UCSF

ChEMBL DrugStore

Binding 10μM Binding 1μM Functional 10μM ADME/T 10μM

Binding 10μM Targets with Highest Number of Available Compounds (1787 in total)

Name (Uniprot) Swissprot ChEMBL Description Size Browse Download (Annotations)
KCNH2_HUMAN Q12809 CHEMBL240 HERG 151 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD2_RAT P61169 CHEMBL339 Dopamine D2 receptor 105 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104304 Z104304 CHEMBL1907610 Adrenergic receptor alpha-1 91 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2A_RAT P14842 CHEMBL322 Serotonin 2a (5-HT2a) receptor 84 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2B_RAT P19328 CHEMBL266 Alpha-2b adrenergic receptor 83 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2A_RAT P22909 CHEMBL327 Alpha-2a adrenergic receptor 82 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2C_RAT P22086 CHEMBL314 Alpha-2c adrenergic receptor 78 Annotations Catalogs SMILES SDF Mol2 Flexibase
SCN2A_HUMAN Q99250 CHEMBL4187 Sodium channel protein type II alpha subunit 74 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2C_RAT P08909 CHEMBL324 Serotonin 2c (5-HT2c) receptor 72 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD2_HUMAN P14416 CHEMBL217 Dopamine D2 receptor 72 Annotations Catalogs SMILES SDF Mol2 Flexibase
SCN1A_HUMAN P35498 CHEMBL1845 Sodium channel protein type I alpha subunit 71 Annotations Catalogs SMILES SDF Mol2 Flexibase
SCN3A_HUMAN Q9NY46 CHEMBL5163 Sodium channel protein type III alpha subunit 71 Annotations Catalogs SMILES SDF Mol2 Flexibase
SCN8A_HUMAN Q9UQD0 CHEMBL5202 Sodium channel protein type VIII alpha subunit 71 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1A_RAT P19327 CHEMBL273 Serotonin 1a (5-HT1a) receptor 69 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2B_RAT P30994 CHEMBL323 Serotonin 2b (5-HT2b) receptor 68 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD1_RAT P18901 CHEMBL265 Dopamine D1 receptor 59 Annotations Catalogs SMILES SDF Mol2 Flexibase
SC6A4_HUMAN P31645 CHEMBL228 Serotonin transporter 56 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH2_HUMAN P00918 CHEMBL205 Carbonic anhydrase II 55 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD3_HUMAN P35462 CHEMBL234 Dopamine D3 receptor 55 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRM_RAT P33535 CHEMBL270 Mu opioid receptor 54 Annotations Catalogs SMILES SDF Mol2 Flexibase
SC6A2_HUMAN P23975 CHEMBL222 Norepinephrine transporter 54 Annotations Catalogs SMILES SDF Mol2 Flexibase
SGMR1_HUMAN Q99720 CHEMBL287 Sigma opioid receptor 53 Annotations Catalogs SMILES SDF Mol2 Flexibase
SC6A3_RAT P23977 CHEMBL338 Dopamine transporter 52 Annotations Catalogs SMILES SDF Mol2 Flexibase
SC6A4_RAT P31652 CHEMBL313 Serotonin transporter 52 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD3_RAT P19020 CHEMBL3138 Dopamine D3 receptor 51 Annotations Catalogs SMILES SDF Mol2 Flexibase
SC6A3_HUMAN Q01959 CHEMBL238 Dopamine transporter 50 Annotations Catalogs SMILES SDF Mol2 Flexibase
SGMR1_RAT Q9R0C9 CHEMBL3602 Sigma opioid receptor 50 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1A_HUMAN P08908 CHEMBL214 Serotonin 1a (5-HT1a) receptor 49 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1A_HUMAN P35348 CHEMBL229 Alpha-1a adrenergic receptor 49 Annotations Catalogs SMILES SDF Mol2 Flexibase
HRH1_HUMAN P35367 CHEMBL231 Histamine H1 receptor 49 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q9WTR4_RAT Q9WTR4 CHEMBL304 Norepinephrine transporter 49 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1B_HUMAN P35368 CHEMBL232 Alpha-1b adrenergic receptor 48 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2A_HUMAN P08913 CHEMBL1867 Alpha-2a adrenergic receptor 48 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRM_HUMAN P35372 CHEMBL233 Mu opioid receptor 48 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRK_HUMAN P41145 CHEMBL237 Kappa opioid receptor 47 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2C_HUMAN P18825 CHEMBL1916 Alpha-2c adrenergic receptor 45 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1B_RAT P28564 CHEMBL3459 Serotonin 1b (5-HT1b) receptor 44 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1D_HUMAN P25100 CHEMBL223 Alpha-1d adrenergic receptor 44 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD4_RAT P30729 CHEMBL3361 Dopamine D4 receptor 43 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH2_HUMAN P35354 CHEMBL230 Cyclooxygenase-2 43 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB2_HUMAN P07550 CHEMBL210 Beta-2 adrenergic receptor 41 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD4_HUMAN P21917 CHEMBL219 Dopamine D4 receptor 41 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD5_RAT P25115 CHEMBL2281 Dopamine D5 receptor 41 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH1_HUMAN P00915 CHEMBL261 Carbonic anhydrase I 40 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM1_HUMAN P11229 CHEMBL216 Muscarinic acetylcholine receptor M1 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRD_RAT P33533 CHEMBL269 Delta opioid receptor 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z50597 Z50597 CHEMBL376 Rattus norvegicus 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2A_HUMAN P28223 CHEMBL224 Serotonin 2a (5-HT2a) receptor 38 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1D_RAT P28565 CHEMBL5450 Serotonin 1d (5-HT1d) receptor 37 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2C_HUMAN P28335 CHEMBL225 Serotonin 2c (5-HT2c) receptor 37 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2B_HUMAN P18089 CHEMBL1942 Alpha-2b adrenergic receptor 37 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH12_HUMAN O43570 CHEMBL3242 Carbonic anhydrase XII 37 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH9_HUMAN Q16790 CHEMBL3594 Carbonic anhydrase IX 37 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH6_HUMAN P23280 CHEMBL3025 Carbonic anhydrase VI 36 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRD_HUMAN P41143 CHEMBL236 Delta opioid receptor 36 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRK_RAT P34975 CHEMBL3614 Kappa opioid receptor 36 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH1_HUMAN P23219 CHEMBL221 Cyclooxygenase-1 36 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104301 Z104301 CHEMBL1907607 GABA-A receptor; anion channel 36 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1F_RAT P30940 CHEMBL4646 Serotonin 1f (5-HT1f) receptor 35 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA3R_HUMAN P33765 CHEMBL256 Adenosine A3 receptor 34 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM2_HUMAN P08172 CHEMBL211 Muscarinic acetylcholine receptor M2 34 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1A_RAT P43140 CHEMBL319 Alpha-1a adrenergic receptor 34 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH4_HUMAN P22748 CHEMBL3729 Carbonic anhydrase IV 34 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACES_HUMAN P22303 CHEMBL220 Acetylcholinesterase 32 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM3_HUMAN P20309 CHEMBL245 Muscarinic acetylcholine receptor M3 31 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM2_RAT P10980 CHEMBL309 Muscarinic acetylcholine receptor M2 30 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH5A_HUMAN P35218 CHEMBL4789 Carbonic anhydrase VA 30 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH7_HUMAN P43166 CHEMBL2326 Carbonic anhydrase VII 30 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104302 Z104302 CHEMBL1907608 Glutamate NMDA receptor 30 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104303 Z104303 CHEMBL1907609 Muscarinic acetylcholine receptor 30 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACE_HUMAN P12821 CHEMBL1808 Angiotensin-converting enzyme 29 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH5B_HUMAN Q9Y2D0 CHEMBL3969 Carbonic anhydrase VB 29 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1D_RAT P23944 CHEMBL326 Alpha-1d adrenergic receptor 28 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM1_RAT P08482 CHEMBL276 Muscarinic acetylcholine receptor M1 27 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH14_HUMAN Q9ULX7 CHEMBL3510 Carbonic anhydrase XIV 27 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD1_HUMAN P21728 CHEMBL2056 Dopamine D1 receptor 27 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB1_HUMAN P08588 CHEMBL213 Beta-1 adrenergic receptor 26 Annotations Catalogs SMILES SDF Mol2 Flexibase
AOFB_HUMAN P27338 CHEMBL2039 Monoamine oxidase B 26 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH15_MOUSE Q99N23 CHEMBL5973 Carbonic anhydrase 15 26 Annotations Catalogs SMILES SDF Mol2 Flexibase
CP19A_HUMAN P11511 CHEMBL1978 Cytochrome P450 19A1 26 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE3A_HUMAN Q14432 CHEMBL241 Phosphodiesterase 3A 26 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE3B_HUMAN Q13370 CHEMBL290 Phosphodiesterase 3B 26 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE4B_HUMAN Q07343 CHEMBL275 Phosphodiesterase 4B 26 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT7R_HUMAN P34969 CHEMBL3155 Serotonin 7 (5-HT7) receptor 25 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE4A_HUMAN P27815 CHEMBL254 Phosphodiesterase 4A 25 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE4D_HUMAN Q08499 CHEMBL288 Phosphodiesterase 4D 25 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB1_RAT P18090 CHEMBL3252 Beta-1 adrenergic receptor 24 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD2_BOVIN P20288 CHEMBL3998 Dopamine D2 receptor 24 Annotations Catalogs SMILES SDF Mol2 Flexibase
ESR1_HUMAN P03372 CHEMBL206 Estrogen receptor alpha 24 Annotations Catalogs SMILES SDF Mol2 Flexibase
KIT_HUMAN P10721 CHEMBL1936 Stem cell growth factor receptor 24 Annotations Catalogs SMILES SDF Mol2 Flexibase
VGFR2_HUMAN P35968 CHEMBL279 Vascular endothelial growth factor receptor 2 24 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT6R_HUMAN P50406 CHEMBL3371 Serotonin 6 (5-HT6) receptor 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT7R_RAT P32305 CHEMBL3223 Serotonin 7 (5-HT7) receptor 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM4_HUMAN P08173 CHEMBL1821 Muscarinic acetylcholine receptor M4 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1A_BOVIN P18130 CHEMBL4892 Alpha-1a adrenergic receptor 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
ESR2_HUMAN Q92731 CHEMBL242 Estrogen receptor beta 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
LOX5_RAT P12527 CHEMBL312 Arachidonate 5-lipoxygenase 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE4C_HUMAN Q08493 CHEMBL291 Phosphodiesterase 4C 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q63380_RAT Q63380 CHEMBL6184 Transporter 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q72874_9HIV1 Q72874 CHEMBL243 Human immunodeficiency virus type 1 protease 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1B_RAT P15823 CHEMBL315 Alpha-1b adrenergic receptor 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH13_MOUSE Q9D6N1 CHEMBL2186 Carbonic anhydrase XIII 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
DYR_HUMAN P00374 CHEMBL202 Dihydrofolate reductase 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
HRH1_RAT P31390 CHEMBL4701 Histamine H1 receptor 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3A_HUMAN P46098 CHEMBL1899 Serotonin 3a (5-HT3a) receptor 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
ABL1_HUMAN P00519 CHEMBL1862 Tyrosine-protein kinase ABL 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAC1C_RAT P22002 CHEMBL3762 Voltage-gated L-type calcium channel alpha-1C subunit 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
ERG2_YEAST P32352 CHEMBL3224 C-8 sterol isomerase 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
LCK_HUMAN P06239 CHEMBL258 Tyrosine-protein kinase LCK 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
MDR1_HUMAN P08183 CHEMBL4302 P-glycoprotein 1 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGFRB_HUMAN P09619 CHEMBL1913 Platelet-derived growth factor receptor beta 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3A_RAT P35563 CHEMBL2411 Serotonin 3a (5-HT3a) receptor 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3B_RAT Q9JJ16 CHEMBL3458 Serotonin 3b (5-HT3b) receptor 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM5_HUMAN P08912 CHEMBL2035 Muscarinic acetylcholine receptor M5 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB3_RAT P26255 CHEMBL4031 Beta-3 adrenergic receptor 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
EGFR_HUMAN P00533 CHEMBL203 Epidermal growth factor receptor erbB1 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q72547_9HIV1 Q72547 CHEMBL247 Human immunodeficiency virus type 1 reverse transcriptase 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2B_HUMAN P41595 CHEMBL1833 Serotonin 2b (5-HT2b) receptor 19 Annotations Catalogs SMILES SDF Mol2 Flexibase
ANDR_HUMAN P10275 CHEMBL1871 Androgen Receptor 19 Annotations Catalogs SMILES SDF Mol2 Flexibase
B5SU02_9CNID B5SU02 CHEMBL1075028 Alpha carbonic anhydrase 19 Annotations Catalogs SMILES SDF Mol2 Flexibase
CHLE_HUMAN P06276 CHEMBL1914 Butyrylcholinesterase 19 Annotations Catalogs SMILES SDF Mol2 Flexibase
EBP_HUMAN Q15125 CHEMBL4931 3-beta-hydroxysteroid-delta(8),delta(7)-isomerase 19 Annotations Catalogs SMILES SDF Mol2 Flexibase
FLT3_HUMAN P36888 CHEMBL1974 Tyrosine-protein kinase receptor FLT3 19 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA1_HUMAN P14867 CHEMBL1962 GABA receptor alpha-1 subunit 19 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGFRA_HUMAN P16234 CHEMBL2007 Platelet-derived growth factor receptor alpha 19 Annotations Catalogs SMILES SDF Mol2 Flexibase
C0IX24_9CNID C0IX24 CHEMBL1649055 Carbonic anhydrase 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA2_HUMAN P47869 CHEMBL4956 GABA receptor alpha-2 subunit 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRG2_HUMAN P18507 CHEMBL1788 GABA receptor gamma-2 subunit 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMD3A_HUMAN Q8TCU5 CHEMBL4787 Glutamate [NMDA] receptor subunit 3A 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMD3B_HUMAN O60391 CHEMBL2913 Glutamate [NMDA] receptor subunit 3B 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE1_HUMAN Q12879 CHEMBL1972 Glutamate [NMDA] receptor subunit epsilon 1 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE2_HUMAN Q13224 CHEMBL1904 Glutamate [NMDA] receptor subunit epsilon 2 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE3_HUMAN Q14957 CHEMBL4109 Glutamate [NMDA] receptor subunit epsilon 3 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE4_HUMAN O15399 CHEMBL2591 Glutamate [NMDA] receptor subunit epsilon 4 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDZ1_HUMAN Q05586 CHEMBL2015 Glutamate (NMDA) receptor subunit zeta 1 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH1_RAT Q63921 CHEMBL4042 Cyclooxygenase-1 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q5AJ71_CANAL Q5AJ71 CHEMBL5337 Carbonic anhydrase 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAC1D_RAT P27732 CHEMBL4132 Voltage-gated L-type calcium channel alpha-1D subunit 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
CSF1R_HUMAN P07333 CHEMBL1844 Macrophage colony stimulating factor receptor 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
FRK_HUMAN P42685 CHEMBL4223 Tyrosine-protein kinase FRK 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA3_HUMAN P34903 CHEMBL3026 GABA receptor alpha-3 subunit 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
PPARG_HUMAN P37231 CHEMBL235 Peroxisome proliferator-activated receptor gamma 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
STK10_HUMAN O94804 CHEMBL3981 Serine/threonine-protein kinase 10 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
THRB_HUMAN P00734 CHEMBL204 Thrombin 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1B_HUMAN P28222 CHEMBL1898 Serotonin 1b (5-HT1b) receptor 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1D_HUMAN P28221 CHEMBL1983 Serotonin 1d (5-HT1d) receptor 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA2AR_HUMAN P29274 CHEMBL251 Adenosine A2a receptor 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM3_RAT P08483 CHEMBL320 Muscarinic acetylcholine receptor M3 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
ALDR_HUMAN P15121 CHEMBL1900 Aldose reductase 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH3_HUMAN P07451 CHEMBL2885 Carbonic anhydrase III 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
DDR1_HUMAN Q08345 CHEMBL5319 Epithelial discoidin domain-containing receptor 1 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
LYN_HUMAN P07948 CHEMBL3905 Tyrosine-protein kinase Lyn 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH2_RAT P35355 CHEMBL2977 Cyclooxygenase-2 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
SRC_HUMAN P12931 CHEMBL267 Tyrosine-protein kinase SRC 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
VGFR1_HUMAN P17948 CHEMBL1868 Vascular endothelial growth factor receptor 1 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT4R_RAT Q62758 CHEMBL4317 Serotonin 4 (5-HT4) receptor 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB2_CANFA P54833 CHEMBL2289 Beta-2 adrenergic receptor 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
AOFB_RAT P19643 CHEMBL2993 Monoamine oxidase B 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAN_YEAST P53615 CHEMBL5931 Carbonic anhydrase 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
CHLE_HORSE P81908 CHEMBL5763 Cholinesterase 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
CYNT_MYCTU O53573 CHEMBL6068 Carbonic anhydrase 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD5_HUMAN P21918 CHEMBL1850 Dopamine D5 receptor 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA5_HUMAN P31644 CHEMBL5112 GABA receptor alpha-5 subunit 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
RET_HUMAN P07949 CHEMBL2041 Tyrosine-protein kinase receptor RET 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
SLK_HUMAN Q9H2G2 CHEMBL4202 Serine/threonine-protein kinase 2 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
Y1284_MYCTU P64797 CHEMBL5631 Uncharacterized protein Rv1284/MT1322 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA1R_RAT P25099 CHEMBL318 Adenosine A1 receptor 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
CYNT_HELPY O24855 CHEMBL4211 Carbonic anhydrase 1 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD1_BOVIN Q95136 CHEMBL2967 Dopamine D1 receptor 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
FABPL_RAT P02692 CHEMBL5738 Fatty acid-binding protein, liver 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRB3_HUMAN P28472 CHEMBL1847 GABA receptor beta-3 subunit 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
VGFR3_HUMAN P35916 CHEMBL1955 Vascular endothelial growth factor receptor 3 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA2AR_RAT P30543 CHEMBL302 Adenosine A2a receptor 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2A_BOVIN Q28838 CHEMBL4744 Alpha-2a adrenergic receptor 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
AMPC_ECOLI P00811 CHEMBL2026 Beta-lactamase 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH4_BOVIN Q95323 CHEMBL281 Carbonic anhydrase IV 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
CTRO_HUMAN O14578 CHEMBL5579 Citron Rho-interacting kinase 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
FGFR1_HUMAN P11362 CHEMBL3650 Fibroblast growth factor receptor 1 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRB2_HUMAN P47870 CHEMBL1920 GABA receptor beta-2 subunit 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
JAK3_HUMAN P52333 CHEMBL2148 Tyrosine-protein kinase JAK3 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
LOX5_HUMAN P09917 CHEMBL215 Arachidonate 5-lipoxygenase 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
M4K5_HUMAN Q9Y4K4 CHEMBL4852 Mitogen-activated protein kinase kinase kinase kinase 5 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
NISCH_HUMAN Q9Y2I1 CHEMBL3923 Nischarin 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
PPARA_HUMAN Q07869 CHEMBL239 Peroxisome proliferator-activated receptor alpha 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA1R_HUMAN P30542 CHEMBL226 Adenosine A1 receptor 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
ALK_HUMAN Q9UM73 CHEMBL4247 ALK tyrosine kinase receptor 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
AOFA_RAT P21396 CHEMBL3358 Monoamine oxidase A 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
BLK_HUMAN P51451 CHEMBL2250 Tyrosine-protein kinase BLK 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH13_HUMAN Q8N1Q1 CHEMBL3912 Carbonic anhydrase XIII 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
CLTR1_HUMAN Q9Y271 CHEMBL1798 Cysteinyl leukotriene receptor 1 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
CLTR2_HUMAN Q9NS75 CHEMBL4330 Cysteinyl leukotriene receptor 2 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
CP17A_HUMAN P05093 CHEMBL3522 Cytochrome P450 17A1 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
DYR_MOUSE P00375 CHEMBL4564 Dihydrofolate reductase 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
FA10_HUMAN P00742 CHEMBL244 Coagulation factor X 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
GAK_HUMAN O14976 CHEMBL4355 Serine/threonine-protein kinase GAK 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE2_RAT Q00960 CHEMBL311 Glutamate [NMDA] receptor subunit epsilon 2 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRM_MOUSE P42866 CHEMBL2858 Mu opioid receptor 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH1_BOVIN O62664 CHEMBL2860 Cyclooxygenase-1 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH1_SHEEP P05979 CHEMBL2949 Cyclooxygenase-1 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH2_SHEEP P79208 CHEMBL4102 Cyclooxygenase-2 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT4R_HUMAN Q13639 CHEMBL1875 Serotonin 4 (5-HT4) receptor 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACES_RAT P37136 CHEMBL3199 Acetylcholinesterase 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM4_RAT P08485 CHEMBL317 Muscarinic acetylcholine receptor M4 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
AGTR1_HUMAN P30556 CHEMBL227 Angiotensin II type 1 receptor 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
AURKC_HUMAN Q9UQB9 CHEMBL3935 Serine/threonine-protein kinase Aurora-C 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
CP51A_HUMAN Q16850 CHEMBL3849 Cytochrome P450 51 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
EDNRA_HUMAN P25101 CHEMBL252 Endothelin receptor ET-A 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
ERBB2_HUMAN P04626 CHEMBL1824 Receptor protein-tyrosine kinase erbB-2 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
FGR_HUMAN P09769 CHEMBL4454 Tyrosine-protein kinase FGR 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
FYN_HUMAN P06241 CHEMBL1841 Tyrosine-protein kinase FYN 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
HCK_HUMAN P08631 CHEMBL3234 Tyrosine-protein kinase HCK 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
O77823_PIG O77823 CHEMBL3333 Phosphodiesterase 4A 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRK_CAVPO P41144 CHEMBL3952 Kappa opioid receptor 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDR5_YEAST P33302 CHEMBL1697658 Pleiotropic ABC efflux transporter of multiple drugs 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH2_BOVIN O62698 CHEMBL3331 Cyclooxygenase-2 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
SGMR1_CAVPO Q60492 CHEMBL4153 Sigma-1 receptor 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
TRY1_HUMAN P07477 CHEMBL209 Trypsin I 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
UFO_HUMAN P30530 CHEMBL4895 Tyrosine-protein kinase receptor UFO 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
YES_HUMAN P07947 CHEMBL2073 Tyrosine-protein kinase YES 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2A_BOVIN Q75Z89 CHEMBL3446 Serotonin 2a (5-HT2a) receptor 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT6R_RAT P31388 CHEMBL3372 Serotonin 6 (5-HT6) receptor 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
ABL2_HUMAN P42684 CHEMBL4014 Tyrosine-protein kinase ABL2 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACES_ELEEL O42275 CHEMBL4078 Acetylcholinesterase 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACE_RAT P47820 CHEMBL2625 Angiotensin-converting enzyme 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB3_HUMAN P13945 CHEMBL246 Beta-3 adrenergic receptor 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
AGTRA_RAT P25095 CHEMBL329 Angiotensin II type 1a (AT-1a) receptor 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
AGTRB_RAT P29089 CHEMBL263 Angiotensin II type 1b (AT-1b) receptor 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
ALDR_RAT P07943 CHEMBL2622 Aldose reductase 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
ANDR_RAT P15207 CHEMBL3072 Androgen Receptor 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
AOFA_HUMAN P21397 CHEMBL1951 Monoamine oxidase A 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH_METTE P40881 CHEMBL3932 Carbonic anhydrase 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
EPHA3_HUMAN P29320 CHEMBL4954 Ephrin type-A receptor 3 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
EPHA6_HUMAN Q9UF33 CHEMBL4526 Ephrin type-A receptor 6 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
ESR1_RAT P06211 CHEMBL2724 Estrogen receptor alpha 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
ESR2_RAT Q62986 CHEMBL3021 Estrogen receptor beta 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA6_HUMAN Q16445 CHEMBL2579 GABA receptor alpha-6 subunit 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
GCR_HUMAN P04150 CHEMBL2034 Glucocorticoid receptor 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
HMDH_HUMAN P04035 CHEMBL402 HMG-CoA reductase 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
HRH3_HUMAN Q9Y5N1 CHEMBL264 Histamine H3 receptor 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
JAK2_HUMAN O60674 CHEMBL2971 Tyrosine-protein kinase JAK2 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
LT4R1_HUMAN Q15722 CHEMBL3911 Leukotriene B4 receptor 1 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
MMP2_HUMAN P08253 CHEMBL333 Matrix metalloproteinase-2 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
NK1R_HUMAN P25103 CHEMBL249 Neurokinin 1 receptor 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDZ1_RAT P35439 CHEMBL330 Glutamate (NMDA) receptor subunit zeta 1 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
NTRK1_HUMAN P04629 CHEMBL2815 Nerve growth factor receptor Trk-A 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRK_MOUSE P33534 CHEMBL4329 Kappa opioid receptor 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE4A_RAT P54748 CHEMBL4964 Phosphodiesterase 4A 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE4B_RAT P14646 CHEMBL3382 Phosphodiesterase 4B 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE4D_RAT P14270 CHEMBL2712 Phosphodiesterase 4D 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
PRGR_HUMAN P06401 CHEMBL208 Progesterone receptor 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
PRIO_HUMAN P04156 CHEMBL4869 Prion protein 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
TA2R_HUMAN P21731 CHEMBL2069 Thromboxane A2 receptor 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
TIE1_HUMAN P35590 CHEMBL5274 Tyrosine-protein kinase receptor Tie-1 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104297 Z104297 CHEMBL1907603 Glutamate NMDA receptor; GRIN1/GRIN2B 10 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACES_BOVIN P23795 CHEMBL4768 Acetylcholinesterase 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACES_MOUSE P21836 CHEMBL3198 Acetylcholinesterase 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACES_TORCA P04058 CHEMBL4780 Acetylcholinesterase 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM1_MOUSE P12657 CHEMBL3733 Muscarinic acetylcholine receptor M1 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB2_BOVIN Q28044 CHEMBL3373 Beta-2 adrenergic receptor 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB2_RAT P10608 CHEMBL3754 Beta-2 adrenergic receptor 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
CLK1_HUMAN P49759 CHEMBL4224 Dual specificty protein kinase CLK1 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
CNR1_HUMAN P21554 CHEMBL218 Cannabinoid CB1 receptor 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
DDR2_HUMAN Q16832 CHEMBL5122 Discoidin domain-containing receptor 2 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
DYR_PNECA P16184 CHEMBL1926 Dihydrofolate reductase 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
DYR_RAT Q920D2 CHEMBL2363 Dihydrofolate reductase 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
EDNRB_HUMAN P24530 CHEMBL1785 Endothelin receptor ET-B 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
EPHA8_HUMAN P29322 CHEMBL4134 Ephrin type-A receptor 8 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
EPHB1_HUMAN P54762 CHEMBL5072 Ephrin type-B receptor 1 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
EPHB4_HUMAN P54760 CHEMBL5147 Ephrin type-B receptor 4 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
FPPS_HUMAN P14324 CHEMBL1782 Farnesyl diphosphate synthase 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA2_RAT P23576 CHEMBL341 GABA receptor alpha-2 subunit 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA4_HUMAN P48169 CHEMBL2472 GABA receptor alpha-4 subunit 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
HDAC3_HUMAN O15379 CHEMBL1829 Histone deacetylase 3 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
HRH3_RAT Q9QYN8 CHEMBL4124 Histamine H3 receptor 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
M4K3_HUMAN Q8IVH8 CHEMBL5432 Mitogen-activated protein kinase kinase kinase kinase 3 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
MERTK_HUMAN Q12866 CHEMBL5331 Proto-oncogene tyrosine-protein kinase MER 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
MK14_HUMAN Q16539 CHEMBL260 MAP kinase p38 alpha 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
MKNK2_HUMAN Q9HBH9 CHEMBL4204 MAP kinase signal-integrating kinase 2 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
MLTK_HUMAN Q9NYL2 CHEMBL3886 Mixed lineage kinase 7 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE3_RAT Q00961 CHEMBL401 Glutamate [NMDA] receptor subunit epsilon 3 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
NTRK2_HUMAN Q16620 CHEMBL4898 Neurotrophic tyrosine kinase receptor type 2 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRM_CAVPO P97266 CHEMBL4354 Mu opioid receptor 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
P96878_MYCTU P96878 CHEMBL5767 PROBABLE TRANSMEMBRANE CARBONIC ANHYDRASE (CARBONATE DEHYDRATASE) (CARBONIC DEHYDRATASE) 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
TBA1A_RAT P68370 CHEMBL4139 Tubulin alpha-1 chain 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
THAS_HUMAN P24557 CHEMBL1835 Thromboxane-A synthase 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
TNI3K_HUMAN Q59H18 CHEMBL5260 Serine/threonine-protein kinase TNNI3K 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104288 Z104288 CHEMBL1907594 Neuronal acetylcholine receptor; alpha3/beta4 9 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1E_HUMAN P28566 CHEMBL2182 Serotonin 1e (5-HT1e) receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2C_MOUSE P34968 CHEMBL3006 Serotonin 2c (5-HT2c) receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3A_MOUSE P23979 CHEMBL4972 Serotonin 3a (5-HT3a) receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3B_HUMAN O95264 CHEMBL3895 Serotonin 3b (5-HT3b) receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3C_HUMAN Q8WXA8 CHEMBL4795 Serotonin 3c (5-HT3c) receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3D_HUMAN Q70Z44 CHEMBL4673 Serotonin 3d (5-HT3d) receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3E_HUMAN A5X5Y0 CHEMBL3812 Serotonin 3e (5-HT3e) receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT5A_RAT P35364 CHEMBL4655 Serotonin 5a (5-HT5a) receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT5B_RAT P35365 CHEMBL2619 Serotonin 5b (5-HT5b) receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHD_TORCA P02718 CHEMBL3916 Acetylcholine receptor protein delta chain 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
AURKB_HUMAN Q96GD4 CHEMBL2185 Serine/threonine-protein kinase Aurora-B 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH5A_MOUSE P23589 CHEMBL2330 Carbonic anhydrase VA 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH5B_MOUSE Q9QZA0 CHEMBL4634 Carbonic anhydrase VB 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
CCKAR_RAT P30551 CHEMBL2871 Cholecystokinin A receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
CDK16_HUMAN Q00536 CHEMBL4597 Serine/threonine-protein kinase PCTAIRE-1 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
CLK4_HUMAN Q9HAZ1 CHEMBL4203 Dual specificity protein kinase CLK4 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
CNR1_RAT P20272 CHEMBL3571 Cannabinoid CB1 receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
CYSP_TRYCR P25779 CHEMBL3563 Cruzipain 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
DPP4_HUMAN P27487 CHEMBL284 Dipeptidyl peptidase IV 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRTS_TOXGO Q07422 CHEMBL2425 Dihydrofolate reductase 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
DYR_LACCA P00381 CHEMBL2902 Dihydrofolate reductase 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
EDNRA_RAT P26684 CHEMBL4566 Endothelin receptor ET-A 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
ELNE_HUMAN P08246 CHEMBL248 Leukocyte elastase 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
EPHA5_HUMAN P54756 CHEMBL3987 Ephrin type-A receptor 5 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
FGFR2_HUMAN P21802 CHEMBL4142 Fibroblast growth factor receptor 2 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
HDAC1_HUMAN Q13547 CHEMBL325 Histone deacetylase 1 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
HDAC2_HUMAN Q92769 CHEMBL1937 Histone deacetylase 2 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
HMDH_RAT P51639 CHEMBL3247 HMG-CoA reductase 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
ITA2B_HUMAN P08514 CHEMBL212 Integrin alpha-IIb 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
ITB3_HUMAN P05106 CHEMBL207 Integrin beta-3 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
M4K1_HUMAN Q92918 CHEMBL5749 Mitogen-activated protein kinase kinase kinase kinase 1 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
M4K4_HUMAN O95819 CHEMBL6166 Mitogen-activated protein kinase kinase kinase kinase 4 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
MCR_HUMAN P08235 CHEMBL1994 Mineralocorticoid receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
MK09_HUMAN P45984 CHEMBL4179 c-Jun N-terminal kinase 2 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMD3B_RAT Q8VHN2 CHEMBL282 Glutamate [NMDA] receptor subunit 3B 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE4C_RAT P14644 CHEMBL4562 Phosphodiesterase 4C 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH2_MOUSE Q05769 CHEMBL4321 Cyclooxygenase-2 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q864F1_PIG Q864F1 CHEMBL3634 Phosphodiesterase 5 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
RENI_HUMAN P00797 CHEMBL286 Renin 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
RIPK2_HUMAN O43353 CHEMBL5014 Serine/threonine-protein kinase RIPK2 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
SCN2A_RAT P04775 CHEMBL3399 Sodium channel protein type II alpha subunit 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
SIK2_HUMAN Q9H0K1 CHEMBL5699 Serine/threonine-protein kinase SIK2 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
TNIK_HUMAN Q9UKE5 CHEMBL4527 TRAF2- and NCK-interacting kinase 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
V2R_HUMAN P30518 CHEMBL1790 Vasopressin V2 receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z100491 Z100491 CHEMBL613288 Sigma 2 receptor 8 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3B_MOUSE Q9JHJ5 CHEMBL3781 Serotonin 3b (5-HT3b) receptor 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA2BR_HUMAN P29275 CHEMBL255 Adenosine A2b receptor 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
AAK1_HUMAN Q2M2I8 CHEMBL3830 Adaptor-associated kinase 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADCY1_HUMAN Q08828 CHEMBL2899 Brain adenylate cyclase 1 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
AK1A1_HUMAN P14550 CHEMBL2246 Aldehyde reductase 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
ALDR_PIG P80276 CHEMBL4559 Aldose reductase 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
AURKA_HUMAN O14965 CHEMBL4722 Serine/threonine-protein kinase Aurora-A 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
BMP2K_HUMAN Q9NSY1 CHEMBL4522 BMP-2-inducible protein kinase 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
C11B1_HUMAN P15538 CHEMBL1908 Cytochrome P450 11B1 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAC1D_HUMAN Q01668 CHEMBL4138 Voltage-gated L-type calcium channel alpha-1D subunit 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
CLK2_HUMAN P49760 CHEMBL4225 Dual specificity protein kinase CLK2 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
CNR2_HUMAN P34972 CHEMBL253 Cannabinoid CB2 receptor 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
CSK_HUMAN P41240 CHEMBL2634 Tyrosine-protein kinase CSK 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
CTRA_BOVIN P00766 CHEMBL3314 Alpha-chymotrypsin 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
FGFR3_HUMAN P22607 CHEMBL2742 Fibroblast growth factor receptor 3 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
GASR_RAT P30553 CHEMBL3508 Cholecystokinin B receptor 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRB1_HUMAN P18505 CHEMBL4558 GABA receptor beta-1 subunit 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRD_HUMAN O14764 CHEMBL3591 GABA receptor delta subunit 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRE_HUMAN P78334 CHEMBL4635 GABA receptor epsilon subunit 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRG1_HUMAN Q8N1C3 CHEMBL4044 GABA receptor gamma-1 subunit 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRG3_HUMAN Q99928 CHEMBL2739 GABA receptor gamma-3 subunit 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRP_HUMAN O00591 CHEMBL3506 GABA receptor pi subunit 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRT_HUMAN Q9UN88 CHEMBL2843 GABA receptor theta subunit 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIA1_MOUSE P23818 CHEMBL3502 Glutamate receptor ionotropic, AMPA 1 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIA2_RAT P19491 CHEMBL3503 Glutamate receptor ionotropic, AMPA 2 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIA3_RAT P19492 CHEMBL3504 Glutamate receptor ionotropic, AMPA 3 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIA4_RAT P19493 CHEMBL3505 Glutamate receptor ionotropic, AMPA 4 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
JAK1_HUMAN P23458 CHEMBL2835 Tyrosine-protein kinase JAK1 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
KC1E_HUMAN P49674 CHEMBL4937 Casein kinase I epsilon 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
KS6A2_HUMAN Q15349 CHEMBL3906 Ribosomal protein S6 kinase alpha 2 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
KS6A4_HUMAN O75676 CHEMBL3125 Ribosomal protein S6 kinase alpha 4 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
KS6A6_HUMAN Q9UK32 CHEMBL4924 Ribosomal protein S6 kinase alpha 6 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
MET_HUMAN P08581 CHEMBL3717 Hepatocyte growth factor receptor 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
MK10_HUMAN P53779 CHEMBL2637 c-Jun N-terminal kinase 3 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
MMP1_HUMAN P03956 CHEMBL332 Matrix metalloproteinase-1 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
MMP9_HUMAN P14780 CHEMBL321 Matrix metalloproteinase 9 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
MYLK2_HUMAN Q9H1R3 CHEMBL2777 myosin light chain kinase 2 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE4_RAT Q62645 CHEMBL303 Glutamate [NMDA] receptor subunit epsilon 4 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
NTRK3_HUMAN Q16288 CHEMBL5608 NT-3 growth factor receptor 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRD_MOUSE P32300 CHEMBL3222 Delta opioid receptor 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE1A_HUMAN P54750 CHEMBL3421 Phosphodiesterase 1A 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE1B_HUMAN Q01064 CHEMBL4425 Phosphodiesterase 1B 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE1C_HUMAN Q14123 CHEMBL4619 Phosphodiesterase 1C 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
PHKG1_HUMAN Q16816 CHEMBL4004 Phosphorylase kinase gamma subunit 1 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
PLK4_HUMAN O00444 CHEMBL3788 Serine/threonine-protein kinase PLK4 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q4U254_9ENTO Q4U254 CHEMBL2857 Human rhinovirus A protease 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
RAF1_HUMAN P04049 CHEMBL1906 Serine/threonine-protein kinase RAF 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
RARG_HUMAN P13631 CHEMBL2003 Retinoic acid receptor gamma 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
S22A6_MOUSE Q8VC69 CHEMBL5653 Solute carrier family 22 member 6 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
SC6A3_MOUSE Q61327 CHEMBL2799 Dopamine transporter 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
SGMR1_MOUSE O55242 CHEMBL3465 Sigma opioid receptor 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
STK33_HUMAN Q9BYT3 CHEMBL6005 Serine/threonine-protein kinase 33 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
STK3_HUMAN Q13188 CHEMBL4708 Serine/threonine-protein kinase MST2 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
TIE2_HUMAN Q02763 CHEMBL4128 Tyrosine-protein kinase TIE-2 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
TOP2A_HUMAN P11388 CHEMBL1806 DNA topoisomerase II alpha 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
TSPO_RAT P16257 CHEMBL4552 Peripheral-type benzodiazepine receptor 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
TXK_HUMAN P42681 CHEMBL4367 Tyrosine-protein kinase TXK 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
V1AR_HUMAN P37288 CHEMBL1889 Vasopressin V1a receptor 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104290 Z104290 CHEMBL1907596 Neuronal acetylcholine receptor; alpha4/beta2 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z50587 Z50587 CHEMBL372 Homo sapiens 7 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1A_MOUSE Q64264 CHEMBL3737 Serotonin 1a (5-HT1a) receptor 6 Annotations Catalogs SMILES SDF Mol2 Flexibase
ABCC9_HUMAN O60706 CHEMBL1971 Sulfonylurea receptor 2 6 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHA7_RAT Q05941 CHEMBL4980 Neuronal acetylcholine receptor protein alpha-7 subunit 6 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM2_MOUSE Q9ERZ4