UCSF

Leadscope via PubChem

Binding 10μM Binding 1μM Functional 10μM ADME/T 10μM

Binding 10μM Targets with Highest Number of Available Compounds (2191 in total)

Name (Uniprot) Swissprot ChEMBL Description Size Browse Download (Annotations)
DRD2_RAT P61169 CHEMBL339 Dopamine D2 receptor 266 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1A_RAT P19327 CHEMBL273 Serotonin 1a (5-HT1a) receptor 196 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2A_RAT P14842 CHEMBL322 Serotonin 2a (5-HT2a) receptor 183 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD1_RAT P18901 CHEMBL265 Dopamine D1 receptor 159 Annotations Catalogs SMILES SDF Mol2 Flexibase
KCNH2_HUMAN Q12809 CHEMBL240 HERG 155 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2C_RAT P08909 CHEMBL324 Serotonin 2c (5-HT2c) receptor 154 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD2_HUMAN P14416 CHEMBL217 Dopamine D2 receptor 148 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACES_HUMAN P22303 CHEMBL220 Acetylcholinesterase 147 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH2_HUMAN P00918 CHEMBL205 Carbonic anhydrase II 137 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104304 Z104304 CHEMBL1907610 Adrenergic receptor alpha-1 137 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104301 Z104301 CHEMBL1907607 GABA-A receptor; anion channel 134 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2B_RAT P30994 CHEMBL323 Serotonin 2b (5-HT2b) receptor 130 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2A_RAT P22909 CHEMBL327 Alpha-2a adrenergic receptor 128 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2B_RAT P19328 CHEMBL266 Alpha-2b adrenergic receptor 125 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD3_RAT P19020 CHEMBL3138 Dopamine D3 receptor 124 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2C_RAT P22086 CHEMBL314 Alpha-2c adrenergic receptor 121 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA1R_RAT P25099 CHEMBL318 Adenosine A1 receptor 116 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRM_RAT P33535 CHEMBL270 Mu opioid receptor 116 Annotations Catalogs SMILES SDF Mol2 Flexibase
SGMR1_HUMAN Q99720 CHEMBL287 Sigma opioid receptor 114 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA2AR_RAT P30543 CHEMBL302 Adenosine A2a receptor 108 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1B_RAT P28564 CHEMBL3459 Serotonin 1b (5-HT1b) receptor 104 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH1_HUMAN P00915 CHEMBL261 Carbonic anhydrase I 102 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD4_RAT P30729 CHEMBL3361 Dopamine D4 receptor 102 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD5_RAT P25115 CHEMBL2281 Dopamine D5 receptor 102 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRM_HUMAN P35372 CHEMBL233 Mu opioid receptor 102 Annotations Catalogs SMILES SDF Mol2 Flexibase
SC6A3_RAT P23977 CHEMBL338 Dopamine transporter 99 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD3_HUMAN P35462 CHEMBL234 Dopamine D3 receptor 96 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2A_HUMAN P28223 CHEMBL224 Serotonin 2a (5-HT2a) receptor 95 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2C_HUMAN P28335 CHEMBL225 Serotonin 2c (5-HT2c) receptor 94 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1A_HUMAN P08908 CHEMBL214 Serotonin 1a (5-HT1a) receptor 90 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRK_HUMAN P41145 CHEMBL237 Kappa opioid receptor 90 Annotations Catalogs SMILES SDF Mol2 Flexibase
SC6A2_HUMAN P23975 CHEMBL222 Norepinephrine transporter 90 Annotations Catalogs SMILES SDF Mol2 Flexibase
SGMR1_RAT Q9R0C9 CHEMBL3602 Sigma opioid receptor 89 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104303 Z104303 CHEMBL1907609 Muscarinic acetylcholine receptor 89 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRD_RAT P33533 CHEMBL269 Delta opioid receptor 86 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH2_HUMAN P35354 CHEMBL230 Cyclooxygenase-2 86 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1D_HUMAN P25100 CHEMBL223 Alpha-1d adrenergic receptor 85 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD4_HUMAN P21917 CHEMBL219 Dopamine D4 receptor 85 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA3R_HUMAN P33765 CHEMBL256 Adenosine A3 receptor 83 Annotations Catalogs SMILES SDF Mol2 Flexibase
SC6A3_HUMAN Q01959 CHEMBL238 Dopamine transporter 83 Annotations Catalogs SMILES SDF Mol2 Flexibase
SC6A4_RAT P31652 CHEMBL313 Serotonin transporter 83 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH9_HUMAN Q16790 CHEMBL3594 Carbonic anhydrase IX 82 Annotations Catalogs SMILES SDF Mol2 Flexibase
SCN2A_HUMAN Q99250 CHEMBL4187 Sodium channel protein type II alpha subunit 82 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM1_HUMAN P11229 CHEMBL216 Muscarinic acetylcholine receptor M1 80 Annotations Catalogs SMILES SDF Mol2 Flexibase
SCN1A_HUMAN P35498 CHEMBL1845 Sodium channel protein type I alpha subunit 79 Annotations Catalogs SMILES SDF Mol2 Flexibase
SCN3A_HUMAN Q9NY46 CHEMBL5163 Sodium channel protein type III alpha subunit 79 Annotations Catalogs SMILES SDF Mol2 Flexibase
SCN8A_HUMAN Q9UQD0 CHEMBL5202 Sodium channel protein type VIII alpha subunit 79 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRD_HUMAN P41143 CHEMBL236 Delta opioid receptor 78 Annotations Catalogs SMILES SDF Mol2 Flexibase
SC6A4_HUMAN P31645 CHEMBL228 Serotonin transporter 77 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM2_RAT P10980 CHEMBL309 Muscarinic acetylcholine receptor M2 76 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH12_HUMAN O43570 CHEMBL3242 Carbonic anhydrase XII 76 Annotations Catalogs SMILES SDF Mol2 Flexibase
CHLE_HUMAN P06276 CHEMBL1914 Butyrylcholinesterase 76 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD2_BOVIN P20288 CHEMBL3998 Dopamine D2 receptor 76 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104302 Z104302 CHEMBL1907608 Glutamate NMDA receptor 74 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM1_RAT P08482 CHEMBL276 Muscarinic acetylcholine receptor M1 71 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA2BR_RAT P29276 CHEMBL2592 Adenosine A2b receptor 70 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRK_RAT P34975 CHEMBL3614 Kappa opioid receptor 70 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1D_RAT P28565 CHEMBL5450 Serotonin 1d (5-HT1d) receptor 69 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM2_HUMAN P08172 CHEMBL211 Muscarinic acetylcholine receptor M2 68 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM3_HUMAN P20309 CHEMBL245 Muscarinic acetylcholine receptor M3 67 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1F_RAT P30940 CHEMBL4646 Serotonin 1f (5-HT1f) receptor 65 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1A_HUMAN P35348 CHEMBL229 Alpha-1a adrenergic receptor 64 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH1_HUMAN P23219 CHEMBL221 Cyclooxygenase-1 64 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH6_HUMAN P23280 CHEMBL3025 Carbonic anhydrase VI 63 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q9WTR4_RAT Q9WTR4 CHEMBL304 Norepinephrine transporter 62 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2A_HUMAN P08913 CHEMBL1867 Alpha-2a adrenergic receptor 60 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH4_HUMAN P22748 CHEMBL3729 Carbonic anhydrase IV 60 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD1_HUMAN P21728 CHEMBL2056 Dopamine D1 receptor 60 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2B_HUMAN P41595 CHEMBL1833 Serotonin 2b (5-HT2b) receptor 59 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH7_HUMAN P43166 CHEMBL2326 Carbonic anhydrase VII 59 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH5A_HUMAN P35218 CHEMBL4789 Carbonic anhydrase VA 57 Annotations Catalogs SMILES SDF Mol2 Flexibase
HRH1_HUMAN P35367 CHEMBL231 Histamine H1 receptor 56 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH5B_HUMAN Q9Y2D0 CHEMBL3969 Carbonic anhydrase VB 55 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1B_HUMAN P35368 CHEMBL232 Alpha-1b adrenergic receptor 53 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3A_HUMAN P46098 CHEMBL1899 Serotonin 3a (5-HT3a) receptor 52 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3A_RAT P35563 CHEMBL2411 Serotonin 3a (5-HT3a) receptor 52 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2C_HUMAN P18825 CHEMBL1916 Alpha-2c adrenergic receptor 52 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3B_RAT Q9JJ16 CHEMBL3458 Serotonin 3b (5-HT3b) receptor 51 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACES_RAT P37136 CHEMBL3199 Acetylcholinesterase 51 Annotations Catalogs SMILES SDF Mol2 Flexibase
AOFB_HUMAN P27338 CHEMBL2039 Monoamine oxidase B 51 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z50597 Z50597 CHEMBL376 Rattus norvegicus 51 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM4_HUMAN P08173 CHEMBL1821 Muscarinic acetylcholine receptor M4 50 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1A_BOVIN P18130 CHEMBL4892 Alpha-1a adrenergic receptor 50 Annotations Catalogs SMILES SDF Mol2 Flexibase
CP19A_HUMAN P11511 CHEMBL1978 Cytochrome P450 19A1 50 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA2_HUMAN P47869 CHEMBL4956 GABA receptor alpha-2 subunit 50 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA2AR_HUMAN P29274 CHEMBL251 Adenosine A2a receptor 49 Annotations Catalogs SMILES SDF Mol2 Flexibase
AOFA_RAT P21396 CHEMBL3358 Monoamine oxidase A 49 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH14_HUMAN Q9ULX7 CHEMBL3510 Carbonic anhydrase XIV 49 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA1_HUMAN P14867 CHEMBL1962 GABA receptor alpha-1 subunit 49 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT6R_HUMAN P50406 CHEMBL3371 Serotonin 6 (5-HT6) receptor 47 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB2_HUMAN P07550 CHEMBL210 Beta-2 adrenergic receptor 47 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA3_HUMAN P34903 CHEMBL3026 GABA receptor alpha-3 subunit 47 Annotations Catalogs SMILES SDF Mol2 Flexibase
LOX5_RAT P12527 CHEMBL312 Arachidonate 5-lipoxygenase 47 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM5_HUMAN P08912 CHEMBL2035 Muscarinic acetylcholine receptor M5 46 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH15_MOUSE Q99N23 CHEMBL5973 Carbonic anhydrase 15 46 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA5_HUMAN P31644 CHEMBL5112 GABA receptor alpha-5 subunit 46 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1A_RAT P43140 CHEMBL319 Alpha-1a adrenergic receptor 43 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2B_HUMAN P18089 CHEMBL1942 Alpha-2b adrenergic receptor 43 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT7R_HUMAN P34969 CHEMBL3155 Serotonin 7 (5-HT7) receptor 42 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA1R_HUMAN P30542 CHEMBL226 Adenosine A1 receptor 42 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM1_MOUSE P12657 CHEMBL3733 Muscarinic acetylcholine receptor M1 42 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRG2_HUMAN P18507 CHEMBL1788 GABA receptor gamma-2 subunit 42 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1D_HUMAN P28221 CHEMBL1983 Serotonin 1d (5-HT1d) receptor 41 Annotations Catalogs SMILES SDF Mol2 Flexibase
ESR1_HUMAN P03372 CHEMBL206 Estrogen receptor alpha 41 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3B_HUMAN O95264 CHEMBL3895 Serotonin 3b (5-HT3b) receptor 40 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3C_HUMAN Q8WXA8 CHEMBL4795 Serotonin 3c (5-HT3c) receptor 40 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3D_HUMAN Q70Z44 CHEMBL4673 Serotonin 3d (5-HT3d) receptor 40 Annotations Catalogs SMILES SDF Mol2 Flexibase
EGFR_HUMAN P00533 CHEMBL203 Epidermal growth factor receptor erbB1 40 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE4A_HUMAN P27815 CHEMBL254 Phosphodiesterase 4A 40 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE4B_HUMAN Q07343 CHEMBL275 Phosphodiesterase 4B 40 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT3E_HUMAN A5X5Y0 CHEMBL3812 Serotonin 3e (5-HT3e) receptor 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
AOFB_RAT P19643 CHEMBL2993 Monoamine oxidase B 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
ESR2_HUMAN Q92731 CHEMBL242 Estrogen receptor beta 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRB3_HUMAN P28472 CHEMBL1847 GABA receptor beta-3 subunit 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMD3A_HUMAN Q8TCU5 CHEMBL4787 Glutamate [NMDA] receptor subunit 3A 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMD3B_HUMAN O60391 CHEMBL2913 Glutamate [NMDA] receptor subunit 3B 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE1_HUMAN Q12879 CHEMBL1972 Glutamate [NMDA] receptor subunit epsilon 1 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE2_HUMAN Q13224 CHEMBL1904 Glutamate [NMDA] receptor subunit epsilon 2 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE3_HUMAN Q14957 CHEMBL4109 Glutamate [NMDA] receptor subunit epsilon 3 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE4_HUMAN O15399 CHEMBL2591 Glutamate [NMDA] receptor subunit epsilon 4 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDZ1_HUMAN Q05586 CHEMBL2015 Glutamate (NMDA) receptor subunit zeta 1 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE4D_HUMAN Q08499 CHEMBL288 Phosphodiesterase 4D 39 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB1_RAT P18090 CHEMBL3252 Beta-1 adrenergic receptor 38 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE4C_HUMAN Q08493 CHEMBL291 Phosphodiesterase 4C 38 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1D_RAT P23944 CHEMBL326 Alpha-1d adrenergic receptor 37 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH3_HUMAN P07451 CHEMBL2885 Carbonic anhydrase III 37 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD1_BOVIN Q95136 CHEMBL2967 Dopamine D1 receptor 37 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB1_HUMAN P08588 CHEMBL213 Beta-1 adrenergic receptor 36 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA2BR_HUMAN P29275 CHEMBL255 Adenosine A2b receptor 35 Annotations Catalogs SMILES SDF Mol2 Flexibase
AOFA_HUMAN P21397 CHEMBL1951 Monoamine oxidase A 35 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1B_HUMAN P28222 CHEMBL1898 Serotonin 1b (5-HT1b) receptor 34 Annotations Catalogs SMILES SDF Mol2 Flexibase
CNR1_RAT P20272 CHEMBL3571 Cannabinoid CB1 receptor 34 Annotations Catalogs SMILES SDF Mol2 Flexibase
NOS1_HUMAN P29475 CHEMBL3568 Nitric-oxide synthase, brain 34 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRD_MOUSE P32300 CHEMBL3222 Delta opioid receptor 34 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE3A_HUMAN Q14432 CHEMBL241 Phosphodiesterase 3A 34 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE3B_HUMAN Q13370 CHEMBL290 Phosphodiesterase 3B 34 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH4_BOVIN Q95323 CHEMBL281 Carbonic anhydrase IV 33 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACE_HUMAN P12821 CHEMBL1808 Angiotensin-converting enzyme 32 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH13_MOUSE Q9D6N1 CHEMBL2186 Carbonic anhydrase XIII 32 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2A_BOVIN Q75Z89 CHEMBL3446 Serotonin 2a (5-HT2a) receptor 31 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA2A_BOVIN Q28838 CHEMBL4744 Alpha-2a adrenergic receptor 31 Annotations Catalogs SMILES SDF Mol2 Flexibase
CNR1_HUMAN P21554 CHEMBL218 Cannabinoid CB1 receptor 31 Annotations Catalogs SMILES SDF Mol2 Flexibase
NOS2_HUMAN P35228 CHEMBL4481 Nitric oxide synthase, inducible 31 Annotations Catalogs SMILES SDF Mol2 Flexibase
SOAT1_HUMAN P35610 CHEMBL2782 Acyl coenzyme A:cholesterol acyltransferase 1 31 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104290 Z104290 CHEMBL1907596 Neuronal acetylcholine receptor; alpha4/beta2 31 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACES_TORCA P04058 CHEMBL4780 Acetylcholinesterase 30 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM3_RAT P08483 CHEMBL320 Muscarinic acetylcholine receptor M3 30 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA6_HUMAN Q16445 CHEMBL2579 GABA receptor alpha-6 subunit 30 Annotations Catalogs SMILES SDF Mol2 Flexibase
MTR1A_HUMAN P48039 CHEMBL1945 Melatonin receptor 1A 30 Annotations Catalogs SMILES SDF Mol2 Flexibase
MTR1B_HUMAN P49286 CHEMBL1946 Melatonin receptor 1B 30 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRM_MOUSE P42866 CHEMBL2858 Mu opioid receptor 30 Annotations Catalogs SMILES SDF Mol2 Flexibase
SGMR1_CAVPO Q60492 CHEMBL4153 Sigma-1 receptor 30 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT7R_RAT P32305 CHEMBL3223 Serotonin 7 (5-HT7) receptor 29 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHA4_RAT P09483 CHEMBL307 Neuronal acetylcholine receptor protein alpha-4 subunit 29 Annotations Catalogs SMILES SDF Mol2 Flexibase
ERG2_YEAST P32352 CHEMBL3224 C-8 sterol isomerase 29 Annotations Catalogs SMILES SDF Mol2 Flexibase
HRH1_RAT P31390 CHEMBL4701 Histamine H1 receptor 29 Annotations Catalogs SMILES SDF Mol2 Flexibase
TA2R_HUMAN P21731 CHEMBL2069 Thromboxane A2 receptor 29 Annotations Catalogs SMILES SDF Mol2 Flexibase
ANDR_HUMAN P10275 CHEMBL1871 Androgen Receptor 28 Annotations Catalogs SMILES SDF Mol2 Flexibase
CNR2_HUMAN P34972 CHEMBL253 Cannabinoid CB2 receptor 28 Annotations Catalogs SMILES SDF Mol2 Flexibase
EBP_HUMAN Q15125 CHEMBL4931 3-beta-hydroxysteroid-delta(8),delta(7)-isomerase 28 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA4_HUMAN P48169 CHEMBL2472 GABA receptor alpha-4 subunit 28 Annotations Catalogs SMILES SDF Mol2 Flexibase
LCK_HUMAN P06239 CHEMBL258 Tyrosine-protein kinase LCK 28 Annotations Catalogs SMILES SDF Mol2 Flexibase
PTAFR_HUMAN P25105 CHEMBL250 Platelet activating factor receptor 28 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHA3_RAT P04757 CHEMBL3818 Neuronal acetylcholine receptor protein alpha-3 subunit 27 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB2_CANFA P54833 CHEMBL2289 Beta-2 adrenergic receptor 27 Annotations Catalogs SMILES SDF Mol2 Flexibase
DYR_HUMAN P00374 CHEMBL202 Dihydrofolate reductase 27 Annotations Catalogs SMILES SDF Mol2 Flexibase
GSK3B_HUMAN P49841 CHEMBL262 Glycogen synthase kinase-3 beta 27 Annotations Catalogs SMILES SDF Mol2 Flexibase
LOX5_HUMAN P09917 CHEMBL215 Arachidonate 5-lipoxygenase 27 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE3_RAT Q00961 CHEMBL401 Glutamate [NMDA] receptor subunit epsilon 3 27 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDZ1_RAT P35439 CHEMBL330 Glutamate (NMDA) receptor subunit zeta 1 27 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q5AJ71_CANAL Q5AJ71 CHEMBL5337 Carbonic anhydrase 27 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104283 Z104283 CHEMBL1907589 Neuronal acetylcholine receptor; alpha4/beta2 27 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACES_ELEEL O42275 CHEMBL4078 Acetylcholinesterase 26 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHA7_RAT Q05941 CHEMBL4980 Neuronal acetylcholine receptor protein alpha-7 subunit 26 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB3_RAT P26255 CHEMBL4031 Beta-3 adrenergic receptor 26 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRK_CAVPO P41144 CHEMBL3952 Kappa opioid receptor 26 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT4R_RAT Q62758 CHEMBL4317 Serotonin 4 (5-HT4) receptor 25 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACH10_RAT Q9JLB5 CHEMBL3461 Neuronal acetylcholine receptor protein alpha-10 subunit 25 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHA7_HUMAN P36544 CHEMBL2492 Neuronal acetylcholine receptor protein alpha-7 subunit 25 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADA1B_RAT P15823 CHEMBL315 Alpha-1b adrenergic receptor 25 Annotations Catalogs SMILES SDF Mol2 Flexibase
ALDR_RAT P07943 CHEMBL2622 Aldose reductase 25 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRB2_HUMAN P47870 CHEMBL1920 GABA receptor beta-2 subunit 25 Annotations Catalogs SMILES SDF Mol2 Flexibase
HRH3_HUMAN Q9Y5N1 CHEMBL264 Histamine H3 receptor 25 Annotations Catalogs SMILES SDF Mol2 Flexibase
MDR1_HUMAN P08183 CHEMBL4302 P-glycoprotein 1 25 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE2_RAT Q00960 CHEMBL311 Glutamate [NMDA] receptor subunit epsilon 2 25 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH1_RAT Q63921 CHEMBL4042 Cyclooxygenase-1 25 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA3R_RAT P28647 CHEMBL3360 Adenosine A3 receptor 24 Annotations Catalogs SMILES SDF Mol2 Flexibase
B5SU02_9CNID B5SU02 CHEMBL1075028 Alpha carbonic anhydrase 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
NOS3_HUMAN P29474 CHEMBL4803 Nitric-oxide synthase, endothelial 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRM_CAVPO P97266 CHEMBL4354 Mu opioid receptor 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH2_RAT P35355 CHEMBL2977 Cyclooxygenase-2 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
SRC_HUMAN P12931 CHEMBL267 Tyrosine-protein kinase SRC 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
THAS_HUMAN P24557 CHEMBL1835 Thromboxane-A synthase 23 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM2_MOUSE Q9ERZ4 CHEMBL3197 Muscarinic acetylcholine receptor M2 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
C0IX24_9CNID C0IX24 CHEMBL1649055 Carbonic anhydrase 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAC1C_RAT P22002 CHEMBL3762 Voltage-gated L-type calcium channel alpha-1C subunit 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
KIT_HUMAN P10721 CHEMBL1936 Stem cell growth factor receptor 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE4_RAT Q62645 CHEMBL303 Glutamate [NMDA] receptor subunit epsilon 4 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH1_SHEEP P05979 CHEMBL2949 Cyclooxygenase-1 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
PPARG_HUMAN P37231 CHEMBL235 Peroxisome proliferator-activated receptor gamma 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q72547_9HIV1 Q72547 CHEMBL247 Human immunodeficiency virus type 1 reverse transcriptase 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
RARG_HUMAN P13631 CHEMBL2003 Retinoic acid receptor gamma 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z100491 Z100491 CHEMBL613288 Sigma 2 receptor 22 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHD_TORCA P02718 CHEMBL3916 Acetylcholine receptor protein delta chain 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
CDK1_HUMAN P06493 CHEMBL308 Cyclin-dependent kinase 1 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIA2_RAT P19491 CHEMBL3503 Glutamate receptor ionotropic, AMPA 2 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIA3_RAT P19492 CHEMBL3504 Glutamate receptor ionotropic, AMPA 3 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIA4_RAT P19493 CHEMBL3505 Glutamate receptor ionotropic, AMPA 4 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
HRH4_HUMAN Q9H3N8 CHEMBL3759 Histamine H4 receptor 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q63380_RAT Q63380 CHEMBL6184 Transporter 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q72874_9HIV1 Q72874 CHEMBL243 Human immunodeficiency virus type 1 protease 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
Y1284_MYCTU P64797 CHEMBL5631 Uncharacterized protein Rv1284/MT1322 21 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA1R_BOVIN P28190 CHEMBL4975 Adenosine A1 receptor 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
ALDR_HUMAN P15121 CHEMBL1900 Aldose reductase 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRD5_HUMAN P21918 CHEMBL1850 Dopamine D5 receptor 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA2_RAT P23576 CHEMBL341 GABA receptor alpha-2 subunit 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIA1_MOUSE P23818 CHEMBL3502 Glutamate receptor ionotropic, AMPA 1 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
KPCA_HUMAN P17252 CHEMBL299 Protein kinase C alpha 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
NISCH_HUMAN Q9Y2I1 CHEMBL3923 Nischarin 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q7ZJM1_9HIV1 Q7ZJM1 CHEMBL3471 Human immunodeficiency virus type 1 integrase 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
RARA_HUMAN P10276 CHEMBL2055 Retinoic acid receptor alpha 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
RARB_HUMAN P10826 CHEMBL2008 Retinoic acid receptor beta 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
VACHT_HUMAN Q16572 CHEMBL4767 Vesicular acetylcholine transporter 20 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACE_RAT P47820 CHEMBL2625 Angiotensin-converting enzyme 19 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHA2_RAT P12389 CHEMBL2584 Neuronal acetylcholine receptor protein alpha-2 subunit 19 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHB2_RAT P12390 CHEMBL3001 Neuronal acetylcholine receptor protein beta-2 subunit 19 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRTS_PLAFK P13922 CHEMBL1939 Dihydrofolate reductase 19 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHB4_RAT P12392 CHEMBL2658 Neuronal acetylcholine receptor protein beta-4 subunit 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
AGTRB_RAT P29089 CHEMBL263 Angiotensin II type 1b (AT-1b) receptor 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
AMPC_ECOLI P00811 CHEMBL2026 Beta-lactamase 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH13_HUMAN Q8N1Q1 CHEMBL3912 Carbonic anhydrase XIII 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAN_YEAST P53615 CHEMBL5931 Carbonic anhydrase 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
CYNT_HELPY O24855 CHEMBL4211 Carbonic anhydrase 1 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
KPCE_HUMAN Q02156 CHEMBL3582 Protein kinase C epsilon 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMD3B_RAT Q8VHN2 CHEMBL282 Glutamate [NMDA] receptor subunit 3B 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
PPARA_HUMAN Q07869 CHEMBL239 Peroxisome proliferator-activated receptor alpha 18 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACES_MOUSE P21836 CHEMBL3198 Acetylcholinesterase 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACM4_RAT P08485 CHEMBL317 Muscarinic acetylcholine receptor M4 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
CHLE_HORSE P81908 CHEMBL5763 Cholinesterase 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
CLTR2_HUMAN Q9NS75 CHEMBL4330 Cysteinyl leukotriene receptor 2 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRB1_HUMAN P18505 CHEMBL4558 GABA receptor beta-1 subunit 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRD_HUMAN O14764 CHEMBL3591 GABA receptor delta subunit 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRE_HUMAN P78334 CHEMBL4635 GABA receptor epsilon subunit 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRG1_HUMAN Q8N1C3 CHEMBL4044 GABA receptor gamma-1 subunit 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRG3_HUMAN Q99928 CHEMBL2739 GABA receptor gamma-3 subunit 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRP_HUMAN O00591 CHEMBL3506 GABA receptor pi subunit 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRT_HUMAN Q9UN88 CHEMBL2843 GABA receptor theta subunit 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
HRH3_RAT Q9QYN8 CHEMBL4124 Histamine H3 receptor 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
I23O1_HUMAN P14902 CHEMBL4685 Indoleamine 2,3-dioxygenase 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
KPCB_HUMAN P05771 CHEMBL3045 Protein kinase C beta 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
KPCD_HUMAN Q05655 CHEMBL2996 Protein kinase C delta 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
MK14_HUMAN Q16539 CHEMBL260 MAP kinase p38 alpha 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
MTR1B_CHICK P51050 CHEMBL4466 Melatonin receptor 1B 17 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT1E_HUMAN P28566 CHEMBL2182 Serotonin 1e (5-HT1e) receptor 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT4R_HUMAN Q13639 CHEMBL1875 Serotonin 4 (5-HT4) receptor 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT5A_HUMAN P47898 CHEMBL3426 Serotonin 5a (5-HT5a) receptor 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHA9_RAT P43144 CHEMBL2585 Neuronal acetylcholine receptor protein alpha-9 subunit 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHP_LYMST P58154 CHEMBL6084 Acetylcholine-binding protein 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAC1D_RAT P27732 CHEMBL4132 Voltage-gated L-type calcium channel alpha-1D subunit 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
CCKAR_RAT P30551 CHEMBL2871 Cholecystokinin A receptor 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
CYNT_MYCTU O53573 CHEMBL6068 Carbonic anhydrase 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
EDNRA_HUMAN P25101 CHEMBL252 Endothelin receptor ET-A 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
EST1_HUMAN P23141 CHEMBL2265 Acyl coenzyme A:cholesterol acyltransferase 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
FAAH1_HUMAN O00519 CHEMBL2243 Anandamide amidohydrolase 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
GASR_RAT P30553 CHEMBL3508 Cholecystokinin B receptor 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
MGLL_HUMAN Q99685 CHEMBL4191 Monoglyceride lipase 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
MTR1A_CHICK P49285 CHEMBL4555 Melatonin receptor 1A 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
MTR1C_CHICK P49288 CHEMBL3196 Melatonin receptor 1C 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
NQO2_HUMAN P16083 CHEMBL3959 Quinone reductase 2 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH2_MOUSE Q05769 CHEMBL4321 Cyclooxygenase-2 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
SC6A1_RAT P23978 CHEMBL4054 GABA transporter 1 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
THRB_HUMAN P00734 CHEMBL204 Thrombin 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
TRY1_HUMAN P07477 CHEMBL209 Trypsin I 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
TYRO_AGABI O42713 CHEMBL3318 Tyrosinase 16 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHA5_RAT P20420 CHEMBL4960 Neuronal acetylcholine receptor protein alpha-5 subunit 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHA6_RAT P43143 CHEMBL4747 Neuronal acetylcholine receptor protein alpha-6 subunit 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHA_RAT P25108 CHEMBL3599 Acetylcholine receptor protein alpha chain 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHB3_RAT P12391 CHEMBL4568 Neuronal acetylcholine receptor protein beta-3 subunit 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHB_RAT P25109 CHEMBL2666 Acetylcholine receptor protein beta chain 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB2_BOVIN Q28044 CHEMBL3373 Beta-2 adrenergic receptor 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
CLTR1_HUMAN Q9Y271 CHEMBL1798 Cysteinyl leukotriene receptor 1 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
CP1B1_HUMAN Q16678 CHEMBL4878 Cytochrome P450 1B1 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
KPCG_HUMAN P05129 CHEMBL2938 Protein kinase C gamma 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
KPCL_HUMAN P24723 CHEMBL3616 Protein kinase C eta 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
KPCT_HUMAN Q04759 CHEMBL3920 Protein kinase C theta 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
MC4R_HUMAN P32245 CHEMBL259 Melanocortin receptor 4 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
NEP_HUMAN P08473 CHEMBL1944 Neprilysin 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
NK1R_HUMAN P25103 CHEMBL249 Neurokinin 1 receptor 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
OPRK_MOUSE P33534 CHEMBL4329 Kappa opioid receptor 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
PARP1_HUMAN P09874 CHEMBL3105 Poly [ADP-ribose] polymerase-1 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH1_BOVIN O62664 CHEMBL2860 Cyclooxygenase-1 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH2_SHEEP P79208 CHEMBL4102 Cyclooxygenase-2 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
RXRA_HUMAN P19793 CHEMBL2061 Retinoid X receptor alpha 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
VGFR2_HUMAN P35968 CHEMBL279 Vascular endothelial growth factor receptor 2 15 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACES_BOVIN P23795 CHEMBL4768 Acetylcholinesterase 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADRB3_HUMAN P13945 CHEMBL246 Beta-3 adrenergic receptor 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
CDK2_HUMAN P24941 CHEMBL301 Cyclin-dependent kinase 2 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
CNR1_MOUSE P47746 CHEMBL3037 Cannabinoid CB1 receptor 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
DHSO_HUMAN Q00796 CHEMBL2275 Sorbitol dehydrogenase 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
FABPL_RAT P02692 CHEMBL5738 Fatty acid-binding protein, liver 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
GAK_HUMAN O14976 CHEMBL4355 Serine/threonine-protein kinase GAK 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
GCR_HUMAN P04150 CHEMBL2034 Glucocorticoid receptor 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
HMDH_HUMAN P04035 CHEMBL402 HMG-CoA reductase 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGFRA_HUMAN P16234 CHEMBL2007 Platelet-derived growth factor receptor alpha 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGH2_BOVIN O62698 CHEMBL3331 Cyclooxygenase-2 14 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHA3_HUMAN P32297 CHEMBL3068 Neuronal acetylcholine receptor protein alpha-3 subunit 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHB2_HUMAN P17787 CHEMBL1883 Neuronal acetylcholine receptor protein beta-2 subunit 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADCY2_RAT P26769 CHEMBL2958 Adenylate cyclase type II 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADCY3_RAT P21932 CHEMBL4864 Adenylate cyclase type III 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADCY4_RAT P26770 CHEMBL2879 Adenylate cyclase type IV 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADCY5_RAT Q04400 CHEMBL2880 Adenylate cyclase type V 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADCY6_RAT Q03343 CHEMBL2975 Adenylate cyclase type VI 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
ADCY8_RAT P40146 CHEMBL3082 Adenylate cyclase type VIII 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
CCNB1_HUMAN P14635 CHEMBL2412 G2/mitotic-specific cyclin B1 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
CCNB2_HUMAN O95067 CHEMBL3723 G2/mitotic-specific cyclin B2 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
CCNB3_HUMAN Q8WWL7 CHEMBL3606 G2/mitotic-specific cyclin B3 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
CNR2_MOUSE P47936 CHEMBL5373 Cannabinoid CB2 receptor 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
CP19A_RAT P22443 CHEMBL3859 Cytochrome P450 19A1 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
FAAH1_RAT P97612 CHEMBL3229 Anandamide amidohydrolase 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIK1_RAT P22756 CHEMBL2919 Glutamate receptor ionotropic kainate 1 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIK3_RAT P42264 CHEMBL3744 Glutamate receptor ionotropic kainate 3 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
GSK3A_HUMAN P49840 CHEMBL2850 Glycogen synthase kinase-3 alpha 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
LT4R1_HUMAN Q15722 CHEMBL3911 Leukotriene B4 receptor 1 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
MCHR1_HUMAN Q99705 CHEMBL344 Melanin-concentrating hormone receptor 1 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
MRP1_HUMAN P33527 CHEMBL3004 Multidrug resistance-associated protein 1 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
MYLK_HUMAN Q15746 CHEMBL2428 Myosin light chain kinase, smooth muscle 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
NMDE1_RAT Q00959 CHEMBL310 Glutamate [NMDA] receptor subunit epsilon 1 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
OXGR1_RAT Q6Y1R5 CHEMBL2325 G protein-coupled receptor 80 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDR5_YEAST P33302 CHEMBL1697658 Pleiotropic ABC efflux transporter of multiple drugs 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
PGFRB_HUMAN P09619 CHEMBL1913 Platelet-derived growth factor receptor beta 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
PRGR_HUMAN P06401 CHEMBL208 Progesterone receptor 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
SLK_HUMAN Q9H2G2 CHEMBL4202 Serine/threonine-protein kinase 2 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
TRPA1_HUMAN O75762 CHEMBL6007 Transient receptor potential cation channel subfamily A member 1 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
XDH_HUMAN P47989 CHEMBL1929 Xanthine dehydrogenase 13 Annotations Catalogs SMILES SDF Mol2 Flexibase
5HT2C_MOUSE P34968 CHEMBL3006 Serotonin 2c (5-HT2c) receptor 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
ABCG2_HUMAN Q9UNQ0 CHEMBL5393 ATP-binding cassette sub-family G member 2 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
ABL1_HUMAN P00519 CHEMBL1862 Tyrosine-protein kinase ABL 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHA4_HUMAN P43681 CHEMBL1882 Neuronal acetylcholine receptor protein alpha-4 subunit 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
ANDR_RAT P15207 CHEMBL3072 Androgen Receptor 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
C11B2_HUMAN P19099 CHEMBL2722 Cytochrome P450 11B2 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
CNR2_RAT Q9QZN9 CHEMBL2470 Cannabinoid CB2 receptor 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
CP17A_HUMAN P05093 CHEMBL3522 Cytochrome P450 17A1 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
CTRO_HUMAN O14578 CHEMBL5579 Citron Rho-interacting kinase 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
DYR_MOUSE P00375 CHEMBL4564 Dihydrofolate reductase 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
DYR_RAT Q920D2 CHEMBL2363 Dihydrofolate reductase 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
FDFT_RAT Q02769 CHEMBL3815 Squalene synthetase 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
FKB1A_HUMAN P62942 CHEMBL1902 FK506-binding protein 1A 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
FLT3_HUMAN P36888 CHEMBL1974 Tyrosine-protein kinase receptor FLT3 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
FRK_HUMAN P42685 CHEMBL4223 Tyrosine-protein kinase FRK 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA1_BOVIN P08219 CHEMBL3627 GABA receptor alpha-1 subunit 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA2_BOVIN P10063 CHEMBL2321 GABA receptor alpha-2 subunit 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA3_BOVIN P10064 CHEMBL3628 GABA receptor alpha-3 subunit 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA4_BOVIN P20237 CHEMBL3140 GABA receptor alpha-4 subunit 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRG1_RAT P23574 CHEMBL296 GABA receptor gamma-1 subunit 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIA1_RAT P19490 CHEMBL3753 Glutamate receptor ionotropic, AMPA 1 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIK2_RAT P42260 CHEMBL3607 Glutamate receptor ionotropic kainate 2 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
KPCD1_HUMAN Q15139 CHEMBL3863 Protein kinase C mu 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
KPCD3_HUMAN O94806 CHEMBL2595 Protein kinase C nu 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
KPCG_RAT P63319 CHEMBL3604 Protein kinase C gamma 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
MCR_HUMAN P08235 CHEMBL1994 Mineralocorticoid receptor 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
MMP2_HUMAN P08253 CHEMBL333 Matrix metalloproteinase-2 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
O77823_PIG O77823 CHEMBL3333 Phosphodiesterase 4A 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE1A_HUMAN P54750 CHEMBL3421 Phosphodiesterase 1A 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE1B_HUMAN Q01064 CHEMBL4425 Phosphodiesterase 1B 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE1C_HUMAN Q14123 CHEMBL4619 Phosphodiesterase 1C 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
PDE5A_HUMAN O76074 CHEMBL1827 Phosphodiesterase 5A 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
Q965D5_PLAFA Q965D5 CHEMBL4150 Enoyl-acyl-carrier protein reductase 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
TSPO_RAT P16257 CHEMBL4552 Peripheral-type benzodiazepine receptor 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
VMAT2_RAT Q01827 CHEMBL4828 Synaptic vesicular amine transporter 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
Z104288 Z104288 CHEMBL1907594 Neuronal acetylcholine receptor; alpha3/beta4 12 Annotations Catalogs SMILES SDF Mol2 Flexibase
A3EZI9_9HEPC A3EZI9 CHEMBL4893 Hepatitis C virus NS3 protease/helicase 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
AA2AR_CAVPO P46616 CHEMBL2605 Adenosine A2a receptor 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
ACHA_TORCA P02710 CHEMBL3097 Acetylcholine receptor protein alpha chain 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH5A_MOUSE P23589 CHEMBL2330 Carbonic anhydrase VA 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH5B_MOUSE Q9QZA0 CHEMBL4634 Carbonic anhydrase VB 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
CAH_METTE P40881 CHEMBL3932 Carbonic anhydrase 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
DDR1_HUMAN Q08345 CHEMBL5319 Epithelial discoidin domain-containing receptor 1 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
DRTS_TOXGO Q07422 CHEMBL2425 Dihydrofolate reductase 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
DYR_LACCA P00381 CHEMBL2902 Dihydrofolate reductase 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
ESR1_RAT P06211 CHEMBL2724 Estrogen receptor alpha 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
ESR2_RAT Q62986 CHEMBL3021 Estrogen receptor beta 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
GABR1_RAT Q9Z0U4 CHEMBL2753 GABA-B receptor 1 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
GABR2_RAT O88871 CHEMBL4686 GABA-B receptor 2 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA3_RAT P20236 CHEMBL328 GABA receptor alpha-3 subunit 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRA5_RAT P19969 CHEMBL300 GABA receptor alpha-5 subunit 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
GBRB3_RAT P63079 CHEMBL316 GABA receptor beta-3 subunit 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIA4_HUMAN P48058 CHEMBL3190 Glutamate receptor ionotropic, AMPA 4 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIK4_RAT Q01812 CHEMBL3044 Glutamate receptor ionotropic kainate 4 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRIK5_RAT Q63273 CHEMBL4041 Glutamate receptor ionotropic kainate 5 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
GRM2_HUMAN Q14416 CHEMBL5137 Metabotropic glutamate receptor 2 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
HDAC1_HUMAN Q13547 CHEMBL325 Histone deacetylase 1 11 Annotations Catalogs SMILES SDF Mol2 Flexibase
KC1D_HUMAN P48730 CHEMBL2828 Casein kinase I delta 11