receptor, Human	260
DRD4_HUMAN	P21917	CHEMBL219	Dopamine D4 Receptor, Human	176
HRH3_HUMAN	Q9Y5N1	CHEMBL264	Histamine H3 Receptor, Human	7
HRH4_HUMAN	Q9H3N8	CHEMBL3759	Histamine H4 Receptor, Human	4
MCHR1_HUMAN	Q99705	CHEMBL344	Melanin-concentrating Hormone Receptor 1, Human	2
MTR1A_HUMAN	P48039	CHEMBL1945	Melatonin Receptor 1A, Human	3
NPY1R_HUMAN	P25929	CHEMBL4777	Neuropeptide Y Receptor Type 1, Human	2
NPY5R_HUMAN	Q15761	CHEMBL4561	Neuropeptide Y Receptor Type 5, Human	2
OPRD_HUMAN	P41143	CHEMBL236	Delta Opioid Receptor, Human	5
OPRK_HUMAN	P41145	CHEMBL237	Kappa Opioid Receptor, Human	11
OPRM_HUMAN	P35372	CHEMBL233	Mu Opioid Receptor, Human	13

Serotonin receptors

Uniprot	Swissprot	Chembl	Description	Number Shared
5HT1B_HUMAN	P28222	CHEMBL1898	Serotonin 1b (5-HT1b) Receptor, Human	422
5HT1D_HUMAN	P28221	CHEMBL1983	Serotonin 1d (5-HT1d) Receptor, Human	434
5HT1E_HUMAN	P28566	CHEMBL2182	Serotonin 1e (5-HT1e) Receptor, Human	42
5HT1F_HUMAN	P30939	CHEMBL1805	Serotonin 1f (5-HT1f) Receptor, Human	72
5HT2A_HUMAN	P28223	CHEMBL224	Serotonin 2a (5-HT2a) Receptor, Human	406
5HT2B_HUMAN	P41595	CHEMBL1833	Serotonin 2b (5-HT2b) Receptor, Human	172
5HT2C_HUMAN	P28335	CHEMBL225	Serotonin 2c (5-HT2c) Receptor, Human	325
5HT4R_HUMAN	Q13639	CHEMBL1875	Serotonin 4 (5-HT4) Receptor, Human	18
5HT5A_HUMAN	P47898	CHEMBL3426	Serotonin 5a (5-HT5a) Receptor, Human	74
5HT6R_HUMAN	P50406	CHEMBL3371	Serotonin 6 (5-HT6) Receptor, Human	133
5HT7R_HUMAN	P34969	CHEMBL3155	Serotonin 7 (5-HT7) Receptor, Human	208

UniProt	Swissprot	ChEMBL	Description	Substances	Purchasable	Natural	In Man
5HT1A_MOUSE	Q64264	CHEMBL3737	Serotonin 1a (5-HT1a) Receptor, Mouse	59	11	7	7
5HT1A_RAT	P19327	CHEMBL273	Serotonin 1a (5-HT1a) Receptor, Rat	3,911	396	74	82

Clustered By Gene (0)

Clustered By Organism (3)

Code	Description	Substances	Purchasable	Natural	In Man
5HT1A-1-E	Serotonin 1a (5-HT1a) Receptor (cluster #1 Of 4), Eukaryotic	5,580	378	83	90
5HT1A-2-E	Serotonin 1a (5-HT1a) Receptor (cluster #2 Of 4), Eukaryotic	23	2	0	0
5HT1A-3-E	Serotonin 1a (5-HT1a) Receptor (cluster #3 Of 4), Eukaryotic	315	63	12	11
5HT1A-4-E	Serotonin 1a (5-HT1a) Receptor (cluster #4 Of 4), Eukaryotic	686	64	14	14

Uniprot	Swissprot	Chembl	Description	Number Shared
DRD2_HUMAN	P14416	CHEMBL217	Dopamine D2 Receptor, Human	590
5HT1D_HUMAN	P28221	CHEMBL1983	Serotonin 1d (5-HT1d) Receptor, Human	430
SC6A4_HUMAN	P31645	CHEMBL228	Serotonin Transporter, Human	430
SC6A4_RAT	P31652	CHEMBL313	Serotonin Transporter, Rat	417
5HT2A_HUMAN	P28223	CHEMBL224	Serotonin 2a (5-HT2a) Receptor, Human	405
5HT1B_HUMAN	P28222	CHEMBL1898	Serotonin 1b (5-HT1b) Receptor, Human	389
5HT2C_HUMAN	P28335	CHEMBL225	Serotonin 2c (5-HT2c) Receptor, Human	324
ADA1B_HUMAN	P35368	CHEMBL232	Alpha-1b Adrenergic Receptor, Human	288
DRD3_HUMAN	P35462	CHEMBL234	Dopamine D3 Receptor, Human	260
ADA1A_HUMAN	P35348	CHEMBL229	Alpha-1a Adrenergic Receptor, Human	257
ADA1D_HUMAN	P25100	CHEMBL223	Alpha-1d Adrenergic Receptor, Human	245
DRD2_RAT	P61169	CHEMBL339	Dopamine D2 Receptor, Rat	226
5HT7R_HUMAN	P34969	CHEMBL3155	Serotonin 7 (5-HT7) Receptor, Human	208
Z104304	Z104304	CHEMBL1907610	Adrenergic Receptor Alpha-1	201
DRD4_HUMAN	P21917	CHEMBL219	Dopamine D4 Receptor, Human	176
5HT2A_RAT	P14842	CHEMBL322	Serotonin 2a (5-HT2a) Receptor, Rat	172
5HT2B_HUMAN	P41595	CHEMBL1833	Serotonin 2b (5-HT2b) Receptor, Human	171
5HT1A_RAT	P19327	CHEMBL273	Serotonin 1a (5-HT1a) Receptor, Rat	143
KCNH2_HUMAN	Q12809	CHEMBL240	HERG, Human	134
5HT6R_HUMAN	P50406	CHEMBL3371	Serotonin 6 (5-HT6) Receptor, Human	133
ADA1A_RAT	P43140	CHEMBL319	Alpha-1a Adrenergic Receptor, Rat	103
5HT7R_RAT	P32305	CHEMBL3223	Serotonin 7 (5-HT7) Receptor, Rat	100
5HT2C_RAT	P08909	CHEMBL324	Serotonin 2c (5-HT2c) Receptor, Rat	98
DRD1_HUMAN	P21728	CHEMBL2056	Dopamine D1 Receptor, Human	95
SC6A2_HUMAN	P23975	CHEMBL222	Norepinephrine Transporter, Human	89
ADA1D_RAT	P23944	CHEMBL326	Alpha-1d Adrenergic Receptor, Rat	85
5HT1B_RAT	P28564	CHEMBL3459	Serotonin 1b (5-HT1b) Receptor, Rat	76
5HT5A_HUMAN	P47898	CHEMBL3426	Serotonin 5a (5-HT5a) Receptor, Human	74
5HT1F_HUMAN	P30939	CHEMBL1805	Serotonin 1f (5-HT1f) Receptor, Human	72
5HT3A_HUMAN	P46098	CHEMBL1899	Serotonin 3a (5-HT3a) Receptor, Human	68
SC6A3_HUMAN	Q01959	CHEMBL238	Dopamine Transporter, Human	60
HRH1_HUMAN	P35367	CHEMBL231	Histamine H1 Receptor, Human	58
DRD3_RAT	P19020	CHEMBL3138	Dopamine D3 Receptor, Rat	53
ADA2A_HUMAN	P08913	CHEMBL1867	Alpha-2a Adrenergic Receptor, Human	51
ADA1A_BOVIN	P18130	CHEMBL4892	Alpha-1a Adrenergic Receptor, Bovin	47
5HT2B_RAT	P30994	CHEMBL323	Serotonin 2b (5-HT2b) Receptor, Rat	46
5HT2A_BOVIN	Q75Z89	CHEMBL3446	Serotonin 2a (5-HT2a) Receptor, Bovin	45
SGMR1_HUMAN	Q99720	CHEMBL287	Sigma Opioid Receptor, Human	45
5HT1E_HUMAN	P28566	CHEMBL2182	Serotonin 1e (5-HT1e) Receptor, Human	42
DRD2_BOVIN	P20288	CHEMBL3998	Dopamine D2 Receptor, Bovin	42
ADA2A_RAT	P22909	CHEMBL327	Alpha-2a Adrenergic Receptor, Rat	41
ADA2B_RAT	P19328	CHEMBL266	Alpha-2b Adrenergic Receptor, Rat	40
ADA2C_RAT	P22086	CHEMBL314	Alpha-2c Adrenergic Receptor, Rat	37
DRD1_RAT	P18901	CHEMBL265	Dopamine D1 Receptor, Rat	37
5HT2A_PIG	P50129	CHEMBL2490	Serotonin 2a (5-HT2a) Receptor, Pig	36
ADA2C_HUMAN	P18825	CHEMBL1916	Alpha-2c Adrenergic Receptor, Human	35
5HT3A_RAT	P35563	CHEMBL2411	Serotonin 3a (5-HT3a) Receptor, Rat	32
5HT3B_RAT	Q9JJ16	CHEMBL3458	Serotonin 3b (5-HT3b) Receptor, Rat	32
DRD1_PIG	P50130	CHEMBL5067	Dopamine D1 Receptor, Pig	32
ADA2B_HUMAN	P18089	CHEMBL1942	Alpha-2b Adrenergic Receptor, Human	29
DRD5_HUMAN	P21918	CHEMBL1850	Dopamine D5 Receptor, Human	28
5HT1D_RAT	P28565	CHEMBL5450	Serotonin 1d (5-HT1d) Receptor, Rat	26
OPRD_RAT	P33533	CHEMBL269	Delta Opioid Receptor, Rat	26
OPRK_RAT	P34975	CHEMBL3614	Kappa Opioid Receptor, Rat	26
OPRM_RAT	P33535	CHEMBL270	Mu Opioid Receptor, Rat	26
SGMR1_RAT	Q9R0C9	CHEMBL3602	Sigma Opioid Receptor, Rat	26
5HT3B_HUMAN	O95264	CHEMBL3895	Serotonin 3b (5-HT3b) Receptor, Human	25
5HT3E_HUMAN	A5X5Y0	CHEMBL3812	Serotonin 3e (5-HT3e) Receptor, Human	25
5HT3C_HUMAN	Q8WXA8	CHEMBL4795	Serotonin 3c (5-HT3c) Receptor, Human	24
5HT3D_HUMAN	Q70Z44	CHEMBL4673	Serotonin 3d (5-HT3d) Receptor, Human	24
DRD4_RAT	P30729	CHEMBL3361	Dopamine D4 Receptor, Rat	24
5HT1F_RAT	P30940	CHEMBL4646	Serotonin 1f (5-HT1f) Receptor, Rat	23
5HT1D_PIG	P79400	CHEMBL4105	Serotonin 1d (5-HT1d) Receptor, Pig	21
ADRB2_HUMAN	P07550	CHEMBL210	Beta-2 Adrenergic Receptor, Human	18
5HT4R_HUMAN	Q13639	CHEMBL1875	Serotonin 4 (5-HT4) Receptor, Human	17
ADRB1_HUMAN	P08588	CHEMBL213	Beta-1 Adrenergic Receptor, Human	17
ERG_HUMAN	P11308	CHEMBL1293191	Transcriptional Regulator ERG, Human	17
DRD1_BOVIN	Q95136	CHEMBL2967	Dopamine D1 Receptor, Bovin	15
ACM1_HUMAN	P11229	CHEMBL216	Muscarinic Acetylcholine Receptor M1, Human	14
ADA1B_MESAU	P18841	CHEMBL3122	Alpha-1b Adrenergic Receptor, Mesau	14
DRD5_RAT	P25115	CHEMBL2281	Dopamine D5 Receptor, Rat	14
5HT1A_MOUSE	Q64264	CHEMBL3737	Serotonin 1a (5-HT1a) Receptor, Mouse	13
AA3R_HUMAN	P33765	CHEMBL256	Adenosine A3 Receptor, Human	13
OPRM_HUMAN	P35372	CHEMBL233	Mu Opioid Receptor, Human	13
HRH2_HUMAN	P25021	CHEMBL1941	Histamine H2 Receptor, Human	12
ACM2_HUMAN	P08172	CHEMBL211	Muscarinic Acetylcholine Receptor M2, Human	11
ACM4_HUMAN	P08173	CHEMBL1821	Muscarinic Acetylcholine Receptor M4, Human	11
ACM5_HUMAN	P08912	CHEMBL2035	Muscarinic Acetylcholine Receptor M5, Human	11
ADA1B_RAT	P15823	CHEMBL315	Alpha-1b Adrenergic Receptor, Rat	11
ADA2A_BOVIN	Q28838	CHEMBL4744	Alpha-2a Adrenergic Receptor, Bovin	11
OPRK_HUMAN	P41145	CHEMBL237	Kappa Opioid Receptor, Human	11
5HT5A_RAT	P35364	CHEMBL4655	Serotonin 5a (5-HT5a) Receptor, Rat	10
ACM3_HUMAN	P20309	CHEMBL245	Muscarinic Acetylcholine Receptor M3, Human	10
Q9WTR4_RAT	Q9WTR4	CHEMBL304	Norepinephrine Transporter, Rat	10
Z50597	Z50597	CHEMBL376	Rattus Norvegicus	9
DRD1_MOUSE	Q61616	CHEMBL3071	Dopamine D1 Receptor, Mouse	8
HRH1_RAT	P31390	CHEMBL4701	Histamine H1 Receptor, Rat	7
Q63380_RAT	Q63380	CHEMBL6184	Transporter, Rat	7
Z80094	Z80094	CHEMBL614558	CHO-MG (Ovarian Cells)	7
5HT4R_CAVPO	O70528	CHEMBL5017	Serotonin 4 (5-HT4) Receptor, Guinea Pig	6
HRH3_HUMAN	Q9Y5N1	CHEMBL264	Histamine H3 Receptor, Human	6
CAC1C_HUMAN	Q13936	CHEMBL1940	Voltage-gated L-type Calcium Channel Alpha-1C Subunit, Human	5
CAC1D_HUMAN	Q01668	CHEMBL4138	Voltage-gated L-type Calcium Channel Alpha-1D Subunit, Human	5
CAC1F_HUMAN	O60840	CHEMBL5593	Voltage-gated L-type Calcium Channel Alpha-1F Subunit, Human	5
CAC1S_HUMAN	Q13698	CHEMBL3805	Voltage-gated L-type Calcium Channel Alpha-1S Subunit, Human	5
CNR1_HUMAN	P21554	CHEMBL218	Cannabinoid CB1 Receptor, Human	5
OPRD_HUMAN	P41143	CHEMBL236	Delta Opioid Receptor, Human	5
SGMR1_CAVPO	Q60492	CHEMBL4153	Sigma-1 Receptor, Guinea Pig	5
5HT2A_MOUSE	P35363	CHEMBL5377	Serotonin 2a (5-HT2a) Receptor, Mouse	4
5HT2B_MOUSE	Q02152	CHEMBL2583	Serotonin 2b (5-HT2b) Receptor, Mouse	4
5HT2C_MOUSE	P34968	CHEMBL3006	Serotonin 2c (5-HT2c) Receptor, Mouse	4
5HT3A_MOUSE	P23979	CHEMBL4972	Serotonin 3a (5-HT3a) Receptor, Mouse	4
HRH4_HUMAN	Q9H3N8	CHEMBL3759	Histamine H4 Receptor, Human	4
MDR1_HUMAN	P08183	CHEMBL4302	P-glycoprotein 1, Human	4
SCN2A_HUMAN	Q99250	CHEMBL4187	Sodium Channel Protein Type II Alpha Subunit, Human	4
SCN3A_HUMAN	Q9NY46	CHEMBL5163	Sodium Channel Protein Type III Alpha Subunit, Human	4
5HT1D_MOUSE	Q61224	CHEMBL4297	Serotonin 1d (5-HT1d) Receptor, Mouse	3
5HT3B_MOUSE	Q9JHJ5	CHEMBL3781	Serotonin 3b (5-HT3b) Receptor, Mouse	3
5HT4R_RAT	Q62758	CHEMBL4317	Serotonin 4 (5-HT4) Receptor, Rat	3
5HT5B_RAT	P35365	CHEMBL2619	Serotonin 5b (5-HT5b) Receptor, Rat	3
AA1R_HUMAN	P30542	CHEMBL226	Adenosine A1 Receptor, Human	3
AA2AR_HUMAN	P29274	CHEMBL251	Adenosine A2a Receptor, Human	3
ACM1_RAT	P08482	CHEMBL276	Muscarinic Acetylcholine Receptor M1, Rat	3
ADCY3_RAT	P21932	CHEMBL4864	Adenylate Cyclase Type III, Rat	3
ADCY5_RAT	Q04400	CHEMBL2880	Adenylate Cyclase Type V, Rat	3
ADRB1_RAT	P18090	CHEMBL3252	Beta-1 Adrenergic Receptor, Rat	3
GNRHR_HUMAN	P30968	CHEMBL1855	Gonadotropin-releasing Hormone Receptor, Human	3
HRH1_CAVPO	P31389	CHEMBL3943	Histamine H1 Receptor, Guinea Pig	3
HRH3_RAT	Q9QYN8	CHEMBL4124	Histamine H3 Receptor, Rat	3
HRH4_RAT	Q91ZY1	CHEMBL4468	Histamine H4 Receptor, Rat	3
MTR1A_HUMAN	P48039	CHEMBL1945	Melatonin Receptor 1A, Human	3
NK2R_HUMAN	P21452	CHEMBL2327	Neurokinin 2 Receptor, Human	3
SCN1A_HUMAN	P35498	CHEMBL1845	Sodium Channel Protein Type I Alpha Subunit, Human	3
SCN8A_HUMAN	Q9UQD0	CHEMBL5202	Sodium Channel Protein Type VIII Alpha Subunit, Human	3
Z104303	Z104303	CHEMBL1907609	Muscarinic Acetylcholine Receptor	3
5HT5A_MOUSE	P30966	CHEMBL3597	Serotonin 5a (5-HT5a) Receptor, Mouse	2
5HT6R_RAT	P31388	CHEMBL3372	Serotonin 6 (5-HT6) Receptor, Rat	2
ACES_HUMAN	P22303	CHEMBL220	Acetylcholinesterase, Human	2
ACM2_RAT	P10980	CHEMBL309	Muscarinic Acetylcholine Receptor M2, Rat	2
ADRB3_HUMAN	P13945	CHEMBL246	Beta-3 Adrenergic Receptor, Human	2
ADRB3_RAT	P26255	CHEMBL4031	Beta-3 Adrenergic Receptor, Rat	2
AOFA_HUMAN	P21397	CHEMBL1951	Monoamine Oxidase A, Human	2
DRD2_CHLAE	P52702	CHEMBL5456	Dopamine D2 Receptor, Chlae	2
DRD2_MOUSE	P61168	CHEMBL3427	Dopamine D2 Receptor, Mouse	2
EBP_CAVPO	Q60490	CHEMBL5525	3-beta-hydroxysteroid-delta(8),delta(7)-isomerase, Guinea Pig	2
EDNRA_HUMAN	P25101	CHEMBL252	Endothelin Receptor ET-A, Human	2
EPYC_HUMAN	Q99645	CHEMBL2080	Small Chondroitin/dermatan Sulfate Proteoglycan, Human	2
GASR_HUMAN	P32239	CHEMBL298	Cholecystokinin B Receptor, Human	2
GBRA1_HUMAN	P14867	CHEMBL1962	GABA Receptor Alpha-1 Subunit, Human	2
GBRA2_HUMAN	P47869	CHEMBL4956	GABA Receptor Alpha-2 Subunit, Human	2
GBRA3_HUMAN	P34903	CHEMBL3026	GABA Receptor Alpha-3 Subunit, Human	2
GBRA4_HUMAN	P48169	CHEMBL2472	GABA Receptor Alpha-4 Subunit, Human	2
GBRA5_HUMAN	P31644	CHEMBL5112	GABA Receptor Alpha-5 Subunit, Human	2
GBRA6_HUMAN	Q16445	CHEMBL2579	GABA Receptor Alpha-6 Subunit, Human	2
GBRB1_HUMAN	P18505	CHEMBL4558	GABA Receptor Beta-1 Subunit, Human	2
GBRB2_HUMAN	P47870	CHEMBL1920	GABA Receptor Beta-2 Subunit, Human	2
GBRB3_HUMAN	P28472	CHEMBL1847	GABA Receptor Beta-3 Subunit, Human	2
GBRD_HUMAN	O14764	CHEMBL3591	GABA Receptor Delta Subunit, Human	2
GBRE_HUMAN	P78334	CHEMBL4635	GABA Receptor Epsilon Subunit, Human	2
GBRG1_HUMAN	Q8N1C3	CHEMBL4044	GABA Receptor Gamma-1 Subunit, Human	2
GBRG2_HUMAN	P18507	CHEMBL1788	GABA Receptor Gamma-2 Subunit, Human	2
GBRG3_HUMAN	Q99928	CHEMBL2739	GABA Receptor Gamma-3 Subunit, Human	2
GBRP_HUMAN	O00591	CHEMBL3506	GABA Receptor Pi Subunit, Human	2
GBRT_HUMAN	Q9UN88	CHEMBL2843	GABA Receptor Theta Subunit, Human	2
GCR_HUMAN	P04150	CHEMBL2034	Glucocorticoid Receptor, Human	2
HRH2_RAT	P25102	CHEMBL4654	Histamine H2 Receptor, Rat	2
LYN_HUMAN	P07948	CHEMBL3905	Tyrosine-protein Kinase Lyn, Human	2
MC4R_HUMAN	P32245	CHEMBL259	Melanocortin Receptor 4, Human	2
MK14_HUMAN	Q16539	CHEMBL260	MAP Kinase P38 Alpha, Human	2
MT3_HUMAN	P25713	CHEMBL1250357	Metallothionein-3, Human	2
NISCH_HUMAN	Q9Y2I1	CHEMBL3923	Nischarin, Human	2
NK1R_HUMAN	P25103	CHEMBL249	Neurokinin 1 Receptor, Human	2
NPY1R_HUMAN	P25929	CHEMBL4777	Neuropeptide Y Receptor Type 1, Human	2
NTR1_HUMAN	P30989	CHEMBL4123	Neurotensin Receptor 1, Human	2
SC5A7_HUMAN	Q9GZV3	CHEMBL4507	High-affinity Choline Transporter, Human	2
SC6A3_RAT	P23977	CHEMBL338	Dopamine Transporter, Rat	2
SMO_HUMAN	Q99835	CHEMBL5971	Smoothened Homolog, Human	2
V1AR_HUMAN	P37288	CHEMBL1889	Vasopressin V1a Receptor, Human	2
VACHT_HUMAN	Q16572	CHEMBL4767	Vesicular Acetylcholine Transporter, Human	2
Z100491	Z100491	CHEMBL613288	Sigma 2 Receptor	2
Z104283	Z104283	CHEMBL1907589	Neuronal Acetylcholine Receptor; Alpha4/beta2	2
Z81247	Z81247	CHEMBL399	HeLa (Cervical Adenocarcinoma Cells)	2
ACM3_RAT	P08483	CHEMBL320	Muscarinic Acetylcholine Receptor M3, Rat	1
ACM4_RAT	P08485	CHEMBL317	Muscarinic Acetylcholine Receptor M4, Rat	1
ACM5_RAT	P08911	CHEMBL277	Muscarinic Acetylcholine Receptor M5, Rat	1
ADA2B_BOVIN	O77700	CHEMBL3523	Alpha-2b Adrenergic Receptor, Bovin	1
ADCY1_HUMAN	Q08828	CHEMBL2899	Brain Adenylate Cyclase 1, Human	1
ADCY2_HUMAN	Q08462	CHEMBL3760	Adenylate Cyclase Type II, Human	1
ADCY2_RAT	P26769	CHEMBL2958	Adenylate Cyclase Type II, Rat	1
ADCY4_RAT	P26770	CHEMBL2879	Adenylate Cyclase Type IV, Rat	1
ADCY6_RAT	Q03343	CHEMBL2975	Adenylate Cyclase Type VI, Rat	1
ADCY8_HUMAN	P40145	CHEMBL2960	Adenylate Cyclase Type VIII, Human	1
ADCY8_RAT	P40146	CHEMBL3082	Adenylate Cyclase Type VIII, Rat	1
ADRB2_CANFA	P54833	CHEMBL2289	Beta-2 Adrenergic Receptor, Canine	1
AP2S1_RAT	P62744	CHEMBL1697667	AP-2 Complex Subunit Sigma, Rat	1
CAC1C_RAT	P22002	CHEMBL3762	Voltage-gated L-type Calcium Channel Alpha-1C Subunit, Rat	1
CAC1D_RAT	P27732	CHEMBL4132	Voltage-gated L-type Calcium Channel Alpha-1D Subunit, Rat	1
CALM_HUMAN	P62158	CHEMBL6093	Calmodulin, Human	1
CCKAR_HUMAN	P32238	CHEMBL1901	Cholecystokinin A Receptor, Human	1
CCNA2_HUMAN	P20248	CHEMBL2582	Cyclin A2, Human	1
CCNB1_HUMAN	P14635	CHEMBL2412	G2/mitotic-specific Cyclin B1, Human	1
CCNB2_HUMAN	O95067	CHEMBL3723	G2/mitotic-specific Cyclin B2, Human	1
CCNB3_HUMAN	Q8WWL7	CHEMBL3606	G2/mitotic-specific Cyclin B3, Human	1
CCNT1_HUMAN	O60563	CHEMBL2108	Cyclin T1, Human	1
CDK1_HUMAN	P06493	CHEMBL308	Cyclin-dependent Kinase 1, Human	1
CDK2_HUMAN	P24941	CHEMBL301	Cyclin-dependent Kinase 2, Human	1
CDK5_HUMAN	Q00535	CHEMBL4036	Cyclin-dependent Kinase 5, Human	1
CDK9_HUMAN	P50750	CHEMBL3116	Cyclin-dependent Kinase 9, Human	1
CNR2_HUMAN	P34972	CHEMBL253	Cannabinoid CB2 Receptor, Human	1
CNR2_MOUSE	P47936	CHEMBL5373	Cannabinoid CB2 Receptor, Mouse	1
CXCR3_HUMAN	P49682	CHEMBL4441	C-X-C Chemokine Receptor Type 3, Human	1
CXCR3_MOUSE	O88410	CHEMBL5200	C-X-C Chemokine Receptor Type 3, Mouse	1
D4A3N4_RAT	D4A3N4	CHEMBL2679	Brain Adenylate Cyclase 1, Rat	1
DRD4_MOUSE	P51436	CHEMBL2574	Dopamine D4 Receptor, Mouse	1
EBP_HUMAN	Q15125	CHEMBL4931	3-beta-hydroxysteroid-delta(8),delta(7)-isomerase, Human	1
ERG2_YEAST	P32352	CHEMBL3224	C-8 Sterol Isomerase, Yeast	1
FAAH1_MOUSE	O08914	CHEMBL3455	Anandamide Amidohydrolase, Mouse	1
GSK3B_HUMAN	P49841	CHEMBL262	Glycogen Synthase Kinase-3 Beta, Human	1
HRH2_CAVPO	P47747	CHEMBL2882	Histamine H2 Receptor, Guinea Pig	1
MCHR1_HUMAN	Q99705	CHEMBL344	Melanin-concentrating Hormone Receptor 1, Human	1
NMD3A_HUMAN	Q8TCU5	CHEMBL4787	Glutamate [NMDA] Receptor Subunit 3A, Human	1
NMD3B_HUMAN	O60391	CHEMBL2913	Glutamate [NMDA] Receptor Subunit 3B, Human	1
NMDE1_HUMAN	Q12879	CHEMBL1972	Glutamate [NMDA] Receptor Subunit Epsilon 1, Human	1
NMDE2_HUMAN	Q13224	CHEMBL1904	Glutamate [NMDA] Receptor Subunit Epsilon 2, Human	1
NMDE3_HUMAN	Q14957	CHEMBL4109	Glutamate [NMDA] Receptor Subunit Epsilon 3, Human	1
NMDE4_HUMAN	O15399	CHEMBL2591	Glutamate [NMDA] Receptor Subunit Epsilon 4, Human	1
NMDZ1_HUMAN	Q05586	CHEMBL2015	Glutamate (NMDA) Receptor Subunit Zeta 1, Human	1
NOS1_HUMAN	P29475	CHEMBL3568	Nitric-oxide Synthase, Brain, Human	1
NOS1_RAT	P29476	CHEMBL3048	Nitric-oxide Synthase, Brain, Rat	1
NOS3_HUMAN	P29474	CHEMBL4803	Nitric-oxide Synthase, Endothelial, Human	1
NPY5R_HUMAN	Q15761	CHEMBL4561	Neuropeptide Y Receptor Type 5, Human	1
PDR5_YEAST	P33302	CHEMBL1697658	Pleiotropic ABC Efflux Transporter Of Multiple Drugs, Yeast	1
PRIO_HUMAN	P04156	CHEMBL4869	Prion Protein, Human	1
Q4U254_9ENTO	Q4U254	CHEMBL2857	Human Rhinovirus A Protease, 9ento	1
Q72874_9HIV1	Q72874	CHEMBL243	Human Immunodeficiency Virus Type 1 Protease, 9hiv1	1
Q8CFM9_RAT	Q8CFM9	CHEMBL3940	Adenylate Cyclase Type VII, Rat	1
SC6A3_BOVIN	P27922	CHEMBL2986	Dopamine Transporter, Bovin	1
SC6A3_MACFA	Q9GJT6	CHEMBL5032	Dopamine Transporter, Macfa	1
SC6A4_MOUSE	Q60857	CHEMBL4642	Serotonin Transporter, Mouse	1
SCN5A_HUMAN	Q14524	CHEMBL1980	Sodium Channel Protein Type V Alpha Subunit, Human	1
SCN9A_HUMAN	Q15858	CHEMBL4296	Sodium Channel Protein Type IX Alpha Subunit, Human	1
SCNAA_HUMAN	Q9Y5Y9	CHEMBL5451	Sodium Channel Protein Type X Alpha Subunit, Human	1
SCNAA_MOUSE	Q6QIY3	CHEMBL5158	Sodium Channel Protein Type 10 Subunit Alpha, Mouse	1
SCNAA_RAT	Q62968	CHEMBL4017	Sodium Channel Protein Type X Alpha Subunit, Rat	1
TRPV1_RAT	O35433	CHEMBL5102	Vanilloid Receptor, Rat	1
TSPOA_HUMAN	P30536	CHEMBL5742	Translocator Protein, Human	1
TSPOB_HUMAN	B1AH88	CHEMBL5139	Peripheral-type Benzodiazepine Receptor, Human	1
TYTR_TRYCR	P28593	CHEMBL5131	Trypanothione Reductase, Trycr	1
UR2R_HUMAN	Q9UKP6	CHEMBL3764	Urotensin II Receptor, Human	1
Z100251	Z100251	CHEMBL612442	Monoclonal Antibody (mAb) 2E2	1
Z104294	Z104294	CHEMBL1907600	Cyclin-dependent Kinase 5/CDK5 Activator 1	1
Z104302	Z104302	CHEMBL1907608	Glutamate NMDA Receptor	1
Z50425	Z50425	CHEMBL364	Plasmodium Falciparum	1
Z50588	Z50588	CHEMBL373	Canis Familiaris	1
Z50592	Z50592	CHEMBL374	Oryctolagus Cuniculus	1
Z50796	Z50796	CHEMBL614874	Monkey	1
Z80088	Z80088	CHEMBL613853	CHO (Ovarian Cells)	1
Z80334	Z80334	CHEMBL613828	NG108-15 (Neuroblastoma-glioma Hybrid Cells)	1